BRPI0909655A2 - Processo para a preparação regioseletiva de derivados de ácido 1-alquil-3-haloalquil-pirazol-4carboxílico - Google Patents
Processo para a preparação regioseletiva de derivados de ácido 1-alquil-3-haloalquil-pirazol-4carboxílicoInfo
- Publication number
- BRPI0909655A2 BRPI0909655A2 BRPI0909655-8A BRPI0909655A BRPI0909655A2 BR PI0909655 A2 BRPI0909655 A2 BR PI0909655A2 BR PI0909655 A BRPI0909655 A BR PI0909655A BR PI0909655 A2 BRPI0909655 A2 BR PI0909655A2
- Authority
- BR
- Brazil
- Prior art keywords
- pyrazol
- haloalkyl
- alkyl
- carboxylic acid
- acid derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP08152532.1 | 2008-03-10 | ||
| EP08152532A EP2100883A1 (de) | 2008-03-10 | 2008-03-10 | Verfahren zur regioselektiven Synthese von 1-Alkyl-3-haloalkyl-pyrazol-4carbonsäure-Derivaten |
| PCT/EP2009/001354 WO2009112157A1 (de) | 2008-03-10 | 2009-02-26 | Verfahren zur regioselektiven synthese von l-alkvl-3-haloalkyl-pvrazol-4-carbonsäure-derivaten |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| BRPI0909655A2 true BRPI0909655A2 (pt) | 2015-08-04 |
| BRPI0909655B1 BRPI0909655B1 (pt) | 2018-06-05 |
Family
ID=39587595
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0909655-8A BRPI0909655B1 (pt) | 2008-03-10 | 2009-02-26 | Processo para a preparação regioseletiva de derivados de ácido 1-alquil-3-haloalquil-pirazol- 4carboxílico |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US8350053B2 (pt) |
| EP (2) | EP2100883A1 (pt) |
| JP (1) | JP5503562B2 (pt) |
| KR (1) | KR101652916B1 (pt) |
| CN (1) | CN101970412B (pt) |
| BR (1) | BRPI0909655B1 (pt) |
| CA (1) | CA2717805C (pt) |
| DK (1) | DK2257532T3 (pt) |
| ES (1) | ES2425972T3 (pt) |
| IL (1) | IL207487A (pt) |
| MX (1) | MX2010008899A (pt) |
| MY (1) | MY155478A (pt) |
| PL (1) | PL2257532T3 (pt) |
| RU (1) | RU2498978C2 (pt) |
| TW (1) | TWI440629B (pt) |
| WO (1) | WO2009112157A1 (pt) |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2009021987A1 (en) | 2007-08-16 | 2009-02-19 | Solvay (Société Anonyme) | Process for the preparation of esters of 4-fluorosubstituted 3-oxo-alcanoic acids |
| EP2133341A1 (de) * | 2008-02-25 | 2009-12-16 | Bayer CropScience AG | Verfahren zur regioselektiven Synthese von 1-Alkyl-3-haloalkyl-pyrazol-4-carbonsäure-Derivaten |
| WO2012025469A1 (en) * | 2010-08-24 | 2012-03-01 | Solvay Sa | Improved process for the preparation of esters of 1-h-pyrazole-4-carboxylic acids |
| EP2623496A1 (de) | 2012-02-01 | 2013-08-07 | Bayer CropScience AG | Verfahren zur Herstellung von 3,5-bis (fluoralkyl)-pyrazol-4-carbonsäure-Derivaten und 3,5-bis(fluoralkyl)-pyrazolen |
| EP2644593A1 (en) * | 2012-03-30 | 2013-10-02 | Solvay Sa | Dialkoxymethyl oxobutyric acid esters, their manufacture and use |
| CN102702104B (zh) * | 2012-06-08 | 2015-02-25 | 巨化集团公司 | 一种3-二氟甲基-1-甲基吡唑-4-甲酸乙酯的连续化合成方法 |
| US8871947B2 (en) | 2013-02-04 | 2014-10-28 | KingChem LLC | Preparation of alkyl 3-difluoromethyl-1-methyl-1H-pyrazole-4-carboxylic acid ester |
