BRPI0920936A2 - 3-aminociclopentanocarboxamidas como moduladores de receptores de quimiocinas - Google Patents

3-aminociclopentanocarboxamidas como moduladores de receptores de quimiocinas Download PDF

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Publication number
BRPI0920936A2
BRPI0920936A2 BRPI0920936-0A BRPI0920936A BRPI0920936A2 BR PI0920936 A2 BRPI0920936 A2 BR PI0920936A2 BR PI0920936 A BRPI0920936 A BR PI0920936A BR PI0920936 A2 BRPI0920936 A2 BR PI0920936A2
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Brazil
Prior art keywords
hept
anhydrous
erythro
methyl
dideoxy
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BRPI0920936-0A
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English (en)
Portuguese (pt)
Inventor
Rajesh Venkateswaran Devraj
Wei Huang
Robert Owen Hughes
Donald Joseph Rogier Jr.
John Isidro Trujillo
Steve Ronald Turner
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Pfizer Inc
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Publication of BRPI0920936A2 publication Critical patent/BRPI0920936A2/pt

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
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    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

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BRPI0920936-0A 2008-11-26 2009-11-20 3-aminociclopentanocarboxamidas como moduladores de receptores de quimiocinas BRPI0920936A2 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US11805308P 2008-11-26 2008-11-26
US61/118,053 2008-11-26
PCT/IB2009/055232 WO2010061329A1 (en) 2008-11-26 2009-11-20 3-aminocyclopentanecarboxamides as chemokine receptor modulators

Publications (1)

Publication Number Publication Date
BRPI0920936A2 true BRPI0920936A2 (pt) 2020-08-11

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BRPI0920936-0A BRPI0920936A2 (pt) 2008-11-26 2009-11-20 3-aminociclopentanocarboxamidas como moduladores de receptores de quimiocinas

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US (2) US8293903B2 (pl)
EP (1) EP2370442B9 (pl)
JP (1) JP5108153B2 (pl)
KR (1) KR101374412B1 (pl)
CN (1) CN102227429B (pl)
AP (1) AP3113A (pl)
AU (1) AU2009321221B2 (pl)
BR (1) BRPI0920936A2 (pl)
CA (1) CA2743030C (pl)
CL (1) CL2011001223A1 (pl)
CO (1) CO6361921A2 (pl)
CR (1) CR20110275A (pl)
CU (1) CU24022B1 (pl)
CY (1) CY1114020T1 (pl)
DK (1) DK2370442T5 (pl)
DO (1) DOP2011000154A (pl)
EA (1) EA020470B1 (pl)
EC (1) ECSP11011081A (pl)
ES (1) ES2415430T3 (pl)
GE (1) GEP20146064B (pl)
HR (1) HRP20130409T2 (pl)
IL (1) IL212732A (pl)
MA (1) MA32834B1 (pl)
ME (1) ME01144B (pl)
MX (1) MX2011005526A (pl)
MY (1) MY152557A (pl)
NI (1) NI201100102A (pl)
NZ (1) NZ592919A (pl)
PE (1) PE20110831A1 (pl)
PL (1) PL2370442T3 (pl)
PT (1) PT2370442E (pl)
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SI (1) SI2370442T1 (pl)
SV (1) SV2011003923A (pl)
TN (1) TN2011000254A1 (pl)
UA (1) UA99978C2 (pl)
WO (1) WO2010061329A1 (pl)
ZA (1) ZA201104069B (pl)

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PL2370442T3 (pl) * 2008-11-26 2013-08-30 Pfizer 3-Aminocyklopentanokarboksamidy jako modulatory receptora chemokiny
KR101303963B1 (ko) * 2011-04-08 2013-09-05 재단법인 경기과학기술진흥원 (1r,2r,3r)-3-아미노사이클로펜탄-1,2-디올을 포함하는 항알러지용 조성물
KR102359214B1 (ko) 2014-04-04 2022-02-07 델 마 파마슈티컬스 폐의 비소세포 암종 및 난소암을 치료하기 위한 디안하이드로갈락티톨 및 이의 유사체 또는 유도체
JP2016029038A (ja) * 2014-07-17 2016-03-03 参天製薬株式会社 加齢黄斑変性の予防または治療剤
PE20190972A1 (es) * 2016-09-14 2019-07-09 Novartis Ag Combinacion de agonistas de fxr
TWI830733B (zh) * 2018-05-11 2024-02-01 中國大陸商迪哲(江蘇)醫藥有限公司 環戊烷化合物

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IL212732A (en) 2016-06-30
GEP20146064B (en) 2014-03-25
SI2370442T1 (sl) 2013-06-28
CN102227429B (zh) 2014-05-28
HK1161261A1 (en) 2012-08-24
EA020470B1 (ru) 2014-11-28
IL212732A0 (en) 2011-07-31
JP5108153B2 (ja) 2012-12-26
CU24022B1 (es) 2014-07-30
CY1114020T1 (el) 2016-07-27
MY152557A (en) 2014-10-31
HRP20130409T1 (en) 2013-06-30
EP2370442A1 (en) 2011-10-05
CO6361921A2 (es) 2012-01-20
US20130197008A1 (en) 2013-08-01
PL2370442T3 (pl) 2013-08-30
EP2370442B9 (en) 2013-09-04
US20110144129A1 (en) 2011-06-16
NZ592919A (en) 2013-05-31
HRP20130409T2 (hr) 2013-11-22
ECSP11011081A (es) 2011-12-30
AU2009321221A1 (en) 2010-06-03
RS52810B9 (sr) 2019-06-28
DK2370442T5 (da) 2013-09-23
CA2743030A1 (en) 2010-06-03
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