BRPI0914918A2 - forma de dosagem farmacêutica, e, método para preparar uma forma de dosagem sólida. - Google Patents

forma de dosagem farmacêutica, e, método para preparar uma forma de dosagem sólida.

Info

Publication number
BRPI0914918A2
BRPI0914918A2 BRPI0914918A BRPI0914918A BRPI0914918A2 BR PI0914918 A2 BRPI0914918 A2 BR PI0914918A2 BR PI0914918 A BRPI0914918 A BR PI0914918A BR PI0914918 A BRPI0914918 A BR PI0914918A BR PI0914918 A2 BRPI0914918 A2 BR PI0914918A2
Authority
BR
Brazil
Prior art keywords
dosage form
preparing
solid dosage
pharmaceutical dosage
pharmaceutical
Prior art date
Application number
BRPI0914918A
Other languages
English (en)
Inventor
Bernd Liepold
Claudia Packhäuser
Jörg Breitenbach
Markus Mägerlein
Thomas Kessler
Original Assignee
Abbott Gmbh & Co Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Gmbh & Co Kg filed Critical Abbott Gmbh & Co Kg
Publication of BRPI0914918A2 publication Critical patent/BRPI0914918A2/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/32—Macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. carbomers, poly(meth)acrylates, or polyvinyl pyrrolidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2095—Tabletting processes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Inorganic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Pain & Pain Management (AREA)
  • Communicable Diseases (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Diabetes (AREA)
  • Biomedical Technology (AREA)
  • Oncology (AREA)
  • Endocrinology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BRPI0914918A 2008-06-30 2009-06-30 forma de dosagem farmacêutica, e, método para preparar uma forma de dosagem sólida. BRPI0914918A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP08159367A EP2140861A1 (en) 2008-06-30 2008-06-30 Pharmaceutical dosage form comprising polymeric carrier composition
PCT/EP2009/058187 WO2010000740A1 (en) 2008-06-30 2009-06-30 Pharmaceutical dosage form comprising polymeric carrier composition

Publications (1)

Publication Number Publication Date
BRPI0914918A2 true BRPI0914918A2 (pt) 2015-10-20

Family

ID=40263268

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0914918A BRPI0914918A2 (pt) 2008-06-30 2009-06-30 forma de dosagem farmacêutica, e, método para preparar uma forma de dosagem sólida.

Country Status (11)

Country Link
US (2) US20110182891A1 (pt)
EP (2) EP2140861A1 (pt)
JP (2) JP5717628B2 (pt)
KR (1) KR101812508B1 (pt)
CN (1) CN102083420B (pt)
AU (1) AU2009265737B2 (pt)
BR (1) BRPI0914918A2 (pt)
CA (1) CA2729148C (pt)
ES (1) ES2699075T3 (pt)
RU (1) RU2519679C9 (pt)
WO (1) WO2010000740A1 (pt)

