BRPI0812054A2 - Processo para preparar compostos, e, compostos. - Google Patents

Processo para preparar compostos, e, compostos.

Info

Publication number
BRPI0812054A2
BRPI0812054A2 BRPI0812054-4A2A BRPI0812054A BRPI0812054A2 BR PI0812054 A2 BRPI0812054 A2 BR PI0812054A2 BR PI0812054 A BRPI0812054 A BR PI0812054A BR PI0812054 A2 BRPI0812054 A2 BR PI0812054A2
Authority
BR
Brazil
Prior art keywords
compounds
preparing
preparing compounds
Prior art date
Application number
BRPI0812054-4A2A
Other languages
English (en)
Inventor
Thomas Zierke
Joachim Rheinheimer
Michael Rack
Sebastian Peer Smidt
Ansgar Gereon Altenhoff
Joachim Schmidt-Leithoff
Nina Challand
Original Assignee
Basf Se
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Se filed Critical Basf Se
Publication of BRPI0812054A2 publication Critical patent/BRPI0812054A2/pt
Publication of BRPI0812054B1 publication Critical patent/BRPI0812054B1/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Catalysts (AREA)
BRPI0812054A 2007-06-01 2008-05-30 processo de preparação de (3-di-halometilpirazol-4-il) carboxamidas n-substituídas BRPI0812054B1 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP07109463 2007-06-01
PCT/EP2008/056712 WO2008145740A1 (de) 2007-06-01 2008-05-30 Verfahren zur herstellung n-substituierter (3-dihalomethyl-1-methyl-pyrazol-4-yl)carboxamide

Publications (2)

Publication Number Publication Date
BRPI0812054A2 true BRPI0812054A2 (pt) 2014-11-18
BRPI0812054B1 BRPI0812054B1 (pt) 2015-12-29

Family

ID=38728715

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0812054A BRPI0812054B1 (pt) 2007-06-01 2008-05-30 processo de preparação de (3-di-halometilpirazol-4-il) carboxamidas n-substituídas

Country Status (19)