| EP2999694B1 (en) * | 2013-05-22 | 2017-05-17 | Bayer CropScience Aktiengesellschaft | Process for preparing 3,5-bis(fluoroalkyl)pyrazole derivatives from alpha,alpha -dihaloamines |
| JP6518654B2 (ja) | 2013-05-22 | 2019-05-22 | バイエル・クロップサイエンス・アクチェンゲゼルシャフト | ３，５−ビス（フルオロアルキル）ピラゾール誘導体の製造方法 |
| CN103360313A (zh) * | 2013-07-12 | 2013-10-23 | 雅本化学股份有限公司 | 3-氟代烷基-1-取代吡唑-4-羧酸及其制备方法 |
| TWI647215B (zh) * | 2013-11-11 | 2019-01-11 | 德商拜耳作物科學股份有限公司 | 自α,α－二鹵胺製備３,５－雙鹵烷基吡唑衍生物之方法 |
| WO2015085464A1 (en) | 2013-12-09 | 2015-06-18 | King Chem, Llc | Process for preparing alkyl 3-difluoromethyl-1-methyl-1h-pyrazole-4-carboxylate and its analogs |
| EP3015458A1 (en) | 2014-11-03 | 2016-05-04 | Bayer CropScience AG | Process for preparing 3,5-bis(haloalkyl)pyrazole derivatives from a,a-dihaloamines and ketimines |
| JP6431088B2 (ja) * | 2014-03-24 | 2018-11-28 | バイエル・クロップサイエンス・アクチェンゲゼルシャフト | α，α−ジハロアミン類およびケチミン類からの３，５−ビス（ハロアルキル）ピラゾール誘導体の製造方法 |
| WO2015155713A1 (en) * | 2014-04-09 | 2015-10-15 | Isagro S.P.A. | Process for the regioselective synthesis of 1,3, 4 -substituted pyrazoles |
| BR112016028702B1 (pt) | 2014-06-11 | 2021-05-04 | Bayer Cropscience Aktiengesellschaft | processo para preparação de derivados de 3,5-bis(haloalquil)pirazole via acilação de hidrazonas |
| EP3154947B1 (en) | 2014-06-11 | 2018-03-28 | Bayer CropScience Aktiengesellschaft | Process for preparing 3,5-bis(haloalkyl)pyrazoles via acylation of ketimines |
| CN105541716B (zh) | 2015-03-26 | 2024-02-23 | Ａｇｃ株式会社 | 吡唑衍生物的制造方法 |
| KR20180021798A (ko) | 2015-06-26 | 2018-03-05 | 바이엘 크롭사이언스 악티엔게젤샤프트 | α,α-디할로알킬아민 및 케트이민으로부터 할로알콕시- 및 할로알킬티오 그룹을 가지는 치환된 피라졸의 제조방법 |
| CN106467492B (zh) * | 2015-08-14 | 2019-12-17 | 联化科技(盐城)有限公司 | 多氟甲基吡唑类化合物的制备方法、中间体及制备方法 |
| CN109689629B (zh) | 2016-09-21 | 2022-11-29 | 拜耳作物科学股份公司 | 制备3-氟烷基-5-吡唑羧酸酯和3-氟烷基-5-吡唑羧酸的方法 |
| CN112041303A (zh) * | 2018-05-21 | 2020-12-04 | Pi工业有限公司 | 制备取代的杂环化合物的方法 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2259356C2 (ru) * | 1999-12-09 | 2005-08-27 | Зингента Партисипейшнс Аг | Пиразолкарбоксамидные и пиразолтиоамидные производные в качестве фунгицидов |
| US7038057B2 (en) | 2001-08-13 | 2006-05-02 | E.I. Du Pont De Nemours And Company | Substituted 1H-dihydropyrazoles, their preparation and use |
| DE10215292A1 (de) | 2002-02-19 | 2003-08-28 | Bayer Cropscience Ag | Disubstitutierte Pyrazolylcarbocanilide |
| DE10349500A1 (de) | 2003-10-23 | 2005-06-02 | Bayer Cropscience Ag | Verfahren zum Herstellen von 2-Dihalogenacyl-3-amino-acrylsäureestern und 3-Dihalogenmethyl-pyrazol-4-carbonsäureestern |
| US20080108686A1 (en) | 2004-06-18 | 2008-05-08 | Basf Aktiengesellschaft | N-(Ortho-Phenyl)-1-Methyl-3-Difluoromethylpyrazole-4-Carboxanilides And Their Use As Fungicides |
| CN101133031B (zh) | 2005-02-25 | 2010-07-21 | 财团法人相模中央化学研究所 | 1-取代-3-氟代烷基吡唑-4-羧酸酯的制造方法 |