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EP2140861A1 (en) * 2008-06-30 2010-01-06 Abbott GmbH & Co. KG Pharmaceutical dosage form comprising polymeric carrier composition
US20110160168A1 (en) 2009-12-31 2011-06-30 Differential Drug Development Associates, Llc Modulation of solubility, stability, absorption, metabolism, and pharmacokinetic profile of lipophilic drugs by sterols
WO2012085236A1 (en) * 2010-12-23 2012-06-28 Abbott Gmbh & Co. Kg Solid retard formulations based on solid dispersions
CN102641252B (zh) * 2012-05-08 2014-06-04 南京臣功制药股份有限公司 盐酸特比萘芬固体分散体及其片剂
WO2014048783A1 (en) * 2012-09-27 2014-04-03 Basf Se A storage-stable dust-free homogeneous particulate formulation comprising at least one water-soluble vitamin e-derivative and at least one hydrophilic polymer
TW201431570A (zh) 2012-11-22 2014-08-16 Ucb Pharma Gmbh 用於經皮投服羅替戈汀(Rotigotine)之多天式貼片
WO2014143127A1 (en) 2013-03-15 2014-09-18 Differential Drug Development Associates Llc Emulsion formulations
CN105358139B (zh) 2013-07-03 2020-10-16 Lts罗曼治疗方法有限公司 具有电子元件的经皮治疗系统
JP6235924B2 (ja) * 2014-02-13 2017-11-22 壽製薬株式会社 フェノフィブラートの固体分散体
ES2954087T3 (es) 2014-05-20 2023-11-20 Lts Lohmann Therapie Systeme Ag Sistema de administración transdérmica que incluye un mediador de interfase
JP6573913B2 (ja) * 2014-05-20 2019-09-11 エルテーエス ローマン テラピー−ジステーメ アーゲー ロチゴチンを含む経皮送達システム
CN106456567A (zh) 2014-05-20 2017-02-22 Lts勒曼治疗系统股份公司 在经皮递送系统中调节活性剂释放的方法
JP6584754B2 (ja) * 2014-07-02 2019-10-02 国立大学法人京都大学 ポリマーアロイ及びその製造方法
MD4399C1 (ro) * 2015-02-19 2016-09-30 Государственный Университет Молд0 Material polimeric cu proprietăţi antibacteriene
CN106265580B (zh) * 2015-05-18 2020-09-08 中国科学院上海药物研究所 Somcl-9112固体分散体、其制备方法及包含其的somcl-9112固体制剂
WO2017009865A1 (en) * 2015-07-10 2017-01-19 Sun Pharma Advanced Research Company Ltd. Multiple pill abuse-resistant immediate release solid dosage form of hydrocodone
JP6914916B2 (ja) * 2015-08-21 2021-08-04 ビーエイエスエフ・ソシエタス・エウロパエアBasf Se N−ビニルピロリドン及びアクリル酸をベースとした水溶性ポリマーの医薬助剤としての使用
EP3492070A1 (en) * 2017-11-30 2019-06-05 BIT Pharma GmbH Process and device for preparing a solid dispersion
CN108295264A (zh) * 2018-03-28 2018-07-20 五邑大学 聚乙烯吡咯烷酮k12的应用
EP3628310A1 (en) * 2018-09-25 2020-04-01 Synbias Pharma AG Pharmaceutical composition comprising solid dispersions of amorphous cladribine and pharmaceutically acceptable water soluble carrier
KR102125624B1 (ko) 2018-11-22 2020-07-07 전북대학교산학협력단 핸드헬드형 분광타원편광계측장치 및 이를 이용한 분광타원편광 파라미터 측정방법
RU2723999C1 (ru) * 2019-04-19 2020-06-18 Общество с ограниченной ответственностью "Химико-фармацевтические технологии" (ООО "ХимФармТех") Композиция для ингибирования активности β-глюкуронидазы
US12403146B2 (en) 2019-10-30 2025-09-02 Marius Pharmaceuticals, Inc. Preferred oral testosterone undecanoate therapy to achieve testosterone replacement treatment
RU2748311C1 (ru) * 2020-01-29 2021-05-21 Общество с ограниченной ответственностью "ФармЭко" Фармацевтическая композиция, содержащая твердые дисперсии аморфного кладрибина и фармацевтически приемлемый водорастворимый носитель
CN112206213A (zh) * 2020-10-26 2021-01-12 广州汇元医药科技有限公司 一种枸橼酸西地那非组合物及其制备方法
CN115671110B (zh) * 2021-07-30 2024-05-10 上海云晟研新生物科技有限公司 帕唑帕尼口服药物组合物、其制备方法及应用
KR20250100660A (ko) 2022-10-25 2025-07-03 베라더믹스 인코포레이티드 변형 방출 미녹시딜의 조성물 및 사용 방법

