BRPI0913840A2 - 3-(n-heterociclil)-pirrolidinil-fenil-oxazolidinonas como agentes antibacterianos - Google Patents

3-(n-heterociclil)-pirrolidinil-fenil-oxazolidinonas como agentes antibacterianos

Info

Publication number: BRPI0913840A2
Authority: BR; Brazil
Prior art keywords: heterocyclyl; antibacterial agents; phenyl oxazolidinones; pyrrolidinyl phenyl; pyrrolidinyl
Prior art date: 2008-07-01

Application number

BRPI0913840A

Other languages

English (en)

Inventor

Albert Palomer

Antonio Guglietta

Montserrat Cano

Original Assignee

Ferrer Int

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2008-07-01

Filing date

2009-06-29

Publication date

2015-10-20

2009-06-29 Application filed by Ferrer Int filed Critical Ferrer Int

2015-10-20 Publication of BRPI0913840A2 publication Critical patent/BRPI0913840A2/pt

Links

YXOYOPPWBOGULQ-UHFFFAOYSA-N 3-phenyl-4-pyrrolidin-1-yl-1,3-oxazolidin-2-one Chemical class C=1C=CC=CC=1N1C(=O)OCC1N1CCCC1 YXOYOPPWBOGULQ-UHFFFAOYSA-N 0.000 title 1
239000003242 anti bacterial agent Substances 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Oncology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Communicable Diseases (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

BRPI0913840A 2008-07-01 2009-06-29 3-(n-heterociclil)-pirrolidinil-fenil-oxazolidinonas como agentes antibacterianos BRPI0913840A2 (pt)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP08159447A EP2141162A1 (en)	2008-07-01	2008-07-01	3-(n-heterocyclyl)-pyrrolidinyl-phenyl-oxazolidinones as antibacterial agents
PCT/EP2009/058126 WO2010000704A1 (en)	2008-07-01	2009-06-29	3-(n-heterocyclyl)-pyrrolidinyl-phenyl-oxazolidinones as antibacterial agents

Publications (1)

Publication Number	Publication Date
BRPI0913840A2 true BRPI0913840A2 (pt)	2015-10-20

Family

ID=40040120

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BRPI0913840A BRPI0913840A2 (pt)	2008-07-01	2009-06-29	3-(n-heterociclil)-pirrolidinil-fenil-oxazolidinonas como agentes antibacterianos

Country Status (17)

Country	Link
US (1)	US20110136829A1 (pt)
EP (2)	EP2141162A1 (pt)
JP (1)	JP2011526590A (pt)
KR (1)	KR20110036603A (pt)
CN (1)	CN102112472A (pt)
AR (1)	AR072390A1 (pt)
AT (1)	ATE555110T1 (pt)
AU (1)	AU2009265791A1 (pt)
BR (1)	BRPI0913840A2 (pt)
CA (1)	CA2729493A1 (pt)
CL (2)	CL2009001494A1 (pt)
MX (1)	MX2011000142A (pt)
PE (1)	PE20110107A1 (pt)
RU (1)	RU2011103484A (pt)
TW (1)	TW201004948A (pt)
UY (1)	UY31954A (pt)
WO (1)	WO2010000704A1 (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
KR101128029B1 (ko)	2010-03-08	2012-03-29	주식회사 레고켐 바이오사이언스	(ｒ)-3-(3-플루오로-4-(1-메틸-5,6-다이하이드로-1,2,4-트리아진-4(1ｈ)-일)페닐)-5-(치환된 메틸)옥사졸리딘-2-온 유도체의 제조방법
US10112924B2 (en) *	2015-12-02	2018-10-30	Astraea Therapeutics, Inc.	Piperdinyl nociceptin receptor compounds

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5688792A (en)	1994-08-16	1997-11-18	Pharmacia & Upjohn Company	Substituted oxazine and thiazine oxazolidinone antimicrobials
DE69522234T2 (de)	1994-10-26	2002-05-16	Pharmacia & Upjohn Co., Kalamazoo	Phenyloxazolidinone mit antimikrobieller wirkung

2008
- 2008-07-01 EP EP08159447A patent/EP2141162A1/en not_active Withdrawn
2009
- 2009-06-26 CL CL2009001494A patent/CL2009001494A1/es unknown
- 2009-06-29 BR BRPI0913840A patent/BRPI0913840A2/pt not_active IP Right Cessation
- 2009-06-29 EP EP09772404A patent/EP2324016B1/en not_active Not-in-force
- 2009-06-29 AT AT09772404T patent/ATE555110T1/de active
- 2009-06-29 KR KR1020117002615A patent/KR20110036603A/ko not_active Withdrawn
- 2009-06-29 RU RU2011103484/04A patent/RU2011103484A/ru not_active Application Discontinuation
- 2009-06-29 CA CA2729493A patent/CA2729493A1/en not_active Abandoned
- 2009-06-29 AR ARP090102399A patent/AR072390A1/es not_active Application Discontinuation
- 2009-06-29 MX MX2011000142A patent/MX2011000142A/es not_active Application Discontinuation
- 2009-06-29 AU AU2009265791A patent/AU2009265791A1/en not_active Abandoned
- 2009-06-29 JP JP2011515414A patent/JP2011526590A/ja active Pending
- 2009-06-29 WO PCT/EP2009/058126 patent/WO2010000704A1/en not_active Ceased
- 2009-06-29 PE PE2010001217A patent/PE20110107A1/es not_active Application Discontinuation
- 2009-06-29 US US13/001,963 patent/US20110136829A1/en not_active Abandoned
- 2009-06-29 CN CN2009801301821A patent/CN102112472A/zh active Pending
- 2009-06-30 TW TW098121938A patent/TW201004948A/zh unknown
- 2009-07-01 UY UY0001031954A patent/UY31954A/es unknown
2010
- 2010-12-28 CL CL2010001590A patent/CL2010001590A1/es unknown

Also Published As

Publication number	Publication date
TW201004948A (en)	2010-02-01
CL2009001494A1 (es)	2009-10-09
EP2324016A1 (en)	2011-05-25
KR20110036603A (ko)	2011-04-07
UY31954A (es)	2010-01-29
JP2011526590A (ja)	2011-10-13
US20110136829A1 (en)	2011-06-09
WO2010000704A1 (en)	2010-01-07
AR072390A1 (es)	2010-08-25
CN102112472A (zh)	2011-06-29
ATE555110T1 (de)	2012-05-15
EP2324016B1 (en)	2012-04-25
RU2011103484A (ru)	2012-08-10
PE20110107A1 (es)	2011-02-23
MX2011000142A (es)	2011-04-05
CL2010001590A1 (es)	2011-08-05
AU2009265791A1 (en)	2010-01-07
CA2729493A1 (en)	2010-01-07
EP2141162A1 (en)	2010-01-06

Legal Events

Date	Code	Title	Description
2015-12-08	B08F	Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]	Free format text: REFERENTE AS 4A, 5A E 6A ANUIDADES.
2016-04-05	B08K	Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]	Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2344 DE 08-12-2015 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.

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