CR20110209A - Composición farmacéutica sólida - Google Patents

Composición farmacéutica sólida

Info

Publication number
CR20110209A
CR20110209A CR20110209A CR20110209A CR20110209A CR 20110209 A CR20110209 A CR 20110209A CR 20110209 A CR20110209 A CR 20110209A CR 20110209 A CR20110209 A CR 20110209A CR 20110209 A CR20110209 A CR 20110209A
Authority
CR
Costa Rica
Prior art keywords
pharmaceutical composition
solid pharmaceutical
formula
calcium antagonist
represented
Prior art date
Application number
CR20110209A
Other languages
English (en)
Inventor
Kazuhiro Hirata
Junya Nomura
Yutaka Tanoue
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42059801&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CR20110209(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of CR20110209A publication Critical patent/CR20110209A/es

Links

Classifications

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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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Abstract

La presente invención se refiere a una preparación sólida que comprende un compuesto representado por la fórmula (i) que se muestra mas adelante, un agente de control de pH y un antagonista de calcio, el cual es superior en estabilidad y propiedad de disolución del compuesto (i) representado por la fórmula (i) y el antagonista de calcio.
CR20110209A 2008-09-25 2011-04-25 Composición farmacéutica sólida CR20110209A (es)

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ECSP11011001A (es) 2011-05-31
KR20110063557A (ko) 2011-06-10
NZ592225A (en) 2012-06-29
CN102223884A (zh) 2011-10-19
UA102271C2 (en) 2013-06-25
GEP20146063B (en) 2014-03-25
WO2010035806A1 (ja) 2010-04-01
CN102223884B (zh) 2015-05-06
BRPI0918955A2 (pt) 2015-12-01
ZA201102715B (en) 2012-07-25
MX2011003261A (es) 2011-04-21
UY32126A (es) 2010-04-30
JPWO2010035806A1 (ja) 2012-02-23
US20110229567A1 (en) 2011-09-22
EP2332535A4 (en) 2013-11-27
IL211886A0 (en) 2011-06-30
PE20110844A1 (es) 2011-12-05
AU2009297522A1 (en) 2010-04-01
EP2332535A1 (en) 2011-06-15
AR073380A1 (es) 2010-11-03
CA2738147C (en) 2016-10-11
CL2011000625A1 (es) 2011-07-08
MA32721B1 (fr) 2011-10-02
TW201014850A (en) 2010-04-16
US9173849B2 (en) 2015-11-03
CA2738147A1 (en) 2010-04-01
JP5570426B2 (ja) 2014-08-13
EA201170483A1 (ru) 2011-10-31
CN104306975A (zh) 2015-01-28

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