BRPI0817804A2 - agente terapêutico para melhorar as propriedades da pele compreendendo um derivado de morfinano ou qualquer um de seus sais de adição de ácido farmacologicamente permissíveis como um ingrediente ativo. - Google Patents

agente terapêutico para melhorar as propriedades da pele compreendendo um derivado de morfinano ou qualquer um de seus sais de adição de ácido farmacologicamente permissíveis como um ingrediente ativo.

Info

Publication number
BRPI0817804A2
BRPI0817804A2 BRPI0817804A BRPI0817804A BRPI0817804A2 BR PI0817804 A2 BRPI0817804 A2 BR PI0817804A2 BR PI0817804 A BRPI0817804 A BR PI0817804A BR PI0817804 A BRPI0817804 A BR PI0817804A BR PI0817804 A2 BRPI0817804 A2 BR PI0817804A2
Authority
BR
Brazil
Prior art keywords
active ingredient
therapeutic agent
acid addition
addition salts
enhancing skin
Prior art date
Application number
BRPI0817804A
Other languages
English (en)
Inventor
Koichiro Takeshita
Masahiro Yamashita
Naoki Ando
Shinji Ona
Original Assignee
Torii Pharmaceutical Co Ltd
Toray Industries
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Torii Pharmaceutical Co Ltd, Toray Industries filed Critical Torii Pharmaceutical Co Ltd
Publication of BRPI0817804A2 publication Critical patent/BRPI0817804A2/pt
Publication of BRPI0817804A8 publication Critical patent/BRPI0817804A8/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D489/00Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:
    • C07D489/06Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: with a hetero atom directly attached in position 14
    • C07D489/08Oxygen atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/49Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/04Antipruritics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/16Emollients or protectives, e.g. against radiation
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00Preparations for care of the skin
    • A61Q19/007Preparations for dry skin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2800/00Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
    • A61K2800/80Process related aspects concerning the preparation of the cosmetic composition or the storage or application thereof
    • A61K2800/92Oral administration

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Dermatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Birds (AREA)
  • Epidemiology (AREA)
  • Toxicology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cosmetics (AREA)
BRPI0817804A 2007-10-05 2008-10-03 Agente terapêutico para melhorar as propriedades da pele compreendendo um derivado de morfinano ou qualquer um de seus sais de adição de ácido farmacologicamente permissíveis como um ingrediente ativo BRPI0817804A8 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2007262015 2007-10-05
PCT/JP2008/068092 WO2009044883A1 (ja) 2007-10-05 2008-10-03 モルヒナン誘導体またはその薬理学的に許容される酸付加塩を有効成分とする皮膚性状改善治療薬

Publications (2)

Publication Number Publication Date
BRPI0817804A2 true BRPI0817804A2 (pt) 2016-10-11
BRPI0817804A8 BRPI0817804A8 (pt) 2017-04-18

Family

ID=40526303

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0817804A BRPI0817804A8 (pt) 2007-10-05 2008-10-03 Agente terapêutico para melhorar as propriedades da pele compreendendo um derivado de morfinano ou qualquer um de seus sais de adição de ácido farmacologicamente permissíveis como um ingrediente ativo

Country Status (14)

Country Link
US (1) US20100222309A1 (pt)
EP (1) EP2196206B8 (pt)
JP (1) JP5613417B2 (pt)
KR (1) KR101173509B1 (pt)
CN (1) CN101848714B (pt)
AU (1) AU2008308005B2 (pt)
BR (1) BRPI0817804A8 (pt)
CA (1) CA2702032C (pt)
ES (1) ES2748274T3 (pt)
MX (1) MX2010003660A (pt)
PL (1) PL2196206T3 (pt)
RU (1) RU2440117C1 (pt)
TW (1) TWI453020B (pt)
WO (1) WO2009044883A1 (pt)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PH12012501552A1 (en) * 2010-01-29 2017-04-26 Toray Industries Therapeutic or prophylactic agent for biliary diseases
WO2012054566A2 (en) * 2010-10-19 2012-04-26 Memorial Sloan-Kettering Cancer Center 6-amido derivatives of 4,5a-epoxymorphinans for treatment of pain
CA2825165C (en) 2011-01-31 2018-07-03 Toray Industries, Inc. Therapeutic or prophylactic agent for cachexia
ES2623262T3 (es) 2012-12-14 2017-07-10 Purdue Pharma Lp Derivados de morfinano que contienen nitrógeno y el uso de los mismos
US8946255B2 (en) 2012-12-28 2015-02-03 Purdue Pharma L.P. Substituted morphinans and the use thereof
EP4212532A3 (en) 2015-04-30 2023-09-27 Memorial Sloan Kettering Cancer Center Mitragynine analogs and uses thereof
CN105461727A (zh) * 2015-12-01 2016-04-06 吕涛 一种纳呋拉啡的精制方法
US11082591B2 (en) 2017-03-03 2021-08-03 Amazon Technologies, Inc. Solar-charging mounting bracket for audio/video recording and communication devices
DK3761982T3 (da) 2018-03-08 2025-01-02 Victoria Link Ltd Anvendelse af nalfurafin til behandling af demyeliniserende sygdomme
TWI893157B (zh) * 2020-06-30 2025-08-11 日商東麗股份有限公司 具有嗎啡喃骨架之化合物或其藥理學上可容許之酸加成鹽的用途
US20240300939A1 (en) 2021-06-14 2024-09-12 Scorpion Therapeutics, Inc. Urea derivatives which can be used to treat cancer

Family Cites Families (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4923875A (en) * 1989-07-10 1990-05-08 Baker Cummins Pharmaceuticals, Inc. Method for treatment of mast cell-mediated dermatologic disorders
JP2521853B2 (ja) 1990-07-25 1996-08-07 タカラベルモント株式会社 化粧料
ES2121988T3 (es) 1992-01-23 1998-12-16 Toray Industries Derivado de morfinano y uso medicinal.
KR100341950B1 (ko) 1993-07-19 2002-11-29 도레이 가부시끼가이샤 뇌세포보호제
NZ268969A (en) * 1993-07-23 1997-06-24 Toray Industries Morphinan derivatives and pharmaceutical compositions
JPH07187990A (ja) 1993-12-24 1995-07-25 Toshiko Yamamoto 化粧料
DE69732868T2 (de) * 1996-11-25 2006-04-13 Toray Industries, Inc. Mittel gegen Juckreiz
US5834480A (en) * 1997-06-13 1998-11-10 Elkhoury; George F. Topical application of opioids for treatment of acne and sebaceous gland disorders
WO1999005146A1 (en) * 1997-07-25 1999-02-04 Toray Industries, Inc. Hyponatremia remedies
JP4359711B2 (ja) 1997-09-02 2009-11-04 東レ株式会社 薬物依存症治療薬
JP2000053572A (ja) 1998-08-11 2000-02-22 Toray Ind Inc ORL1(opioid orphan)受容体拮抗薬
CN1204139C (zh) 1999-08-24 2005-06-01 东丽株式会社 神经性疼痛治疗剂
US8338442B2 (en) 2001-03-30 2012-12-25 Toray Industries, Inc. Remedies for psychoneurosis
JP4239592B2 (ja) 2001-05-08 2009-03-18 東レ株式会社 敗血症治療剤
JP2004107209A (ja) 2002-09-13 2004-04-08 Nippon Oruganon Kk 掻痒治療薬
RU2221545C1 (ru) * 2002-11-13 2004-01-20 Открытое Акционерное Общество "Фаберлик" Косметическое средство, улучшающее физиологическое состояние кожных покровов
WO2004074277A1 (ja) * 2003-02-19 2004-09-02 Hisamitsu Medical Co., Ltd. N-アリール又はn-ヘテロアリールピペラジン誘導体及びそれを含有する医薬
JP2004352714A (ja) 2003-05-08 2004-12-16 Kyorin Pharmaceut Co Ltd 新規な4−(2−フロイル)アミノピペリジン誘導体
JP4381157B2 (ja) * 2004-02-03 2009-12-09 久光製薬株式会社 2,2−ジフェニル−1−エタノン誘導体及びそれを含有する医薬
PL1833498T3 (pl) * 2004-11-29 2010-06-30 Unilever Nv Doustna kompozycja do polepszania właściwości skóry
AU2006221314B2 (en) * 2005-03-10 2012-09-06 Toray Industries, Inc. Antipruritic agent for pruritus caused by multiple sclerosis
EP1901742A2 (en) * 2005-06-03 2008-03-26 The University of Chicago Modulation of cell barrier dysfunction
RU2299724C1 (ru) * 2005-11-14 2007-05-27 Открытое Акционерное Общество "Фаберлик" Средство, улучшающее физиологическое состояние клеток кожи

Also Published As

Publication number Publication date
JP5613417B2 (ja) 2014-10-22
EP2196206A4 (en) 2010-09-22
ES2748274T3 (es) 2020-03-16
CA2702032A1 (en) 2009-04-09
CN101848714B (zh) 2014-08-20
PL2196206T3 (pl) 2020-02-28
KR101173509B1 (ko) 2012-08-14
MX2010003660A (es) 2010-08-10
AU2008308005B2 (en) 2012-06-07
US20100222309A1 (en) 2010-09-02
JPWO2009044883A1 (ja) 2011-02-10
KR20100049683A (ko) 2010-05-12
WO2009044883A1 (ja) 2009-04-09
BRPI0817804A8 (pt) 2017-04-18
CN101848714A (zh) 2010-09-29
EP2196206A1 (en) 2010-06-16
RU2440117C1 (ru) 2012-01-20
EP2196206B8 (en) 2019-11-13
AU2008308005A1 (en) 2009-04-09
TWI453020B (zh) 2014-09-21
EP2196206B1 (en) 2019-07-17
TW200927116A (en) 2009-07-01
CA2702032C (en) 2013-04-02

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]
B25A Requested transfer of rights approved

Owner name: TORAY INDUSTRIES, INC. (JP)

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]
B350 Update of information on the portal [chapter 15.35 patent gazette]