BRPI0918955A2 - preparação sólida, e, método para estabilizar um composto, e para melhorar a dissoulução de um composto - Google Patents

preparação sólida, e, método para estabilizar um composto, e para melhorar a dissoulução de um composto

Info

Publication number: BRPI0918955A2
Authority: BR; Brazil
Prior art keywords: compound; dissoulution; stabilizing; improving; solid preparation
Prior art date: 2008-09-25

Application number

BRPI0918955A

Other languages

English (en)

Inventor

Junya Nomura

Kazuhiro Hirata

Yutaka Tanoue

Original Assignee

Takeda Pharmaceutical

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2008-09-25

Filing date

2009-09-25

Publication date

2015-12-01

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42059801&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0918955(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2009-09-25 Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical

2015-12-01 Publication of BRPI0918955A2 publication Critical patent/BRPI0918955A2/pt

Links

Classifications

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- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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BRPI0918955A 2008-09-25 2009-09-25 preparação sólida, e, método para estabilizar um composto, e para melhorar a dissoulução de um composto BRPI0918955A2 (pt)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US10010808P	2008-09-25	2008-09-25
PCT/JP2009/066690 WO2010035806A1 (ja)	2008-09-25	2009-09-25	固形医薬組成物

Publications (1)

Publication Number	Publication Date
BRPI0918955A2 true BRPI0918955A2 (pt)	2015-12-01

Family

ID=42059801

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BRPI0918955A BRPI0918955A2 (pt)	2008-09-25	2009-09-25	preparação sólida, e, método para estabilizar um composto, e para melhorar a dissoulução de um composto

Country Status (25)

Country	Link
US (1)	US9173849B2 (pt)
EP (1)	EP2332535A4 (pt)
JP (1)	JP5570426B2 (pt)
KR (1)	KR20110063557A (pt)
CN (2)	CN102223884B (pt)
AR (1)	AR073380A1 (pt)
AU (1)	AU2009297522A1 (pt)
BR (1)	BRPI0918955A2 (pt)
CA (1)	CA2738147C (pt)
CL (1)	CL2011000625A1 (pt)
CO (1)	CO6361934A2 (pt)
CR (1)	CR20110209A (pt)
EA (1)	EA201170483A1 (pt)
EC (1)	ECSP11011001A (pt)
GE (1)	GEP20146063B (pt)
IL (1)	IL211886A0 (pt)
MA (1)	MA32721B1 (pt)
MX (1)	MX2011003261A (pt)
NZ (1)	NZ592225A (pt)
PE (1)	PE20110844A1 (pt)
TW (1)	TW201014850A (pt)
UA (1)	UA102271C2 (pt)
UY (1)	UY32126A (pt)
WO (1)	WO2010035806A1 (pt)
ZA (1)	ZA201102715B (pt)

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2009
- 2009-09-16 UY UY0001032126A patent/UY32126A/es not_active Application Discontinuation
- 2009-09-16 TW TW098131167A patent/TW201014850A/zh unknown
- 2009-09-16 AR ARP090103548A patent/AR073380A1/es not_active Application Discontinuation
- 2009-09-25 KR KR1020117009104A patent/KR20110063557A/ko not_active Withdrawn
- 2009-09-25 BR BRPI0918955A patent/BRPI0918955A2/pt not_active IP Right Cessation
- 2009-09-25 EP EP09816220.9A patent/EP2332535A4/en not_active Withdrawn
- 2009-09-25 JP JP2010530880A patent/JP5570426B2/ja not_active Expired - Fee Related
- 2009-09-25 US US12/998,167 patent/US9173849B2/en not_active Expired - Fee Related
- 2009-09-25 CN CN200980146684.3A patent/CN102223884B/zh not_active Expired - Fee Related
- 2009-09-25 NZ NZ592225A patent/NZ592225A/en not_active IP Right Cessation
- 2009-09-25 WO PCT/JP2009/066690 patent/WO2010035806A1/ja not_active Ceased
- 2009-09-25 AU AU2009297522A patent/AU2009297522A1/en not_active Abandoned
- 2009-09-25 PE PE2011000787A patent/PE20110844A1/es not_active Application Discontinuation
- 2009-09-25 CN CN201410471654.2A patent/CN104306975A/zh active Pending
- 2009-09-25 MX MX2011003261A patent/MX2011003261A/es unknown
- 2009-09-25 EA EA201170483A patent/EA201170483A1/ru unknown
- 2009-09-25 UA UAA201105161A patent/UA102271C2/ru unknown
- 2009-09-25 CA CA2738147A patent/CA2738147C/en not_active Expired - Fee Related
- 2009-09-25 GE GEAP200912204A patent/GEP20146063B/en unknown
2011
- 2011-03-23 IL IL211886A patent/IL211886A0/en unknown
- 2011-03-24 CL CL2011000625A patent/CL2011000625A1/es unknown
- 2011-04-12 ZA ZA2011/02715A patent/ZA201102715B/en unknown
- 2011-04-20 MA MA33782A patent/MA32721B1/fr unknown
- 2011-04-25 CR CR20110209A patent/CR20110209A/es unknown
- 2011-04-25 EC EC2011011001A patent/ECSP11011001A/es unknown
- 2011-04-25 CO CO11050084A patent/CO6361934A2/es not_active Application Discontinuation