Country Link
US (1) US8153820B2 (pt)
EP (1) EP2164831B1 (pt)
JP (1) JP5456663B2 (pt)
KR (1) KR101517254B1 (pt)
CN (1) CN101679282B (pt)
AR (1) AR066802A1 (pt)
AU (1) AU2008257515B2 (pt)
BR (1) BRPI0812054B1 (pt)
CA (1) CA2686659A1 (pt)
DK (1) DK2164831T3 (pt)
EA (1) EA016615B1 (pt)
ES (1) ES2431341T3 (pt)
IL (1) IL201940A (pt)
MX (1) MX2009012020A (pt)
PL (1) PL2164831T3 (pt)
SI (1) SI2164831T1 (pt)
UA (1) UA99460C2 (pt)
WO (1) WO2008145740A1 (pt)
ZA (1) ZA200909030B (pt)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5456663B2 (ja) 2007-06-01 2014-04-02 ビーエーエスエフ ソシエタス・ヨーロピア N−置換(3−ジハロメチル−1−メチル−ピラゾール−4−イル)カルボキサミドの製造方法
AU2008263883B2 (en) 2007-06-15 2014-03-13 Basf Se Method for producing difluoromethyl-substituted pyrazole compounds
EP2008996A1 (en) * 2007-06-27 2008-12-31 Syngeta Participations AG Process for the production of pyrazoles
WO2009007344A1 (en) * 2007-07-12 2009-01-15 Basf Se Novel crystalline form of 3-(difluormethyl)-1-methyl-n -(3',4',5'-trifluor[1,1'-biphenyl]-2-yl)-1h-pyrazol-4-carboxamide
DE102008015773A1 (de) * 2008-03-26 2009-10-01 Albert-Ludwigs-Universität Freiburg Verfahren zur decarboxylativen Hydroformylierung alpha,beta-ungesättigter Carbonsäuren
JP5602131B2 (ja) 2008-05-02 2014-10-08 ビーエーエスエフ ソシエタス・ヨーロピア ハロゲン置換2−(アミノメチリデン)−3−オキソ酪酸エステルの製造方法
BRPI0911898A2 (pt) * 2008-05-02 2015-10-13 Basf Se processo para preparar compostos, e, composto.
US8598222B2 (en) * 2008-05-05 2013-12-03 Basf Se Method for preparing 1,3,4-substituted pyrazol compounds
US8703992B2 (en) 2008-05-27 2014-04-22 Basf Se Method for producing aromatic and heteroaromatic carboxylic acids, carboxylic acid esters and carboxylic acid amides
EP2307384B1 (en) 2008-07-21 2012-04-25 Basf Se Process for preparing 1,3-disubstituted pyrazolecarboxylic esters
US8853410B2 (en) 2009-04-30 2014-10-07 Basf Se Process for preparing substituted isoxazoline compounds and their precursors
CN102596912B (zh) * 2009-11-05 2015-08-12 巴斯夫欧洲公司 制备1,3-二取代吡唑化合物的方法
BR112012032496A2 (pt) 2010-06-23 2015-09-15 Basf Se processos para produzir um composto de carbonila da fórmula i e de imina da fórmula iii, compostos de imina da fórmula (iii), composições agrícolas e veterinária, uso de um composto de imina da fórmula iii e material de propagação de planta
CN103282345A (zh) 2010-11-03 2013-09-04 巴斯夫欧洲公司 制备取代的异噁唑啉化合物及其前体4-氯-、4-溴-或4-碘苯甲醛肟的方法
US20130338369A1 (en) 2011-03-07 2013-12-19 Basf Se Process for the Synthesis of Aminobiphenylene
EP2546229A1 (de) 2011-07-15 2013-01-16 Friedrich-Alexander-Universität Erlangen-Nürnberg Verfahren zur Synthese von Aminobiphenylen
BR112013032988A2 (pt) 2011-06-21 2016-08-16 Bayer Ip Gmbh método para a produção de pirazolilcarboxanilidas
CN102516016A (zh) * 2011-10-31 2012-06-27 滨海康杰化学有限公司 一溴二氟甲基苯类化合物或三氟甲苯类化合物的制备方法
CA2855904C (en) 2011-11-24 2021-01-19 Weldobot Ltd. System and method for modular portable welding and seam tracking
CN104220417B (zh) 2012-03-07 2017-10-13 巴斯夫欧洲公司 使用芳基肼合成氨基联苯类的方法
DK2885277T3 (en) * 2012-07-19 2016-12-12 Bayer Cropscience Ag PROCESS FOR THE PREPARATION OF 5-FLUORO-1H-pyrazoles
ES2607807T3 (es) * 2012-08-07 2017-04-04 Janssen Pharmaceutica Nv Procedimiento para la preparación de los inibidores de las quinasas c-fms
EP3046908B1 (en) * 2013-09-20 2017-08-16 Bayer CropScience Aktiengesellschaft Process for preparing 5-fluoro-1-alkyl-3-fluoroalkyl-1h-pyrazole-4-carbaldehyde
BR112016021563B1 (pt) 2014-03-20 2021-12-21 Mitsui Chemicals Agro, Inc Composição para o controle de doença de pantas e método para controlar doença de plantas por aplicação da mesma
EP3178813A1 (en) 2015-12-09 2017-06-14 Basf Se Method for preparing halogenated 3-oxocarboxylates carrying a 2-alkoxymethylidene or a 2-dialkylaminomethylidene group
US11591312B2 (en) * 2018-01-23 2023-02-28 Basf Se Halogenation of pyridine derivatives
CN109369533A (zh) * 2018-12-26 2019-02-22 浙江本立科技股份有限公司 3-二氟甲基-1-甲基-吡啶-4-羰酰氯的制备方法
CN111303035A (zh) * 2020-03-18 2020-06-19 徐州圣元化工有限公司 一种3-(二氟甲基)-1-甲基-1h-吡唑-4-羧酸的制备方法
WO2021219424A1 (en) * 2020-04-29 2021-11-04 Basf Se Preparation of aromatic carboxyamides by a palladium-catalyzed carbonylation reaction
KR102812263B1 (ko) * 2022-03-17 2025-05-26 솔브레인 주식회사 디플루오로인산염의 제조방법

