BRPI0907204A2 - pirazolopirimidinas, um processo para sua preparação e seu uso como medicamento - Google Patents

pirazolopirimidinas, um processo para sua preparação e seu uso como medicamento

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Publication number
BRPI0907204A2
BRPI0907204A2 BRPI0907204-7A BRPI0907204A BRPI0907204A2 BR PI0907204 A2 BRPI0907204 A2 BR PI0907204A2 BR PI0907204 A BRPI0907204 A BR PI0907204A BR PI0907204 A2 BRPI0907204 A2 BR PI0907204A2
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Brazil
Prior art keywords
preparation
pyrazolopyrimidines
medicine
compounds
relates
Prior art date
Application number
BRPI0907204-7A
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English (en)
Inventor
Henrich Markus
Weil Tanja
Muller Sibylle
Nagel Jens
Gravius Andreas
Kauss Valerjans
Zemribo Ronalds
Erdmane Elina
Original Assignee
Merz Pharma Gmbh & Co. Kgaa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by Merz Pharma Gmbh & Co. Kgaa filed Critical Merz Pharma Gmbh & Co. Kgaa
Publication of BRPI0907204A2 publication Critical patent/BRPI0907204A2/pt

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    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

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Abstract

pirazolopirimidinas, um processo para sua preparação e seu uso como medicamento a invenção está relacionada aos derivados de pirazolopirirnidina de fórmula (i) , em que r1 representa cloro ou bromo; a representa (a); (b); (c); (d); ou (e), bem corno seus sais farrnaceuticarnente aceitáveis. a invenção ainda está relacionada a um processo para a preparação desses compostos. os compostos da invenção são rnoduladores de rnglurs e, portanto, são úteis para o controle e prevenção de distúrbios neurológicos agudos e/ou crônicos.
BRPI0907204-7A 2008-02-01 2009-01-30 pirazolopirimidinas, um processo para sua preparação e seu uso como medicamento BRPI0907204A2 (pt)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US6342108P 2008-02-01 2008-02-01
EP082503962 2008-02-01
US61/063,421 2008-02-01
EP08250396A EP2085398A1 (en) 2008-02-01 2008-02-01 Pyrazolopyrimidines, a process for their preparation and their use as medicine
PCT/EP2009/000616 WO2009095254A1 (en) 2008-02-01 2009-01-30 Pyrazolopyrimidines, a process for their preparation and their use as medicine

Publications (1)

Publication Number Publication Date
BRPI0907204A2 true BRPI0907204A2 (pt) 2019-02-26

Family

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BRPI0907204-7A BRPI0907204A2 (pt) 2008-02-01 2009-01-30 pirazolopirimidinas, um processo para sua preparação e seu uso como medicamento

Country Status (13)

Country Link
US (1) US20110003820A1 (pt)
EP (2) EP2085398A1 (pt)
JP (1) JP2011510943A (pt)
KR (1) KR20100117640A (pt)
CN (1) CN101939323A (pt)
AU (1) AU2009210197A1 (pt)
BR (1) BRPI0907204A2 (pt)
CA (1) CA2711575A1 (pt)
IL (1) IL207110A0 (pt)
MX (1) MX2010008469A (pt)
RU (1) RU2010136661A (pt)
WO (1) WO2009095254A1 (pt)
ZA (1) ZA201004862B (pt)

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