Also Published As

Publication number	Publication date
MX2011003261A (es)	2011-04-21
AU2009297522A1 (en)	2010-04-01
US20110229567A1 (en)	2011-09-22
PE20110844A1 (es)	2011-12-05
US9173849B2 (en)	2015-11-03
AR073380A1 (es)	2010-11-03
NZ592225A (en)	2012-06-29
ZA201102715B (en)	2012-07-25
UY32126A (es)	2010-04-30
EP2332535A1 (en)	2011-06-15
WO2010035806A1 (ja)	2010-04-01
GEP20146063B (en)	2014-03-25
KR20110063557A (ko)	2011-06-10
CN102223884B (zh)	2015-05-06
TW201014850A (en)	2010-04-16
IL211886A0 (en)	2011-06-30
EP2332535A4 (en)	2013-11-27
CO6361934A2 (es)	2012-01-20
CL2011000625A1 (es)	2011-07-08
JPWO2010035806A1 (ja)	2012-02-23
CA2738147A1 (en)	2010-04-01
EA201170483A1 (ru)	2011-10-31
CN104306975A (zh)	2015-01-28
MA32721B1 (fr)	2011-10-02
CA2738147C (en)	2016-10-11
JP5570426B2 (ja)	2014-08-13
CN102223884A (zh)	2011-10-19
UA102271C2 (en)	2013-06-25
ECSP11011001A (es)	2011-05-31
CR20110209A (es)	2011-05-27

Legal Events

Date	Code	Title	Description
2016-06-07	B08F	Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]	Free format text: REFERENTE A 6A ANUIDADE.
2016-09-27	B08K	Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]	Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2370 DE 07-06-2016 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.

Publication	Publication Date	Title
BRPI0918955A2 (pt)	2015-12-01	preparação sólida, e, método para estabilizar um composto, e para melhorar a dissoulução de um composto
BRPI0906906A2 (pt)	2015-07-21	Método para preparar um composto e composto
BRPI0909691A8 (pt)	2018-01-02	composto, método para preparar um composto, e, composição farmacêutica
BRPI0919937A2 (pt)	2016-02-16	composto, e, método para melhorar a atividade de adjuvante de uma imidazoquinolina
BRPI0917196A2 (pt)	2015-11-10	método para a preparação de um complexo, e, forma cristalina de um composto.
BR112012000623A2 (pt)	2016-02-10	composição de emulsão estabilizada, método, e, método para preparar uma composição de emulsão estabilizada
BRPI0911254A2 (pt)	2015-10-06	processo para a preparação de um composto
BRPI1010937A2 (pt)	2019-09-24	composto, uso de um composto, e, método para tratar câncer
BRPI0912384A2 (pt)	2015-10-13	composição, e, método para preparar uma composição
BRPI0906098A2 (pt)	2015-06-30	Método de preparação de um composto
BRPI1010775A2 (pt)	2016-03-22	composição, método para preparar uma composição, e, uso de uma composição.
BRPI0914040A2 (pt)	2015-11-03	composição de catalisador e método para transaminar um composto reagente
BRPI0914038A2 (pt)	2015-11-03	composição de catalisador e método para transaminar um composto reagente
BRPI1010933A2 (pt)	2016-04-05	processo para a preparação de um pó, e, composto
BRPI0909198A2 (pt)	2019-09-24	composto antifolato, composto, método para preparar um composto antifolato, composição farmacêutica, método para tratar
BRPI0815550A2 (pt)	2015-02-18	Método para estabilizar fenilefrina
BR112012001998A2 (pt)	2017-01-31	solução oftálmica, uso de um composto, e, método para preparação de uma solução oftálmica.
BRPI0908252A2 (pt)	2015-07-21	Processo para preparar um composto, e, uso de um composto
BRPI1012978A2 (pt)	2016-03-29	composição tópica, método para preparar a mesma, e, uso de um composto
BRPI0911897A2 (pt)	2015-07-28	Processo para a preparação de compostos, e, composto
BRPI1014691A2 (pt)	2015-08-25	Composto, e, processo para a preparação de um composto.
BR112014010479A2 (pt)	2017-04-25	composto, método para preparar um composto, método para a preparação de icotinib a partir de um composto e método para a preparação de cloridrato de icotinib a partir de um composto
BRPI0919410A2 (pt)	2015-12-15	método para produção de um composto oxidado
BR112012004173A2 (pt)	2017-05-30	"composto, composição, método para preparar uma composição, e, uso de um composto"
BR112013009590A2 (pt)	2016-07-19	composto, composição fungicida e método