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Publication number Priority date Publication date Assignee Title
JPS5946273A (ja) 1982-08-31 1984-03-15 Daikin Ind Ltd 含フツ素ヘテロ環化合物の製造方法
DE3934924C2 (de) * 1989-10-20 1994-01-27 Huels Chemische Werke Ag Verfahren zur Herstellung von 4-Alkoxycarbonyl-3-chlormethyl-2H-pyrazolen
US5093347A (en) 1991-01-28 1992-03-03 Monsanto Company 3-difluoromethylpyrazolecarboxamide fungicides, compositions and use
US5223526A (en) 1991-12-06 1993-06-29 Monsanto Company Pyrazole carboxanilide fungicides and use
JPH07196637A (ja) * 1993-11-24 1995-08-01 Mitsui Toatsu Chem Inc イソチアゾールカルボン酸アミド誘導体の製造法
DE10215292A1 (de) * 2002-02-19 2003-08-28 Bayer Cropscience Ag Disubstitutierte Pyrazolylcarbocanilide
DK1599742T3 (da) * 2003-02-25 2009-07-27 Oticon As Fremgangsmåde til detektering af en taleaktivitet i en kommunikationsanordning
DE10331496A1 (de) 2003-07-01 2005-01-27 Bayer Cropscience Ag Verfahren zum Herstellen von Difluoracetessigsäurealkylestern
DE10349500A1 (de) 2003-10-23 2005-06-02 Bayer Cropscience Ag Verfahren zum Herstellen von 2-Dihalogenacyl-3-amino-acrylsäureestern und 3-Dihalogenmethyl-pyrazol-4-carbonsäureestern
DE10351088A1 (de) * 2003-10-31 2005-06-02 Bayer Cropscience Gmbh Verfahren zum Herstellen von fluormethyl-substituierten Heterocyclen
CN101962364B (zh) 2005-09-16 2013-01-09 先正达参股股份有限公司 酰胺的制备方法
TW200732320A (en) * 2005-10-31 2007-09-01 Biolipox Ab Pyrazoles useful in the treatment of inflammation
DE102006039909A1 (de) 2006-08-25 2008-03-13 Bayer Cropscience Ag Verfahren zum Herstellen von 3-Dihalomethyl-pyrazol-4-carbonsäurederivaten
UA97498C2 (ru) * 2006-11-03 2012-02-27 Басф Се Способ получения дифторметилпиразолилкарбоксилатов
MX2009005863A (es) * 2006-12-21 2009-06-12 Basf Se Procedimiento para la preparacion de compuestos heterociclicos sustituidos por fluorometilo.
JP5456663B2 (ja) 2007-06-01 2014-04-02 ビーエーエスエフ ソシエタス・ヨーロピア N−置換(3−ジハロメチル−1−メチル−ピラゾール−4−イル)カルボキサミドの製造方法
AU2008263883B2 (en) 2007-06-15 2014-03-13 Basf Se Method for producing difluoromethyl-substituted pyrazole compounds

Also Published As

Publication number Publication date
ZA200909030B (en) 2011-04-28
IL201940A0 (en) 2010-06-16
CN101679282A (zh) 2010-03-24
KR20100021628A (ko) 2010-02-25
CA2686659A1 (en) 2008-12-04
EP2164831B1 (de) 2013-07-17
AR066802A1 (es) 2009-09-16
JP2010529006A (ja) 2010-08-26
DK2164831T3 (da) 2013-10-14
IL201940A (en) 2014-07-31
JP5456663B2 (ja) 2014-04-02
SI2164831T1 (sl) 2013-09-30
CN101679282B (zh) 2012-11-28
US20100174094A1 (en) 2010-07-08
EA016615B1 (ru) 2012-06-29
PL2164831T3 (pl) 2013-12-31
UA99460C2 (ru) 2012-08-27
KR101517254B1 (ko) 2015-04-30
AU2008257515A1 (en) 2008-12-04
WO2008145740A1 (de) 2008-12-04
US8153820B2 (en) 2012-04-10
MX2009012020A (es) 2009-11-18
EA200901600A1 (ru) 2010-06-30
ES2431341T3 (es) 2013-11-26
BRPI0812054B1 (pt) 2015-12-29
EP2164831A1 (de) 2010-03-24
AU2008257515B2 (en) 2014-01-23

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Legal Events

Date Code Title Description
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 30/05/2008, OBSERVADAS AS CONDICOES LEGAIS.