BRPI0921084A2 - compostos, composição farmacêutica, uso de um composto, e, método de tratamento de dor - Google Patents
compostos, composição farmacêutica, uso de um composto, e, método de tratamento de dorInfo
- Publication number
- BRPI0921084A2 BRPI0921084A2 BRPI0921084A BRPI0921084A BRPI0921084A2 BR PI0921084 A2 BRPI0921084 A2 BR PI0921084A2 BR PI0921084 A BRPI0921084 A BR PI0921084A BR PI0921084 A BRPI0921084 A BR PI0921084A BR PI0921084 A2 BRPI0921084 A2 BR PI0921084A2
- Authority
- BR
- Brazil
- Prior art keywords
- compounds
- compound
- pharmaceutical composition
- treatment method
- pain treatment
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title 2
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pain & Pain Management (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Rheumatology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP08168286 | 2008-11-04 | ||
| PCT/EP2009/064490 WO2010052198A1 (en) | 2008-11-04 | 2009-11-03 | ( pyrrolidin-2 -yl) phenyl derivatives for use in the treatment of pain |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0921084A2 true BRPI0921084A2 (pt) | 2015-12-15 |
Family
ID=40251652
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0921084A BRPI0921084A2 (pt) | 2008-11-04 | 2009-11-03 | compostos, composição farmacêutica, uso de um composto, e, método de tratamento de dor |
Country Status (13)
| Country | Link |
|---|---|
| EP (1) | EP2356105B1 (pt) |
| JP (1) | JP5642690B2 (pt) |
| KR (2) | KR20150028342A (pt) |
| CN (1) | CN102203077B (pt) |
| AR (1) | AR074085A1 (pt) |
| AU (1) | AU2009312855B2 (pt) |
| BR (1) | BRPI0921084A2 (pt) |
| CA (1) | CA2741332C (pt) |
| IL (1) | IL212302A0 (pt) |
| MX (1) | MX2011004750A (pt) |
| TW (1) | TW201022233A (pt) |
| WO (1) | WO2010052198A1 (pt) |
| ZA (1) | ZA201103134B (pt) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2011076723A1 (en) | 2009-12-22 | 2011-06-30 | N.V. Organon | Amino-heteroaryl derivatives as hcn blockers |
| KR20140014184A (ko) * | 2011-02-25 | 2014-02-05 | 아이알엠 엘엘씨 | Trk 억제제로서의 화합물 및 조성물 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PL200427B1 (pl) * | 1999-05-21 | 2009-01-30 | Abbott Lab | Związek aminoazacykliczny, kompozycja farmaceutyczna go zawierająca i jego zastosowanie |
| EP1297136A2 (en) * | 2000-05-24 | 2003-04-02 | Akzo Nobel N.V. | Full length human hcn1 ih channel subunit and variants |
| MX2007004661A (es) * | 2004-10-18 | 2007-06-22 | Lilly Co Eli | Derivados de 1-(hetero)aril-3-amino-pirrolidina para usarse como antagonistas del receptor mglur3. |
-
2009
- 2009-10-27 TW TW098136332A patent/TW201022233A/zh unknown
- 2009-11-03 EP EP09744410.3A patent/EP2356105B1/en active Active
- 2009-11-03 KR KR20157002833A patent/KR20150028342A/ko not_active Ceased
- 2009-11-03 AU AU2009312855A patent/AU2009312855B2/en not_active Ceased
- 2009-11-03 JP JP2011533753A patent/JP5642690B2/ja not_active Expired - Fee Related
- 2009-11-03 AR ARP090104238A patent/AR074085A1/es unknown
- 2009-11-03 BR BRPI0921084A patent/BRPI0921084A2/pt not_active Application Discontinuation
- 2009-11-03 CN CN200980143666.XA patent/CN102203077B/zh not_active Expired - Fee Related
- 2009-11-03 CA CA2741332A patent/CA2741332C/en not_active Expired - Fee Related
- 2009-11-03 MX MX2011004750A patent/MX2011004750A/es active IP Right Grant
- 2009-11-03 KR KR1020117010949A patent/KR101526643B1/ko not_active Expired - Fee Related
- 2009-11-03 WO PCT/EP2009/064490 patent/WO2010052198A1/en not_active Ceased
-
2011
- 2011-04-13 IL IL212302A patent/IL212302A0/en unknown
- 2011-04-28 ZA ZA2011/03134A patent/ZA201103134B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| AU2009312855A1 (en) | 2010-05-14 |
| AR074085A1 (es) | 2010-12-22 |
| EP2356105A1 (en) | 2011-08-17 |
| ZA201103134B (en) | 2012-01-25 |
| CA2741332A1 (en) | 2010-05-14 |
| AU2009312855B2 (en) | 2014-05-01 |
| TW201022233A (en) | 2010-06-16 |
| JP5642690B2 (ja) | 2014-12-17 |
| KR101526643B1 (ko) | 2015-06-05 |
| CA2741332C (en) | 2016-07-12 |
| IL212302A0 (en) | 2011-06-30 |
| WO2010052198A1 (en) | 2010-05-14 |
| CN102203077A (zh) | 2011-09-28 |
| CN102203077B (zh) | 2014-07-09 |
| JP2012507490A (ja) | 2012-03-29 |
| EP2356105B1 (en) | 2013-04-10 |
| KR20110082174A (ko) | 2011-07-18 |
| KR20150028342A (ko) | 2015-03-13 |
| MX2011004750A (es) | 2011-06-01 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B25A | Requested transfer of rights approved |
Owner name: MSD OSS B.V. (NL) |
|
| B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
| B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] | ||
| B25A | Requested transfer of rights approved |
Owner name: ORGANON BIOSCIENCES NEDERLAND B.V. (NL) |
|
| B25A | Requested transfer of rights approved |
Owner name: MERCK SHARP AND DOHME B.V. (NL) |
|
| B07E | Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette] | ||
| B11B | Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements |