BRPI0923675A2 - formulação para administração de medicamento com baixa quantidade de lipídeos por via transmucosal oral - Google Patents
formulação para administração de medicamento com baixa quantidade de lipídeos por via transmucosal oralInfo
- Publication number
- BRPI0923675A2 BRPI0923675A2 BRPI0923675A BRPI0923675A BRPI0923675A2 BR PI0923675 A2 BRPI0923675 A2 BR PI0923675A2 BR PI0923675 A BRPI0923675 A BR PI0923675A BR PI0923675 A BRPI0923675 A BR PI0923675A BR PI0923675 A2 BRPI0923675 A2 BR PI0923675A2
- Authority
- BR
- Brazil
- Prior art keywords
- lipid
- formulation
- drug administration
- lowering drug
- oral transmucosal
- Prior art date
Links
- 239000003524 antilipemic agent Substances 0.000 title 1
- 238000001647 drug administration Methods 0.000 title 1
- 238000009472 formulation Methods 0.000 title 1
- 239000000203 mixture Substances 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/006—Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Nutrition Science (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Physiology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Vascular Medicine (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0858947A FR2940116B1 (fr) | 2008-12-22 | 2008-12-22 | Formulation pour l'administration d'hypolipemiant par voie trans-muqueuse buccale |
| PCT/FR2009/052591 WO2010072950A1 (fr) | 2008-12-22 | 2009-12-17 | Formulation pour l'administration d'hypolipemiants par voie trans-muqueuse buccale |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| BRPI0923675A2 true BRPI0923675A2 (pt) | 2016-01-19 |
| BRPI0923675A8 BRPI0923675A8 (pt) | 2018-05-29 |
Family
ID=40872056
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0923675A BRPI0923675A8 (pt) | 2008-12-22 | 2009-12-17 | formulação para a administração de hipolipemiantes por via transmucosa oral |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US8889663B2 (pt) |
| EP (1) | EP2379054A1 (pt) |
| JP (1) | JP5529165B2 (pt) |
| CN (1) | CN102264346A (pt) |
| BR (1) | BRPI0923675A8 (pt) |
| FR (1) | FR2940116B1 (pt) |
| MX (1) | MX2011006797A (pt) |
| RU (1) | RU2528897C2 (pt) |
| WO (1) | WO2010072950A1 (pt) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2906140B1 (fr) * | 2006-09-22 | 2008-12-05 | Philippe Perovitch | Forme galenique pour l'administration par voie trans-muqueuse de principes actifs |
| GB2497728A (en) * | 2011-12-14 | 2013-06-26 | Londonpharma Ltd | Statin formulations for transmucosal delivery |
| FR3000896B1 (fr) * | 2013-01-14 | 2016-08-26 | Philippe Perovitch | Forme galenique pour l'administration de principe(s) actif(s) permettant l'induction acceleree du sommeil et/ou le traitement des troubles du sommeil |
| FR3031668A1 (fr) | 2015-01-20 | 2016-07-22 | Philippe Perovitch | Dispositif d'administration d'un principe actif par voie per-muqueuse buccale. |
| FR3053244A1 (fr) | 2016-07-01 | 2018-01-05 | Philippe Perovitch | Dispositif d'administration d'au moins un principe actif par voie per-muqueuse buccale. |
| US20260027048A1 (en) * | 2022-06-03 | 2026-01-29 | Polaryx Therapeutics, Inc. | Gemfibrozil formulation |
| CN116270507A (zh) * | 2023-03-02 | 2023-06-23 | 青岛海洋生物医药研究院股份有限公司 | 一种含脂蛋白脂酶刺激剂的舌下含片及其制备方法和应用 |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5582838A (en) * | 1994-12-22 | 1996-12-10 | Merck & Co., Inc. | Controlled release drug suspension delivery device |
| US20030077229A1 (en) * | 1997-10-01 | 2003-04-24 | Dugger Harry A. | Buccal, polar and non-polar spray or capsule containing cardiovascular or renal drugs |
| US20030095925A1 (en) * | 1997-10-01 | 2003-05-22 | Dugger Harry A. | Buccal, polar and non-polar spray or capsule containing drugs for treating metabolic disorders |
| DE19929197A1 (de) * | 1999-06-25 | 2000-12-28 | Novosis Pharma Ag | Transdermalsysteme zur Abgabe von 5-HT3-Rezeptor-Antagonisten und ihre Verwendung zur antiemitischen Behandlung |
| US20070225379A1 (en) * | 2001-08-03 | 2007-09-27 | Carrara Dario Norberto R | Transdermal delivery of systemically active central nervous system drugs |
| US7033612B2 (en) * | 2003-01-03 | 2006-04-25 | Kang David S | Composition and method for treating age-related disorders |
| JP2004231603A (ja) * | 2003-01-31 | 2004-08-19 | Hideji Watanabe | コエンザイムq10を主成分とする口腔内塗布剤及びその製造方法 |
| US20050281868A1 (en) * | 2004-06-21 | 2005-12-22 | Fairfield Clinical Trials, Llc | Transdermal delivery system for statin combination therapy |
| BRPI0501708A (pt) * | 2005-05-10 | 2007-05-02 | Jean Marc Millet | dispositivo de liberação lenta por processo transdérmico de um medicamento contra o excesso de colesterol e método de produção de um dispositivo transdérmico |
| CN1778296B (zh) * | 2005-07-19 | 2010-04-14 | 淮北辉克药业有限公司 | 他汀类药物的长效制剂 |
| FR2906140B1 (fr) * | 2006-09-22 | 2008-12-05 | Philippe Perovitch | Forme galenique pour l'administration par voie trans-muqueuse de principes actifs |
| US20080249120A1 (en) * | 2006-11-22 | 2008-10-09 | Glenmark Pharmaceuticals Limited | Pharmaceutical compositions |
| FR2910317B1 (fr) * | 2006-12-21 | 2009-02-13 | Philippe Perovitch | Forme galenique pour l'administration par voie transmuqueuse de paracetamol |
| CA2673049C (en) * | 2006-12-22 | 2016-02-23 | Novadel Pharma Inc. | Stable anti-nausea oral spray formulations and methods |
| JP2010526054A (ja) * | 2007-05-01 | 2010-07-29 | シグモイド・ファーマ・リミテッド | 併用医薬組成物 |
| FR2947729B1 (fr) * | 2009-07-10 | 2012-01-20 | Philippe Perovitch | Composition pharmaceutique pour le traitement du diabete de type ii par voie trans-muqueuse buccale |
-
2008
- 2008-12-22 FR FR0858947A patent/FR2940116B1/fr not_active Expired - Fee Related
-
2009
- 2009-12-17 BR BRPI0923675A patent/BRPI0923675A8/pt not_active Application Discontinuation
- 2009-12-17 MX MX2011006797A patent/MX2011006797A/es active IP Right Grant
- 2009-12-17 JP JP2011542870A patent/JP5529165B2/ja not_active Expired - Fee Related
- 2009-12-17 US US13/141,597 patent/US8889663B2/en not_active Expired - Fee Related
- 2009-12-17 EP EP09805727A patent/EP2379054A1/fr not_active Withdrawn
- 2009-12-17 CN CN200980152796XA patent/CN102264346A/zh active Pending
- 2009-12-17 WO PCT/FR2009/052591 patent/WO2010072950A1/fr not_active Ceased
- 2009-12-17 RU RU2011130508/15A patent/RU2528897C2/ru not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| JP2012513454A (ja) | 2012-06-14 |
| JP5529165B2 (ja) | 2014-06-25 |
| FR2940116B1 (fr) | 2012-07-06 |
| RU2528897C2 (ru) | 2014-09-20 |
| US8889663B2 (en) | 2014-11-18 |
| EP2379054A1 (fr) | 2011-10-26 |
| CN102264346A (zh) | 2011-11-30 |
| WO2010072950A1 (fr) | 2010-07-01 |
| RU2011130508A (ru) | 2013-01-27 |
| MX2011006797A (es) | 2011-09-06 |
| FR2940116A1 (fr) | 2010-06-25 |
| US20110257149A1 (en) | 2011-10-20 |
| BRPI0923675A8 (pt) | 2018-05-29 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B06F | Objections, documents and/or translations needed after an examination request according art. 34 industrial property law | ||
| B06T | Formal requirements before examination | ||
| B07D | Technical examination (opinion) related to article 229 of industrial property law |
Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS. |
|
| B07E | Notice of approval relating to section 229 industrial property law | ||
| B07A | Technical examination (opinion): publication of technical examination (opinion) | ||
| B09B | Decision: refusal | ||
| B09B | Decision: refusal |
Free format text: MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL |