BRPI0921059A2 - derivados de bifenilacetamida - Google Patents

derivados de bifenilacetamida

Info

Publication number: BRPI0921059A2
Authority: BR; Brazil
Prior art keywords: atom; different; same; fluorine atom; alkyl
Prior art date: 2008-11-14

Application number

BRPI0921059-8A

Other languages

English (en)

Japanese (ja)

Inventor

Iwama Seiji

Tanaka Tomoyuki

Yajima Nana

Original Assignee

Dainippon Sumitomo Pharma Co., Ltd.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2008-11-14

Filing date

2009-11-13

Publication date

2018-10-16

2009-11-13 Application filed by Dainippon Sumitomo Pharma Co., Ltd. filed Critical Dainippon Sumitomo Pharma Co., Ltd.

2018-10-16 Publication of BRPI0921059A2 publication Critical patent/BRPI0921059A2/pt

Links

JCNHQILGQVWEKA-UHFFFAOYSA-N acetamide;1,1'-biphenyl Chemical class CC(N)=O.C1=CC=CC=C1C1=CC=CC=C1 JCNHQILGQVWEKA-UHFFFAOYSA-N 0.000 title 1
229910052731 fluorine Inorganic materials 0.000 abstract 5
125000001153 fluoro group Chemical group F* 0.000 abstract 5
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 4
125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 3
206010010904 Convulsion Diseases 0.000 abstract 3
125000004191 (C1-C6) alkoxy group Chemical group 0.000 abstract 2
229910052801 chlorine Inorganic materials 0.000 abstract 2
125000001309 chloro group Chemical group Cl* 0.000 abstract 2
WKBOTKDWSSQWDR-UHFFFAOYSA-N Bromine atom Chemical group [Br] WKBOTKDWSSQWDR-UHFFFAOYSA-N 0.000 abstract 1
206010061334 Partial seizures Diseases 0.000 abstract 1
239000003795 chemical substances by application Substances 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 abstract 1
125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
230000002265 prevention Effects 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
- C07C235/02—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton
- C07C235/32—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
- C07C235/34—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton containing six-membered aromatic rings having the nitrogen atoms of the carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C233/00—Carboxylic acid amides
- C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C233/02—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having nitrogen atoms of carboxamide groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
- C07C233/11—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having nitrogen atoms of carboxamide groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with carbon atoms of carboxamide groups bound to carbon atoms of an unsaturated carbon skeleton containing six-membered aromatic rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C255/00—Carboxylic acid nitriles
- C07C255/49—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
- C07C255/57—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and carboxyl groups, other than cyano groups, bound to the carbon skeleton
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C317/00—Sulfones; Sulfoxides
- C07C317/44—Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
- C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
- C07C323/62—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atom of at least one of the thio groups bound to a carbon atom of a six-membered aromatic ring of the carbon skeleton
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/02—Systems containing only non-condensed rings with a three-membered ring

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Engineering & Computer Science (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Biomedical Technology (AREA)
Chemical Kinetics & Catalysis (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Anesthesiology (AREA)
Psychiatry (AREA)
Pain & Pain Management (AREA)
Epidemiology (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

BRPI0921059-8A 2008-11-14 2009-11-13 derivados de bifenilacetamida BRPI0921059A2 (pt)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
JP2008-292682		2008-11-14
JP2008292682		2008-11-14
PCT/JP2009/069355 WO2010055911A1 (ja)	2008-11-14	2009-11-13	ビフェニルアセトアミド誘導体

Publications (1)

Publication Number	Publication Date
BRPI0921059A2 true BRPI0921059A2 (pt)	2018-10-16

Family

ID=42170041

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BRPI0921059-8A BRPI0921059A2 (pt)	2008-11-14	2009-11-13	derivados de bifenilacetamida

Country Status (13)

Country	Link
US (2)	US20110224304A1 (pt)
EP (1)	EP2374790A4 (pt)
JP (1)	JPWO2010055911A1 (pt)
KR (1)	KR20110086152A (pt)
CN (1)	CN102282124A (pt)
AU (1)	AU2009314879A1 (pt)
BR (1)	BRPI0921059A2 (pt)
CA (1)	CA2742679A1 (pt)
IL (1)	IL212683A0 (pt)
MX (1)	MX2011005098A (pt)
RU (1)	RU2011123777A (pt)
TW (1)	TW201023854A (pt)
WO (1)	WO2010055911A1 (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP2511273B8 (en) *	2011-04-15	2019-06-26	Hivih	Inhibitors of viral replication, their process of preparation and their therapeutical uses
US9199959B2 (en) *	2011-10-25	2015-12-01	Shionogi & Co., Ltd.	HIV replication inhibitor
KR101475115B1 (ko) *	2012-06-15	2014-12-23	중앙대학교 산학협력단	탐식작용 억제 효과를 가지는 자가 면역질환의 예방 또는 치료용 화합물
EP2821104A1 (en)	2013-07-05	2015-01-07	Laboratoire Biodim	Inhibitors of viral replication, their process of preparation and their therapeutical uses
US12624011B2 (en) *	2020-03-17	2026-05-12	Sumitomo Pharma Co., Ltd.	Oxadiazole derivative

