BRPI0921084A2 - compostos, composição farmacêutica, uso de um composto, e, método de tratamento de dor - Google Patents

compostos, composição farmacêutica, uso de um composto, e, método de tratamento de dor

Info

Publication number
BRPI0921084A2
BRPI0921084A2 BRPI0921084A BRPI0921084A BRPI0921084A2 BR PI0921084 A2 BRPI0921084 A2 BR PI0921084A2 BR PI0921084 A BRPI0921084 A BR PI0921084A BR PI0921084 A BRPI0921084 A BR PI0921084A BR PI0921084 A2 BRPI0921084 A2 BR PI0921084A2
Authority
BR
Brazil
Prior art keywords
compounds
compound
pharmaceutical composition
treatment method
pain treatment
Prior art date
Application number
BRPI0921084A
Other languages
English (en)
Inventor
Ashvinkumar Dhirubhai Mistry
John Kinnaird Ferguson Maclean
Ronald Palin
Simon James Anthony Grove
Original Assignee
Organon Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Organon Nv filed Critical Organon Nv
Publication of BRPI0921084A2 publication Critical patent/BRPI0921084A2/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/10Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BRPI0921084A 2008-11-04 2009-11-03 compostos, composição farmacêutica, uso de um composto, e, método de tratamento de dor BRPI0921084A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP08168286 2008-11-04
PCT/EP2009/064490 WO2010052198A1 (en) 2008-11-04 2009-11-03 ( pyrrolidin-2 -yl) phenyl derivatives for use in the treatment of pain

Publications (1)

Publication Number Publication Date
BRPI0921084A2 true BRPI0921084A2 (pt) 2015-12-15

Family

ID=40251652

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0921084A BRPI0921084A2 (pt) 2008-11-04 2009-11-03 compostos, composição farmacêutica, uso de um composto, e, método de tratamento de dor

Country Status (13)

Country Link
EP (1) EP2356105B1 (pt)
JP (1) JP5642690B2 (pt)
KR (2) KR20150028342A (pt)
CN (1) CN102203077B (pt)
AR (1) AR074085A1 (pt)
AU (1) AU2009312855B2 (pt)
BR (1) BRPI0921084A2 (pt)
CA (1) CA2741332C (pt)
IL (1) IL212302A0 (pt)
MX (1) MX2011004750A (pt)
TW (1) TW201022233A (pt)
WO (1) WO2010052198A1 (pt)
ZA (1) ZA201103134B (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2011076723A1 (en) 2009-12-22 2011-06-30 N.V. Organon Amino-heteroaryl derivatives as hcn blockers
KR20140014184A (ko) * 2011-02-25 2014-02-05 아이알엠 엘엘씨 Trk 억제제로서의 화합물 및 조성물

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL200427B1 (pl) * 1999-05-21 2009-01-30 Abbott Lab Związek aminoazacykliczny, kompozycja farmaceutyczna go zawierająca i jego zastosowanie
EP1297136A2 (en) * 2000-05-24 2003-04-02 Akzo Nobel N.V. Full length human hcn1 ih channel subunit and variants
MX2007004661A (es) * 2004-10-18 2007-06-22 Lilly Co Eli Derivados de 1-(hetero)aril-3-amino-pirrolidina para usarse como antagonistas del receptor mglur3.

Also Published As

Publication number Publication date
AU2009312855A1 (en) 2010-05-14
AR074085A1 (es) 2010-12-22
EP2356105A1 (en) 2011-08-17
ZA201103134B (en) 2012-01-25
CA2741332A1 (en) 2010-05-14
AU2009312855B2 (en) 2014-05-01
TW201022233A (en) 2010-06-16
JP5642690B2 (ja) 2014-12-17
KR101526643B1 (ko) 2015-06-05
CA2741332C (en) 2016-07-12
IL212302A0 (en) 2011-06-30
WO2010052198A1 (en) 2010-05-14
CN102203077A (zh) 2011-09-28
CN102203077B (zh) 2014-07-09
JP2012507490A (ja) 2012-03-29
EP2356105B1 (en) 2013-04-10
KR20110082174A (ko) 2011-07-18
KR20150028342A (ko) 2015-03-13
MX2011004750A (es) 2011-06-01

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Legal Events

Date Code Title Description
B25A Requested transfer of rights approved

Owner name: MSD OSS B.V. (NL)

B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B25A Requested transfer of rights approved

Owner name: ORGANON BIOSCIENCES NEDERLAND B.V. (NL)

B25A Requested transfer of rights approved

Owner name: MERCK SHARP AND DOHME B.V. (NL)

B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]
B11B Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements