BRPI0814210A2 - Profármacos aminoacila como susbstância ativa farmacêutica para doenças tromboebólicas. - Google Patents

Profármacos aminoacila como susbstância ativa farmacêutica para doenças tromboebólicas.

Info

Publication number
BRPI0814210A2
BRPI0814210A2 BRPI0814210-6A2A BRPI0814210A BRPI0814210A2 BR PI0814210 A2 BRPI0814210 A2 BR PI0814210A2 BR PI0814210 A BRPI0814210 A BR PI0814210A BR PI0814210 A2 BRPI0814210 A2 BR PI0814210A2
Authority
BR
Brazil
Prior art keywords
thromboebolic
propharmaces
aminoacyl
diseases
active substance
Prior art date
Application number
BRPI0814210-6A2A
Other languages
English (en)
Inventor
Hans-Georg Lerchen
Ursula Krenz
Michael Haerter
Mark Jean Gnoth
Georges Von Degenfeld
Elke Dittrich-Wengenroth
Anja Buchmueller
Susanne Roehrig
Swen Allerheiligen
Elisabeth Perzborn
Christoph Gerdes
Karl-Heinz Schlemmer
Metin Ankaba
Original Assignee
Bayer Schering Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Schering Pharma Ag filed Critical Bayer Schering Pharma Ag
Publication of BRPI0814210A2 publication Critical patent/BRPI0814210A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
BRPI0814210-6A2A 2007-07-11 2008-06-28 Profármacos aminoacila como susbstância ativa farmacêutica para doenças tromboebólicas. BRPI0814210A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102007032345A DE102007032345A1 (de) 2007-07-11 2007-07-11 Aminoacyl-Prodrugs
PCT/EP2008/005303 WO2009007027A1 (de) 2007-07-11 2008-06-28 Aminoacyl-prodrugs als arzneimittelwirkstoff für thromboembolische erkrankungen

Publications (1)

Publication Number Publication Date
BRPI0814210A2 true BRPI0814210A2 (pt) 2015-01-27

Family

ID=39789505

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0814210-6A2A BRPI0814210A2 (pt) 2007-07-11 2008-06-28 Profármacos aminoacila como susbstância ativa farmacêutica para doenças tromboebólicas.

Country Status (12)

Country Link
US (1) US20110172232A1 (pt)
EP (1) EP2167500A1 (pt)
JP (1) JP2010532771A (pt)
KR (1) KR20100031535A (pt)
CN (1) CN101730695A (pt)
AU (1) AU2008274578A1 (pt)
BR (1) BRPI0814210A2 (pt)
CA (1) CA2693507A1 (pt)
DE (1) DE102007032345A1 (pt)
IL (1) IL202488A0 (pt)
RU (1) RU2010104475A (pt)
WO (1) WO2009007027A1 (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102007028320A1 (de) * 2007-06-20 2008-12-24 Bayer Healthcare Ag Substituierte Oxazolidinone und ihre Verwendung
US7816355B1 (en) * 2009-04-28 2010-10-19 Apotex Pharmachem Inc Processes for the preparation of rivaroxaban and intermediates thereof
CN102796092B (zh) * 2011-05-24 2015-04-08 北大方正集团有限公司 噁唑烷酮衍生物及其制备方法和应用
EP2838897A1 (en) * 2012-04-16 2015-02-25 Ranbaxy Laboratories Limited Process for the preparation of rivaroxaban and intermediates thereof
CN104193739A (zh) * 2014-09-11 2014-12-10 北京诺泓医药科技有限公司 一种利伐沙班的制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE248835T1 (de) 1999-06-25 2003-09-15 Vertex Pharma Prodrugs von impdh-inhibierenden carbamaten
US7049443B2 (en) 2001-07-12 2006-05-23 Pharmacia & Upjohn Company Amide-containing compound having improved solubility and method of improving the solubility of an amide-containing compound
DE10300111A1 (de) 2003-01-07 2004-07-15 Bayer Healthcare Ag Verfahren zur Herstellung von 5-Chlor-N-({(5S)-2-oxo-3-[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidin-5-yl}-methyl)-2-thiophencarboxamid
US7265140B2 (en) 2003-09-23 2007-09-04 Pfizer Inc Acyloxymethylcarbamate prodrugs of oxazolidinones
DE102006007146A1 (de) * 2006-02-16 2007-08-23 Bayer Healthcare Ag Aminoacyl-Prodrugs

Also Published As

Publication number Publication date
RU2010104475A (ru) 2011-08-20
KR20100031535A (ko) 2010-03-22
DE102007032345A1 (de) 2009-01-15
CN101730695A (zh) 2010-06-09
IL202488A0 (en) 2010-06-30
JP2010532771A (ja) 2010-10-14
WO2009007027A1 (de) 2009-01-15
US20110172232A1 (en) 2011-07-14
AU2008274578A1 (en) 2009-01-15
EP2167500A1 (de) 2010-03-31
CA2693507A1 (en) 2009-01-15

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Legal Events

Date Code Title Description
B11A Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing
B11Y Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette]