BRPI0817804A2 - agente terapêutico para melhorar as propriedades da pele compreendendo um derivado de morfinano ou qualquer um de seus sais de adição de ácido farmacologicamente permissíveis como um ingrediente ativo. - Google Patents
agente terapêutico para melhorar as propriedades da pele compreendendo um derivado de morfinano ou qualquer um de seus sais de adição de ácido farmacologicamente permissíveis como um ingrediente ativo.Info
- Publication number
- BRPI0817804A2 BRPI0817804A2 BRPI0817804A BRPI0817804A BRPI0817804A2 BR PI0817804 A2 BRPI0817804 A2 BR PI0817804A2 BR PI0817804 A BRPI0817804 A BR PI0817804A BR PI0817804 A BRPI0817804 A BR PI0817804A BR PI0817804 A2 BRPI0817804 A2 BR PI0817804A2
- Authority
- BR
- Brazil
- Prior art keywords
- active ingredient
- therapeutic agent
- acid addition
- addition salts
- enhancing skin
- Prior art date
Links
- 239000002253 acid Substances 0.000 title 1
- 239000004480 active ingredient Substances 0.000 title 1
- 239000003814 drug Substances 0.000 title 1
- 230000002708 enhancing effect Effects 0.000 title 1
- INAXVFBXDYWQFN-XHSDSOJGSA-N morphinan Chemical class C1C2=CC=CC=C2[C@]23CCCC[C@H]3[C@@H]1NCC2 INAXVFBXDYWQFN-XHSDSOJGSA-N 0.000 title 1
- 150000003839 salts Chemical class 0.000 title 1
- 229940124597 therapeutic agent Drugs 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D489/00—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:
- C07D489/06—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: with a hetero atom directly attached in position 14
- C07D489/08—Oxygen atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/04—Antipruritics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/16—Emollients or protectives, e.g. against radiation
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q19/00—Preparations for care of the skin
- A61Q19/007—Preparations for dry skin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2800/00—Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
- A61K2800/80—Process related aspects concerning the preparation of the cosmetic composition or the storage or application thereof
- A61K2800/92—Oral administration
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Dermatology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Birds (AREA)
- Epidemiology (AREA)
- Toxicology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cosmetics (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2007262015 | 2007-10-05 | ||
| PCT/JP2008/068092 WO2009044883A1 (ja) | 2007-10-05 | 2008-10-03 | モルヒナン誘導体またはその薬理学的に許容される酸付加塩を有効成分とする皮膚性状改善治療薬 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| BRPI0817804A2 true BRPI0817804A2 (pt) | 2016-10-11 |
| BRPI0817804A8 BRPI0817804A8 (pt) | 2017-04-18 |
Family
ID=40526303
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0817804A BRPI0817804A8 (pt) | 2007-10-05 | 2008-10-03 | Agente terapêutico para melhorar as propriedades da pele compreendendo um derivado de morfinano ou qualquer um de seus sais de adição de ácido farmacologicamente permissíveis como um ingrediente ativo |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US20100222309A1 (pt) |
| EP (1) | EP2196206B8 (pt) |
| JP (1) | JP5613417B2 (pt) |
| KR (1) | KR101173509B1 (pt) |
| CN (1) | CN101848714B (pt) |
| AU (1) | AU2008308005B2 (pt) |
| BR (1) | BRPI0817804A8 (pt) |
| CA (1) | CA2702032C (pt) |
| ES (1) | ES2748274T3 (pt) |
| MX (1) | MX2010003660A (pt) |
| PL (1) | PL2196206T3 (pt) |
| RU (1) | RU2440117C1 (pt) |
| TW (1) | TWI453020B (pt) |
| WO (1) | WO2009044883A1 (pt) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX362830B (es) * | 2010-01-29 | 2019-02-14 | Toray Industries | Agente terapeutico o profilactico para enfermedades del tracto biliar. |
| WO2012054566A2 (en) * | 2010-10-19 | 2012-04-26 | Memorial Sloan-Kettering Cancer Center | 6-amido derivatives of 4,5a-epoxymorphinans for treatment of pain |
| ES2586655T3 (es) | 2011-01-31 | 2016-10-18 | Toray Industries, Inc. | (-)-17-(ciclopropilmetil)-3,14beta-dihidroxi-4,5alfa-epoxi-6beta-[N-metil-trans-3-(3-furil)acrilamido]morfinano para su utilización en el tratamiento o prevención de la caquexia por cáncer |
| EP2931725B1 (en) | 2012-12-14 | 2017-02-15 | Purdue Pharma LP | Nitrogen containing morphinan derivatives and the use thereof |
| CA2896202A1 (en) | 2012-12-28 | 2014-07-03 | Purdue Pharma L.P. | Substituted morphinans and the use thereof |
| WO2016176657A1 (en) | 2015-04-30 | 2016-11-03 | Memorial Sloan-Kettering Cancer Center | Mitragynine analogs and uses thereof |
| CN105461727A (zh) * | 2015-12-01 | 2016-04-06 | 吕涛 | 一种纳呋拉啡的精制方法 |
| WO2018160500A1 (en) | 2017-03-03 | 2018-09-07 | Ring Inc. | Solar-charging mounting bracket for audio/video recording and communication devices |
| HUE069820T2 (hu) | 2018-03-08 | 2025-04-28 | Victoria Link Ltd | Nalfurafin alkalmazása demielinizációs betegségek kezelésére |
| TWI893157B (zh) * | 2020-06-30 | 2025-08-11 | 日商東麗股份有限公司 | 具有嗎啡喃骨架之化合物或其藥理學上可容許之酸加成鹽的用途 |
| CR20230576A (es) | 2021-06-14 | 2024-04-05 | Scorpion Therapeutics Inc | Derivados de la urea que pueden ser utilizados para tratar el cáncer |
Family Cites Families (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4923875A (en) * | 1989-07-10 | 1990-05-08 | Baker Cummins Pharmaceuticals, Inc. | Method for treatment of mast cell-mediated dermatologic disorders |
| JP2521853B2 (ja) | 1990-07-25 | 1996-08-07 | タカラベルモント株式会社 | 化粧料 |
| US6323212B1 (en) | 1992-01-23 | 2001-11-27 | Toray Industries, Inc. | Morphinan derivative and its pharmaceutical applications |
| EP0661283B1 (en) | 1993-07-19 | 1998-10-21 | Toray Industries, Inc. | Brain cell protective |
| EP0663401B1 (en) * | 1993-07-23 | 2000-06-07 | Toray Industries, Inc. | Morphinan derivative and medicinal use |
| JPH07187990A (ja) | 1993-12-24 | 1995-07-25 | Toshiko Yamamoto | 化粧料 |
| ATE359076T1 (de) * | 1996-11-25 | 2007-05-15 | Toray Industries | Mittel gegen juckreiz |
| US5834480A (en) * | 1997-06-13 | 1998-11-10 | Elkhoury; George F. | Topical application of opioids for treatment of acne and sebaceous gland disorders |
| WO1999005146A1 (en) | 1997-07-25 | 1999-02-04 | Toray Industries, Inc. | Hyponatremia remedies |
| JP4359711B2 (ja) | 1997-09-02 | 2009-11-04 | 東レ株式会社 | 薬物依存症治療薬 |
| JP2000053572A (ja) | 1998-08-11 | 2000-02-22 | Toray Ind Inc | ORL1(opioid orphan)受容体拮抗薬 |
| DE60039444D1 (de) | 1999-08-24 | 2008-08-21 | Toray Industries | Heilmittel für neuropathischen schmerz und versuchstier-modelle des neuropathischen schmerzes |
| CA2442423C (en) | 2001-03-30 | 2009-11-03 | Toray Industries, Inc. | Therapeutic drug for psychoneurotic disorders |
| EP1402899A4 (en) | 2001-05-08 | 2009-03-11 | Toray Industries | MEANS FOR THE TREATMENT OF SEPSIS |