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3049564A (en) *	1958-07-23	1962-08-14	Ici Ltd	2-phenylbenzamide derivatives and procedures for making same
US4277471A (en)	1979-03-12	1981-07-07	Eli Lilly And Company	1,1-Biphenyl-2-yl alkylamines, formulations and antiarrhythmic treatment
EP1042275B1 (en) *	1997-12-10	2005-11-09	Nps Pharmaceuticals, Inc.	Anticonvulsant and central nervous system-active bis(fluorophenyl)alkylamides
US7550474B2 (en)	2003-04-10	2009-06-23	Johnson & Johnson Pharmaceuticals Research & Development, L.L.C.	Substituted phenyl acetamides and their use as protease inhibitors
EP1704856A4 (en) *	2003-12-26	2009-08-19	Kyowa Hakko Kirin Co Ltd	PROTEIN INHIBITOR OF THE HSP90 FAMILY
JP5220359B2 (ja)	2007-07-23	2013-06-26	Ｎｔｎ株式会社	動圧軸受装置

2009
- 2009-11-13 US US13/129,394 patent/US20110224304A1/en not_active Abandoned
- 2009-11-13 RU RU2011123777/04A patent/RU2011123777A/ru not_active Application Discontinuation
- 2009-11-13 AU AU2009314879A patent/AU2009314879A1/en not_active Abandoned
- 2009-11-13 CN CN2009801545934A patent/CN102282124A/zh active Pending
- 2009-11-13 MX MX2011005098A patent/MX2011005098A/es not_active Application Discontinuation
- 2009-11-13 TW TW098138567A patent/TW201023854A/zh unknown
- 2009-11-13 JP JP2010537814A patent/JPWO2010055911A1/ja active Pending
- 2009-11-13 WO PCT/JP2009/069355 patent/WO2010055911A1/ja not_active Ceased
- 2009-11-13 CA CA2742679A patent/CA2742679A1/en not_active Abandoned
- 2009-11-13 KR KR1020117013390A patent/KR20110086152A/ko not_active Withdrawn
- 2009-11-13 EP EP09826157A patent/EP2374790A4/en not_active Withdrawn
- 2009-11-13 BR BRPI0921059-8A patent/BRPI0921059A2/pt not_active IP Right Cessation
2011
- 2011-05-04 IL IL212683A patent/IL212683A0/en unknown
2012
- 2012-02-07 US US13/368,325 patent/US20120142771A1/en not_active Abandoned

Also Published As

Publication number	Publication date
US20110224304A1 (en)	2011-09-15
KR20110086152A (ko)	2011-07-27
US20120142771A1 (en)	2012-06-07
CN102282124A (zh)	2011-12-14
WO2010055911A1 (ja)	2010-05-20
MX2011005098A (es)	2011-05-31
AU2009314879A1 (en)	2011-06-30
EP2374790A1 (en)	2011-10-12
TW201023854A (en)	2010-07-01
JPWO2010055911A1 (ja)	2012-04-12
EP2374790A4 (en)	2012-05-30
RU2011123777A (ru)	2012-12-20
CA2742679A1 (en)	2010-05-20
IL212683A0 (en)	2011-07-31

Legal Events

Date	Code	Title	Description
2018-10-30	B07D	Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]	Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS.
2018-10-30	B08F	Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]	Free format text: REFERENTE AS 5A, 6A, 7A, 8A E 9A ANUIDADES.
2019-03-19	B08K	Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]	Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2495 DE 30-10-2018 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.

Publication	Publication Date	Title
JO3116B1 (ar)	2017-09-20	مشتق بيرازولوكينولين كمثبطات ل pde9
UA110647C2 (uk)	2016-01-25	Похідне азолу, спосіб його одержання, проміжна сполука і хімічний агент, призначений для застосування в сільському господарстві і садівництві, і агент для захисту промислових матеріалів
EA200901609A1 (ru)	2010-06-30	Амиды пиразолкарбоновой кислоты, применимые в качестве микробиоцидов
MX2013002233A (es)	2013-05-06	Agente de control de plagas.
MY153910A (en)	2015-04-15	BICYCLIC y-AMINO ACID DERIVATIVE
MX2009009492A (es)	2009-09-15	Compuestos organicos biciclicos adecuados para el tratamiento de condiciones inflamatorias o alergicas.
MY142807A (en)	2011-01-14	Benzimidazole derivative and use thereof.
MX2010009736A (es)	2010-09-30	Compuesto heterociclico.
NO20084350L (no)	2008-10-16	Heterocykliske amider til anvendelse som farmasoytika
SMAP201100019A (it)	2011-05-06	Composti organici.
HRP20130653T1 (en)	2013-08-31	Pyrrole compounds
EA201491936A1 (ru)	2015-03-31	Азотсодержащее гетероциклическое соединение
WO2009051244A1 (ja)	2009-04-23	複素環化合物
WO2008126858A1 (ja)	2008-10-23	アミド化合物の製造方法
WO2009156861A8 (en)	2012-04-26	Substituted pyrimidone derivatives
EA201301040A1 (ru)	2014-01-30	Гетероциклическое соединение и его применение
MY169179A (en)	2019-02-25	Novel piperidine compound or salt thereof
CR9830A (es)	2008-05-21	Compuestos de amino-5-[4-(difluorometoxi)fenil]-5-fenilimidazolona para la inhibicion de la b-secretasa
UY31834A (es)	2010-01-05	Nuevo ácido l-glutámico y derivado l-glutamina (iii), uso de los mismos y método para obtenerlos
MX368178B (es)	2019-09-23	Compuestos de ácido dimetilbenzoico.
WO2010003084A3 (en)	2010-03-25	Phosphodiesterase 4 inhibitors
WO2013037705A3 (en)	2013-06-06	Aniline derivatives,their preparation and their therapeutic application
EA201100920A1 (ru)	2012-01-30	Новые гербициды
AR066268A1 (es)	2009-08-05	Compuesto de imidazol sustituido y su uso
ES2553030T3 (es)	2015-12-03	Compuestos plaguicidas