| DE102006039909A1 (de) | 2006-08-25 | 2008-03-13 | Bayer Cropscience Ag | Verfahren zum Herstellen von 3-Dihalomethyl-pyrazol-4-carbonsäurederivaten |
| JP5284266B2 (ja) * | 2006-11-03 | 2013-09-11 | ビーエーエスエフ ソシエタス・ヨーロピア | ジフルオロメチルピラゾリルカルボキシレートの調製方法 |
| EP2133341A1 (de) * | 2008-02-25 | 2009-12-16 | Bayer CropScience AG | Verfahren zur regioselektiven Synthese von 1-Alkyl-3-haloalkyl-pyrazol-4-carbonsäure-Derivaten |
-
2008
- 2008-03-10 EP EP08152532A patent/EP2100883A1/de not_active Ceased
-
2009
- 2009-02-26 MX MX2010008899A patent/MX2010008899A/es active IP Right Grant
- 2009-02-26 ES ES09719701T patent/ES2425972T3/es active Active
- 2009-02-26 WO PCT/EP2009/001354 patent/WO2009112157A1/de not_active Ceased
- 2009-02-26 CA CA2717805A patent/CA2717805C/en active Active
- 2009-02-26 PL PL09719701T patent/PL2257532T3/pl unknown
- 2009-02-26 JP JP2010550058A patent/JP5503562B2/ja active Active
- 2009-02-26 BR BRPI0909655-8A patent/BRPI0909655B1/pt active IP Right Grant
- 2009-02-26 EP EP09719701.6A patent/EP2257532B1/de active Active
- 2009-02-26 RU RU2010141358/04A patent/RU2498978C2/ru active
- 2009-02-26 KR KR1020107019740A patent/KR101652916B1/ko active Active
- 2009-02-26 CN CN2009801077008A patent/CN101970412B/zh active Active
- 2009-02-26 MY MYPI2010004113A patent/MY155478A/en unknown
- 2009-02-26 DK DK09719701.6T patent/DK2257532T3/da active
- 2009-02-26 US US12/921,719 patent/US8350053B2/en active Active
- 2009-03-09 TW TW098107485A patent/TWI440629B/zh active
-
2010
- 2010-08-09 IL IL207487A patent/IL207487A/en active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| DK2257532T3 (da) | 2013-09-08 |
| US20110028735A1 (en) | 2011-02-03 |
| RU2498978C2 (ru) | 2013-11-20 |
| CN101970412A (zh) | 2011-02-09 |
| JP5503562B2 (ja) | 2014-05-28 |
| PL2257532T3 (pl) | 2013-11-29 |
| EP2257532B1 (de) | 2013-05-29 |
| MX2010008899A (es) | 2010-10-25 |
| ES2425972T3 (es) | 2013-10-18 |
| TWI440629B (zh) | 2014-06-11 |
| EP2257532A1 (de) | 2010-12-08 |
| RU2010141358A (ru) | 2012-04-20 |
| MY155478A (en) | 2015-10-30 |
| KR20100137443A (ko) | 2010-12-30 |
| US8350053B2 (en) | 2013-01-08 |
| CN101970412B (zh) | 2013-06-26 |
| IL207487A (en) | 2014-06-30 |
| JP2011513446A (ja) | 2011-04-28 |
| IL207487A0 (en) | 2010-12-30 |
| CA2717805C (en) | 2016-02-23 |
| BRPI0909655B1 (pt) | 2018-06-05 |
| KR101652916B1 (ko) | 2016-08-31 |
| WO2009112157A1 (de) | 2009-09-17 |
| TW200951113A (en) | 2009-12-16 |
| CA2717805A1 (en) | 2009-09-17 |
| EP2100883A1 (de) | 2009-09-16 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B25A | Requested transfer of rights approved |
Owner name: BAYER INTELLECTUAL PROPERTY GMBH (DE) |
|
| B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
| B06A | Patent application procedure suspended [chapter 6.1 patent gazette] | ||
| B09A | Decision: intention to grant [chapter 9.1 patent gazette] | ||
| B16A | Patent or certificate of addition of invention granted [chapter 16.1 patent gazette] | ||
| B25A | Requested transfer of rights approved |