| JP2004107209A (ja) | 2002-09-13 | 2004-04-08 | Nippon Oruganon Kk | 掻痒治療薬 |
| RU2221545C1 (ru) * | 2002-11-13 | 2004-01-20 | Открытое Акционерное Общество "Фаберлик" | Косметическое средство, улучшающее физиологическое состояние кожных покровов |
| JP4499034B2 (ja) * | 2003-02-19 | 2010-07-07 | 久光製薬株式会社 | N−アリール又はn−ヘテロアリールピペラジン誘導体及びそれを含有する医薬 |
| JP2004352714A (ja) | 2003-05-08 | 2004-12-16 | Kyorin Pharmaceut Co Ltd | 新規な4−(2−フロイル)アミノピペリジン誘導体 |
| JP4381157B2 (ja) | 2004-02-03 | 2009-12-09 | 久光製薬株式会社 | 2,2−ジフェニル−1−エタノン誘導体及びそれを含有する医薬 |
| ATE456373T1 (de) * | 2004-11-29 | 2010-02-15 | Unilever Nv | Orale zusammensetzung zur verbesserung der hauteigenschaften |
| PT1870413E (pt) * | 2005-03-10 | 2013-10-01 | Toray Industries | Agente antiprurítico para o pruridro provocado pela esclerose múltipla |
| WO2007053194A2 (en) * | 2005-06-03 | 2007-05-10 | The University Of Chicago | Modulation of cell barrier dysfunction |
| RU2299724C1 (ru) * | 2005-11-14 | 2007-05-27 | Открытое Акционерное Общество "Фаберлик" | Средство, улучшающее физиологическое состояние клеток кожи |
-
2008
- 2008-10-03 MX MX2010003660A patent/MX2010003660A/es not_active Application Discontinuation
- 2008-10-03 RU RU2010117649/15A patent/RU2440117C1/ru active
- 2008-10-03 KR KR1020107007134A patent/KR101173509B1/ko not_active Expired - Fee Related
- 2008-10-03 BR BRPI0817804A patent/BRPI0817804A8/pt not_active IP Right Cessation
- 2008-10-03 TW TW097138034A patent/TWI453020B/zh not_active IP Right Cessation
- 2008-10-03 WO PCT/JP2008/068092 patent/WO2009044883A1/ja not_active Ceased
- 2008-10-03 PL PL08835121T patent/PL2196206T3/pl unknown
- 2008-10-03 CA CA2702032A patent/CA2702032C/en not_active Expired - Fee Related
- 2008-10-03 AU AU2008308005A patent/AU2008308005B2/en not_active Ceased
- 2008-10-03 JP JP2009536121A patent/JP5613417B2/ja not_active Expired - Fee Related
- 2008-10-03 US US12/680,908 patent/US20100222309A1/en not_active Abandoned
- 2008-10-03 CN CN200880110176.5A patent/CN101848714B/zh not_active Expired - Fee Related
- 2008-10-03 ES ES08835121T patent/ES2748274T3/es active Active
- 2008-10-03 EP EP08835121.8A patent/EP2196206B8/en not_active Not-in-force
Also Published As
| Publication number | Publication date |
|---|---|
| CA2702032A1 (en) | 2009-04-09 |
| AU2008308005A1 (en) | 2009-04-09 |
| TWI453020B (zh) | 2014-09-21 |
| MX2010003660A (es) | 2010-08-10 |
| ES2748274T3 (es) | 2020-03-16 |
| CN101848714B (zh) | 2014-08-20 |
| JPWO2009044883A1 (ja) | 2011-02-10 |
| BRPI0817804A8 (pt) | 2017-04-18 |
| EP2196206A4 (en) | 2010-09-22 |
| CA2702032C (en) | 2013-04-02 |
| WO2009044883A1 (ja) | 2009-04-09 |
| KR20100049683A (ko) | 2010-05-12 |
| PL2196206T3 (pl) | 2020-02-28 |
| EP2196206A1 (en) | 2010-06-16 |
| RU2440117C1 (ru) | 2012-01-20 |
| CN101848714A (zh) | 2010-09-29 |
| US20100222309A1 (en) | 2010-09-02 |
| EP2196206B8 (en) | 2019-11-13 |
| EP2196206B1 (en) | 2019-07-17 |
| TW200927116A (en) | 2009-07-01 |
| JP5613417B2 (ja) | 2014-10-22 |
| KR101173509B1 (ko) | 2012-08-14 |
| AU2008308005B2 (en) | 2012-06-07 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] | ||
| B25A | Requested transfer of rights approved |
Owner name: TORAY INDUSTRIES, INC. (JP) |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] | ||
| B350 | Update of information on the portal [chapter 15.35 patent gazette] |