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DE19602206A1 (de) * 1996-01-23 1997-07-24 Basf Ag Zubereitungen nichtsteroidaler Analgetika
US20030119882A1 (en) * 2001-10-22 2003-06-26 Markus Maegerlein Solid pharmaceutical composition containing torasemide
MY140561A (en) * 2002-02-20 2009-12-31 Nycomed Gmbh Dosage form containing pde 4 inhibitor as active ingredient
US7820732B2 (en) * 2004-04-30 2010-10-26 Advanced Cardiovascular Systems, Inc. Methods for modulating thermal and mechanical properties of coatings on implantable devices
KR101086254B1 (ko) 2004-11-04 2011-11-24 에스케이케미칼주식회사 생체이용률이 개선된 프란루카스트 고체분산체 조성물 및그 고체분산체의 제조방법
EP1690528A1 (de) * 2005-02-11 2006-08-16 Abbott GmbH & Co. KG Herstellung von Dosierungsformen mit einer festen Dispersion eines mikrokristallinen Wirkstoffs
DE102005026755A1 (de) * 2005-06-09 2006-12-14 Basf Ag Herstellung von festen Lösungen schwerlöslicher Wirkstoffe durch Kurzzeitüberhitzung und schnelle Trocknung
RU2423997C9 (ru) * 2005-07-05 2011-11-20 Эббетт ГмбХ унд Ко. КГ Композиция и лекарственная форма, содержащие твердую или полутвердую матрицу
WO2007062347A2 (en) * 2005-11-22 2007-05-31 Smithkline Beecham Corporation Foamed substrate and method for making same
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EP2260022B1 (de) 2008-03-27 2017-01-04 Grünenthal GmbH Substituierte cyclohexyldiamine
EP2140861A1 (en) * 2008-06-30 2010-01-06 Abbott GmbH & Co. KG Pharmaceutical dosage form comprising polymeric carrier composition

Also Published As

Publication number Publication date
US9402909B2 (en) 2016-08-02
JP2015063549A (ja) 2015-04-09
CA2729148C (en) 2016-05-17
AU2009265737A1 (en) 2010-01-07
EP2140861A1 (en) 2010-01-06
CN102083420A (zh) 2011-06-01
CN102083420B (zh) 2013-06-05
ES2699075T3 (es) 2019-02-07
US20140200278A1 (en) 2014-07-17
WO2010000740A1 (en) 2010-01-07
RU2519679C2 (ru) 2014-06-20
KR20110046457A (ko) 2011-05-04
RU2011103085A (ru) 2012-08-10
EP2303242B1 (en) 2018-05-02
CA2729148A1 (en) 2010-01-07
US20110182891A1 (en) 2011-07-28
KR101812508B1 (ko) 2017-12-27
AU2009265737B2 (en) 2015-04-16
RU2519679C9 (ru) 2015-02-27
EP2303242A1 (en) 2011-04-06
JP5717628B2 (ja) 2015-05-13
JP2011526592A (ja) 2011-10-13
JP5976086B2 (ja) 2016-08-23

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Legal Events

Date Code Title Description
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B07E Notice of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]

Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI

B06T Formal requirements before examination [chapter 6.20 patent gazette]
B06A Notification to applicant to reply to the report for non-patentability or inadequacy of the application [chapter 6.1 patent gazette]
B15K Others concerning applications: alteration of classification

Free format text: AS CLASSIFICACOES ANTERIORES ERAM: A61K 9/20 , A61K 47/32

Ipc: A61K 47/32 (1990.01), A61K 9/20 (1974.07), A61K 9/

B09B Patent application refused [chapter 9.2 patent gazette]
B15K Others concerning applications: alteration of classification

Free format text: AS CLASSIFICACOES ANTERIORES ERAM: A61K 47/32 , A61K 9/20 , A61K 9/28

Ipc: A61K 9/20 (2006.01), A61K 9/28 (2006.01)

B12B Appeal: appeal against refusal
B08F Application fees: application dismissed [chapter 8.6 patent gazette]

Free format text: REFERENTE A 12A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2626 DE 04-05-2021 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.