BRPI0719956A2 - Radiofluoração - Google Patents

Radiofluoração

Info

Publication number: BRPI0719956A2
Authority: BR; Brazil
Prior art keywords: radiofluoration
Prior art date: 2006-10-02

Application number

BRPI0719956-2A2A

Other languages

English (en)

Inventor

Ananth Srinivasan

Ulrike Roehn

Timo Stellfeld

Simon Ametamey

Ulrich Klar

Aileen Hoehne

Linjing Mu

Lutz Lehmann

Original Assignee

Bayer Schering Pharma Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2006-10-02

Filing date

2007-09-07

Publication date

2014-04-29

2006-10-02 Priority claimed from EP06076823A external-priority patent/EP1908472A1/en

2006-10-11 Priority claimed from EP06076869A external-priority patent/EP1911452A1/en

2007-03-12 Priority claimed from EP07090043A external-priority patent/EP1970064A1/en

2007-04-23 Priority claimed from EP07090079A external-priority patent/EP1985624A3/en

2007-09-07 Application filed by Bayer Schering Pharma Ag filed Critical Bayer Schering Pharma Ag

2014-04-29 Publication of BRPI0719956A2 publication Critical patent/BRPI0719956A2/pt

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/13—Labelling of peptides
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/695—Silicon compounds
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K49/00—Preparations for testing in vivo
- A61K49/06—Nuclear magnetic resonance [NMR] contrast preparations; Magnetic resonance imaging [MRI] contrast preparations
- A61K49/08—Nuclear magnetic resonance [NMR] contrast preparations; Magnetic resonance imaging [MRI] contrast preparations characterised by the carrier
- A61K49/085—Nuclear magnetic resonance [NMR] contrast preparations; Magnetic resonance imaging [MRI] contrast preparations characterised by the carrier conjugated systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K49/00—Preparations for testing in vivo
- A61K49/06—Nuclear magnetic resonance [NMR] contrast preparations; Magnetic resonance imaging [MRI] contrast preparations
- A61K49/08—Nuclear magnetic resonance [NMR] contrast preparations; Magnetic resonance imaging [MRI] contrast preparations characterised by the carrier
- A61K49/10—Organic compounds
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K49/00—Preparations for testing in vivo
- A61K49/06—Nuclear magnetic resonance [NMR] contrast preparations; Magnetic resonance imaging [MRI] contrast preparations
- A61K49/08—Nuclear magnetic resonance [NMR] contrast preparations; Magnetic resonance imaging [MRI] contrast preparations characterised by the carrier
- A61K49/10—Organic compounds
- A61K49/14—Peptides, e.g. proteins
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
- A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
- A61K51/04—Organic compounds
- A61K51/0491—Sugars, nucleosides, nucleotides, oligonucleotides, nucleic acids, e.g. DNA, RNA, nucleic acid aptamers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B59/00—Introduction of isotopes of elements into organic compounds ; Labelled organic compounds per se
- C07B59/004—Acyclic, carbocyclic or heterocyclic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen, sulfur, selenium or tellurium
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B59/00—Introduction of isotopes of elements into organic compounds ; Labelled organic compounds per se
- C07B59/008—Peptides; Proteins
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/0834—Compounds having one or more O-Si linkage
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/0896—Compounds with a Si-H linkage
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/12—Organo silicon halides
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/02—Linear peptides containing at least one abnormal peptide link
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/08—Linear peptides containing only normal peptide links having 12 to 20 amino acids
- C07K7/086—Bombesin; Related peptides

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Biochemistry (AREA)
Epidemiology (AREA)
Molecular Biology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Genetics & Genomics (AREA)
Biophysics (AREA)
Radiology & Medical Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Analytical Chemistry (AREA)
Physics & Mathematics (AREA)
Optics & Photonics (AREA)
Biotechnology (AREA)
Engineering & Computer Science (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Nuclear Medicine (AREA)
Peptides Or Proteins (AREA)

BRPI0719956-2A2A 2006-10-02 2007-09-07 Radiofluoração BRPI0719956A2 (pt)

Applications Claiming Priority (5)

Application Number	Priority Date	Filing Date	Title
EP06076823A EP1908472A1 (en)	2006-10-02	2006-10-02	Silicon derivatives for PET imaging
EP06076869A EP1911452A1 (en)	2006-10-11	2006-10-11	Silicon-derivates for PET-Imaging
EP07090043A EP1970064A1 (en)	2007-03-12	2007-03-12	Silicon-derivatives for pet-imaging
EP07090079A EP1985624A3 (en)	2007-04-23	2007-04-23	Single step method of radiofluorination of biologically active compounds or biomolecules
PCT/EP2007/008044 WO2008040441A2 (en)	2006-10-02	2007-09-07	Silicon derivatives for pet imaging

Publications (1)

Publication Number	Publication Date
BRPI0719956A2 true BRPI0719956A2 (pt)	2014-04-29

Family

ID=39030886

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BRPI0719956-2A2A BRPI0719956A2 (pt)	2006-10-02	2007-09-07	Radiofluoração

Country Status (21)

Country	Link
US (1)	US20090035215A1 (pt)
EP (1)	EP2074135A2 (pt)
JP (1)	JP2010505776A (pt)
KR (1)	KR20090085599A (pt)
AR (1)	AR062795A1 (pt)
AU (1)	AU2007304508A1 (pt)
BR (1)	BRPI0719956A2 (pt)
CA (1)	CA2664700A1 (pt)
CO (1)	CO6180444A2 (pt)
CR (1)	CR10703A (pt)
IL (1)	IL197817A0 (pt)
MA (1)	MA30824B1 (pt)
MX (1)	MX2009003617A (pt)
NO (1)	NO20091735L (pt)
PA (1)	PA8747601A1 (pt)
PE (1)	PE20081173A1 (pt)
SV (1)	SV2009003205A (pt)
TN (1)	TN2009000100A1 (pt)
TW (1)	TW200820988A (pt)
UY (1)	UY30596A1 (pt)
WO (1)	WO2008040441A2 (pt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US9285360B2 (en)	2010-01-25	2016-03-15	Institut National De La Sante Et De La Recherche Medicale (Inserm)	Silylated biomolecules
JP5717138B2 (ja) *	2011-05-23	2015-05-13	独立行政法人産業技術総合研究所	タンパク質固定化表面修飾材料
KR102344233B1 (ko) *	2013-06-06	2021-12-27	닛산 가가쿠 가부시키가이샤	액정 배향제, 액정 배향막 및 액정 표시 소자
EP3303349B1 (en)	2015-05-26	2022-07-06	The Regents of the University of California	Novel heteroaromatic silicon-fluoride-acceptors useful for 18f labeling of molecules and biomolecules, and methods of preparing same
WO2019055825A1 (en)	2017-09-15	2019-03-21	The Regents Of The University Of California	INHIBITION OF AMINOACYLASE 3 (AA3) IN THE TREATMENT OF CANCER
US20230226228A1 (en) *	2020-05-04	2023-07-20	The Research Foundation For The State University Of New York	Positron imaging tomography imaging agent composition and method for detection of bacterial infection
CN116075344B (zh) *	2020-09-28	2025-07-15	国立研究开发法人量子科学技术研究开发机构	放射性标识物的制造方法、放射性标识物的制造装置以及放射性金属核素的蒸发浓缩方法

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5084555A (en) *	1989-08-21	1992-01-28	The Administrators Of The Tulane Educational Fund	An octapeptide bombesin analog
US5732578A (en) *	1995-02-24	1998-03-31	Hyundai Metal Co., Ltd.	Device for maintaining the horizontality of a door lock lever
TW432073B (en) *	1995-12-28	2001-05-01	Pfizer	Pyrazolopyridine compounds
US6639076B1 (en) *	1998-08-18	2003-10-28	Eli Lilly And Company	Growth hormone secretagogues
CA2375920A1 (en) *	1999-06-14	2000-12-21	Eli Lilly And Company	Compounds
US7115766B2 (en) *	2000-11-30	2006-10-03	Indiana University Research & Technology Corp.	Nucleophilic approach for preparing radiolabeled imaging agents and associated compounds
GB0206750D0 (en) *	2002-03-22	2002-05-01	Amersham Plc	Radiofluorination methods
US7342095B2 (en) *	2003-02-20	2008-03-11	University Of South Florida	Peptidomimetic inhibitors of STAT activity and uses thereof
GB0305704D0 (en) *	2003-03-13	2003-04-16	Amersham Plc	Radiofluorination methods
WO2005077967A1 (en) *	2004-02-13	2005-08-25	The University Of British Columbia	Radiolabeled compounds and compositions, their precursors and methods for their production
US20080029548A1 (en) *	2006-05-05	2008-02-07	Ann De Wree	Fabric treatment dispensing package

2007
- 2007-09-07 KR KR1020097009044A patent/KR20090085599A/ko not_active Withdrawn
- 2007-09-07 EP EP07818173A patent/EP2074135A2/en not_active Withdrawn
- 2007-09-07 BR BRPI0719956-2A2A patent/BRPI0719956A2/pt not_active IP Right Cessation
- 2007-09-07 CA CA002664700A patent/CA2664700A1/en not_active Abandoned
- 2007-09-07 WO PCT/EP2007/008044 patent/WO2008040441A2/en not_active Ceased
- 2007-09-07 MX MX2009003617A patent/MX2009003617A/es not_active Application Discontinuation
- 2007-09-07 US US11/851,936 patent/US20090035215A1/en not_active Abandoned
- 2007-09-07 JP JP2009530773A patent/JP2010505776A/ja active Pending
- 2007-09-07 AU AU2007304508A patent/AU2007304508A1/en not_active Abandoned
- 2007-09-10 TW TW096133834A patent/TW200820988A/zh unknown
- 2007-09-14 PA PA20078747601A patent/PA8747601A1/es unknown
- 2007-09-14 AR ARP070104086A patent/AR062795A1/es unknown
- 2007-09-14 UY UY30596A patent/UY30596A1/es not_active Application Discontinuation
- 2007-09-14 PE PE2007001246A patent/PE20081173A1/es not_active Application Discontinuation
2009
- 2009-03-25 TN TN2009000100A patent/TN2009000100A1/fr unknown
- 2009-03-26 IL IL197817A patent/IL197817A0/en unknown
- 2009-04-01 CR CR10703A patent/CR10703A/es not_active Application Discontinuation
- 2009-04-02 SV SV2009003205A patent/SV2009003205A/es not_active Application Discontinuation
- 2009-04-02 CO CO09034043A patent/CO6180444A2/es not_active Application Discontinuation
- 2009-04-30 NO NO20091735A patent/NO20091735L/no not_active Application Discontinuation
- 2009-04-30 MA MA31834A patent/MA30824B1/fr unknown

Also Published As

Publication number	Publication date
US20090035215A1 (en)	2009-02-05
MA30824B1 (fr)	2009-10-01
MX2009003617A (es)	2009-04-22
SV2009003205A (es)	2009-10-19
NO20091735L (no)	2009-06-30
PE20081173A1 (es)	2008-11-06
CA2664700A1 (en)	2008-04-10
WO2008040441A2 (en)	2008-04-10
IL197817A0 (en)	2009-12-24
JP2010505776A (ja)	2010-02-25
CO6180444A2 (es)	2010-07-19
TN2009000100A1 (en)	2010-08-19
AU2007304508A8 (en)	2009-05-14
TW200820988A (en)	2008-05-16
EP2074135A2 (en)	2009-07-01
PA8747601A1 (es)	2009-08-26
KR20090085599A (ko)	2009-08-07
UY30596A1 (es)	2008-05-02
CR10703A (es)	2009-06-25
AR062795A1 (es)	2008-12-03
WO2008040441A3 (en)	2009-01-08
AU2007304508A1 (en)	2008-04-10

Legal Events

Date	Code	Title	Description
2014-08-26	B08L	Patent application lapsed because of non payment of annual fee [chapter 8.12 patent gazette]	Free format text: REFERENTE AO NAO RECOLHIMENTO DAS 5A, 6A E 7A ANUIDADES.
2020-11-10	B08I	Publication cancelled [chapter 8.9 patent gazette]	Free format text: ANULADA A PUBLICACAO CODIGO 8.12 NA RPI NO 2277 DE 26/08/2014 POR TER SIDO INDEVIDA.
2020-11-17	B08F	Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]	Free format text: REFERENTE AS 5A, 6A, 7A, 8A, 9A, 10A, 11A, 12A E 13A ANUIDADES.
2021-03-09	B08K	Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]	Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2602 DE 17-11-2020 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.

Publication	Publication Date	Title
DE602006019782D1 (de)	2011-03-03	Kapselperforationsmodul
DE602007008423D1 (de)	2010-09-23	Flüssigkeitshärtung
DE602007009267D1 (de)	2010-10-28	Reifenaufblasverfahren
ATE546437T1 (de)	2012-03-15	Aminomethyl-4-imidazole
DE502007000218D1 (de)	2008-12-18	nsetzungen
DE112007003147A5 (de)	2009-09-24	Rohr-Biegevorrichtung
FI20061014A0 (fi)	2006-11-17	Diffuusiopinnoitusmenetelmä
DE602007012951D1 (de)	2011-04-21	Verbundschraubenausräumtür
DE502007005975D1 (de)	2011-01-27	Wischblatt
NO20065996L (no)	2008-06-23	SmartPacker
FI20060691A0 (fi)	2006-07-19	Laitekotelointi
ITPD20060387A1 (it)	2008-04-20	Espositore
DE112007001125A5 (de)	2009-02-05	Käfigmutter
NO20065028L (no)	2008-05-05	Limkobling
NO20060756L (no)	2007-08-17	Transportsystem
ITMI20062042A1 (it)	2008-04-25	Elettrovalvola
SE0700923L (sv)	2008-05-10	Halogenhårtork
FR2896376B1 (fr)	2010-03-26	Desherbeuse-emietteuse
FI7437U1 (fi)	2007-03-09	Katafalkki
FI7169U1 (fi)	2006-07-28	Paalileikkuri
FI7353U1 (fi)	2007-01-12	Riipukeläpivienti
FI7355U1 (fi)	2007-01-12	Esiintymislava
FI7243U1 (fi)	2006-10-18	Hiirenpyydys
ES1064558Y (es)	2007-07-01	Salva-tendedero
FI7103U1 (fi)	2006-06-08	Pyrstömormuska