BRPI0816372A2 - Ácidos 6-fenilnicotínicos substituídos e seu uso - Google Patents

Ácidos 6-fenilnicotínicos substituídos e seu uso

Info

Publication number: BRPI0816372A2
Authority: BR; Brazil
Prior art keywords: phenylnicotinic; acids; replaced; phenylnicotinic acids
Prior art date: 2007-09-07

Application number

BRPI0816372-3A2A

Other languages

English (en)

Inventor

Lars Baerfacker

Jens Schamberger

Klemens Lustig

Barbara Albrecht-Kuepper

Peter Kolkhof

Yolanda Cancho Grande

Adam Nitsche

Heinrich Meier

Carsten Schmeck

Original Assignee

Bayer Animal Health Gmbh

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2007-09-07

Filing date

2008-08-26

Publication date

2015-02-24

2008-08-26 Application filed by Bayer Animal Health Gmbh filed Critical Bayer Animal Health Gmbh

2015-02-24 Publication of BRPI0816372A2 publication Critical patent/BRPI0816372A2/pt

Links

239000002253 acid Substances 0.000 title 1
150000007513 acids Chemical class 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/79—Acids; Esters
- C07D213/80—Acids; Esters in position 3
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Cardiology (AREA)
Physical Education & Sports Medicine (AREA)
Dermatology (AREA)
Rheumatology (AREA)
Heart & Thoracic Surgery (AREA)
Hematology (AREA)
Diabetes (AREA)
Pain & Pain Management (AREA)
Oncology (AREA)
Urology & Nephrology (AREA)
Pulmonology (AREA)
Orthopedic Medicine & Surgery (AREA)
Vascular Medicine (AREA)
Hospice & Palliative Care (AREA)
Communicable Diseases (AREA)
Psychiatry (AREA)
Obesity (AREA)
Gastroenterology & Hepatology (AREA)
Psychology (AREA)
Virology (AREA)
Immunology (AREA)
Endocrinology (AREA)

BRPI0816372-3A2A 2007-09-07 2008-08-26 Ácidos 6-fenilnicotínicos substituídos e seu uso BRPI0816372A2 (pt)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE102007042754A DE102007042754A1 (de)	2007-09-07	2007-09-07	Substituierte 6-Phenylnikotinsäuren und ihre Verwendung
PCT/EP2008/006969 WO2009033561A1 (de)	2007-09-07	2008-08-26	Substituierte 6-phenylnikotinsäuren und ihre verwendung

Publications (1)

Publication Number	Publication Date
BRPI0816372A2 true BRPI0816372A2 (pt)	2015-02-24

Family

ID=40032794

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BRPI0816372-3A2A BRPI0816372A2 (pt)	2007-09-07	2008-08-26	Ácidos 6-fenilnicotínicos substituídos e seu uso

Country Status (16)

Country	Link
US (1)	US8143411B2 (pt)
EP (1)	EP2197846A1 (pt)
JP (1)	JP2010538025A (pt)
KR (1)	KR20100066545A (pt)
AU (1)	AU2008298021A1 (pt)
BR (1)	BRPI0816372A2 (pt)
CA (1)	CA2698471A1 (pt)
CL (1)	CL2008002537A1 (pt)
DE (1)	DE102007042754A1 (pt)
MX (1)	MX2010002565A (pt)
NZ (1)	NZ583697A (pt)
PA (1)	PA8794401A1 (pt)
PE (1)	PE20090954A1 (pt)
TW (1)	TW200914002A (pt)
UY (1)	UY31310A1 (pt)
WO (1)	WO2009033561A1 (pt)

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DK3068392T5 (da)	2013-11-12	2021-09-20	Vertex Pharma	Fremgangsmåde til fremstilling af farmaceutiske sammensætninger til behandlingen af cftr-medierede sygdomme
WO2016081556A1 (en)	2014-11-18	2016-05-26	Vertex Pharmaceuticals Incorporated	Process of conducting high throughput testing high performance liquid chromatography
WO2021252951A1 (en)	2020-06-12	2021-12-16	Vanderbilt University	Methods of treatment for gastrointestinal motility disorders

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2007
- 2007-09-07 DE DE102007042754A patent/DE102007042754A1/de not_active Withdrawn
2008
- 2008-08-26 EP EP08801700A patent/EP2197846A1/de not_active Withdrawn
- 2008-08-26 BR BRPI0816372-3A2A patent/BRPI0816372A2/pt not_active IP Right Cessation
- 2008-08-26 CA CA2698471A patent/CA2698471A1/en not_active Abandoned
- 2008-08-26 NZ NZ583697A patent/NZ583697A/en not_active IP Right Cessation
- 2008-08-26 JP JP2010523302A patent/JP2010538025A/ja not_active Withdrawn
- 2008-08-26 WO PCT/EP2008/006969 patent/WO2009033561A1/de not_active Ceased
- 2008-08-26 KR KR1020107007500A patent/KR20100066545A/ko not_active Withdrawn
- 2008-08-26 MX MX2010002565A patent/MX2010002565A/es active IP Right Grant
- 2008-08-26 AU AU2008298021A patent/AU2008298021A1/en not_active Abandoned
- 2008-08-26 US US12/676,568 patent/US8143411B2/en active Active
- 2008-08-27 UY UY31310A patent/UY31310A1/es not_active Application Discontinuation
- 2008-08-28 PA PA20088794401A patent/PA8794401A1/es unknown
- 2008-08-28 PE PE2008001459A patent/PE20090954A1/es not_active Application Discontinuation
- 2008-08-28 CL CL2008002537A patent/CL2008002537A1/es unknown
- 2008-09-05 TW TW097133999A patent/TW200914002A/zh unknown

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Publication number	Publication date
WO2009033561A8 (de)	2010-06-10
US20100234432A1 (en)	2010-09-16
AU2008298021A1 (en)	2009-03-19
MX2010002565A (es)	2010-04-30
UY31310A1 (es)	2009-04-30
EP2197846A1 (de)	2010-06-23
TW200914002A (en)	2009-04-01
PA8794401A1 (es)	2009-07-23
US8143411B2 (en)	2012-03-27
KR20100066545A (ko)	2010-06-17
CA2698471A1 (en)	2009-03-19
DE102007042754A1 (de)	2009-03-12
JP2010538025A (ja)	2010-12-09
WO2009033561A1 (de)	2009-03-19
CL2008002537A1 (es)	2009-03-20
NZ583697A (en)	2012-04-27
PE20090954A1 (es)	2009-07-24

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2015-12-01	B08F	Application fees: application dismissed [chapter 8.6 patent gazette]	Free format text: REFERENTE AS 6A E 7A ANUIDADES.
2016-03-29	B08K	Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]	Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2343 DE 01-12-2015 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.

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