BRPI0921084A2 - compostos, composição farmacêutica, uso de um composto, e, método de tratamento de dor - Google Patents

compostos, composição farmacêutica, uso de um composto, e, método de tratamento de dor

Info

Publication number
BRPI0921084A2
BRPI0921084A2 BRPI0921084A BRPI0921084A BRPI0921084A2 BR PI0921084 A2 BRPI0921084 A2 BR PI0921084A2 BR PI0921084 A BRPI0921084 A BR PI0921084A BR PI0921084 A BRPI0921084 A BR PI0921084A BR PI0921084 A2 BRPI0921084 A2 BR PI0921084A2
Authority
BR
Brazil
Prior art keywords
compounds
compound
pharmaceutical composition
treatment method
pain treatment
Prior art date
Application number
BRPI0921084A
Other languages
English (en)
Inventor
Ashvinkumar Dhirubhai Mistry
John Kinnaird Ferguson Maclean
Ronald Palin
Simon James Anthony Grove
Original Assignee
Organon Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Organon Nv filed Critical Organon Nv
Publication of BRPI0921084A2 publication Critical patent/BRPI0921084A2/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BRPI0921084A 2008-11-04 2009-11-03 compostos, composição farmacêutica, uso de um composto, e, método de tratamento de dor BRPI0921084A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP08168286 2008-11-04
PCT/EP2009/064490 WO2010052198A1 (en) 2008-11-04 2009-11-03 ( pyrrolidin-2 -yl) phenyl derivatives for use in the treatment of pain

Publications (1)

Publication Number Publication Date
BRPI0921084A2 true BRPI0921084A2 (pt) 2015-12-15

Family

ID=40251652

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0921084A BRPI0921084A2 (pt) 2008-11-04 2009-11-03 compostos, composição farmacêutica, uso de um composto, e, método de tratamento de dor

Country Status (13)

Country Link
EP (1) EP2356105B1 (pt)
JP (1) JP5642690B2 (pt)
KR (2) KR101526643B1 (pt)
CN (1) CN102203077B (pt)
AR (1) AR074085A1 (pt)
AU (1) AU2009312855B2 (pt)
BR (1) BRPI0921084A2 (pt)
CA (1) CA2741332C (pt)
IL (1) IL212302A0 (pt)
MX (1) MX2011004750A (pt)
TW (1) TW201022233A (pt)
WO (1) WO2010052198A1 (pt)
ZA (1) ZA201103134B (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR079543A1 (es) 2009-12-22 2012-02-01 Organon Nv Derivados de amino-heteroarilo
BR112013021638A2 (pt) * 2011-02-25 2016-08-02 Irm Llc "compostos inibidores de trk, seu uso e composições que os compreendem"

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2226844T3 (es) * 1999-05-21 2005-04-01 Abbott Laboratories Aminoazaciclos heterociclicos sustituidos utiles como agentes activos sobre el sistema nervioso central.
US7329510B2 (en) * 2000-05-24 2008-02-12 N.V. Organon Full length human HCN1Ih channel subunit and variants
ES2336130T3 (es) * 2004-10-18 2010-04-08 Eli Lilly And Company Derivados 1-(hetero)aril-3-amino-pirrolidina para uso como antagonistas del receptor de mglur3.

Also Published As

Publication number Publication date
KR20110082174A (ko) 2011-07-18
IL212302A0 (en) 2011-06-30
CA2741332C (en) 2016-07-12
CN102203077A (zh) 2011-09-28
JP2012507490A (ja) 2012-03-29
KR20150028342A (ko) 2015-03-13
EP2356105B1 (en) 2013-04-10
EP2356105A1 (en) 2011-08-17
WO2010052198A1 (en) 2010-05-14
AR074085A1 (es) 2010-12-22
TW201022233A (en) 2010-06-16
ZA201103134B (en) 2012-01-25
KR101526643B1 (ko) 2015-06-05
AU2009312855B2 (en) 2014-05-01
JP5642690B2 (ja) 2014-12-17
CN102203077B (zh) 2014-07-09
AU2009312855A1 (en) 2010-05-14
CA2741332A1 (en) 2010-05-14
MX2011004750A (es) 2011-06-01

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Legal Events

Date Code Title Description
B25A Requested transfer of rights approved

Owner name: MSD OSS B.V. (NL)

B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B25A Requested transfer of rights approved

Owner name: ORGANON BIOSCIENCES NEDERLAND B.V. (NL)

B25A Requested transfer of rights approved

Owner name: MERCK SHARP AND DOHME B.V. (NL)

B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]
B11B Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements