BRPI1008340A2 - forma cristalina, composição farmacêutica, processos para fabricar uma composição farmacêutica e uma forma, uso da forma cristalina, e, método para tratar uma condição de doença - Google Patents

forma cristalina, composição farmacêutica, processos para fabricar uma composição farmacêutica e uma forma, uso da forma cristalina, e, método para tratar uma condição de doença

Info

Publication number
BRPI1008340A2
BRPI1008340A2 BRPI1008340A BRPI1008340A BRPI1008340A2 BR PI1008340 A2 BRPI1008340 A2 BR PI1008340A2 BR PI1008340 A BRPI1008340 A BR PI1008340A BR PI1008340 A BRPI1008340 A BR PI1008340A BR PI1008340 A2 BRPI1008340 A2 BR PI1008340A2
Authority
BR
Brazil
Prior art keywords
pharmaceutical composition
crystalline form
treating
processes
manufacturing
Prior art date
Application number
BRPI1008340A
Other languages
English (en)
Inventor
David Peter Hoile
Karin Assarsson
Sharon Ann Bowden
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of BRPI1008340A2 publication Critical patent/BRPI1008340A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965—Non-condensed pyrazines
    • A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BRPI1008340A 2009-02-13 2010-02-11 forma cristalina, composição farmacêutica, processos para fabricar uma composição farmacêutica e uma forma, uso da forma cristalina, e, método para tratar uma condição de doença BRPI1008340A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0902406.8A GB0902406D0 (en) 2009-02-13 2009-02-13 Crystalline polymorphic form
PCT/GB2010/050216 WO2010092386A1 (en) 2009-02-13 2010-02-11 Crystalline polymorphic form 631

Publications (1)

Publication Number Publication Date
BRPI1008340A2 true BRPI1008340A2 (pt) 2016-02-23

Family

ID=40548139

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI1008340A BRPI1008340A2 (pt) 2009-02-13 2010-02-11 forma cristalina, composição farmacêutica, processos para fabricar uma composição farmacêutica e uma forma, uso da forma cristalina, e, método para tratar uma condição de doença

Country Status (15)

Country Link
US (1) US8093252B2 (pt)
EP (1) EP2396317A1 (pt)
JP (1) JP2012517990A (pt)
KR (1) KR20110120941A (pt)
CN (1) CN102395580B (pt)
AR (1) AR075418A1 (pt)
AU (1) AU2010212605A1 (pt)
BR (1) BRPI1008340A2 (pt)
CA (1) CA2749994A1 (pt)
GB (1) GB0902406D0 (pt)
MX (1) MX2011008576A (pt)
RU (1) RU2011135628A (pt)
TW (1) TW201040161A (pt)
UY (1) UY32446A (pt)
WO (1) WO2010092386A1 (pt)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW200600086A (en) * 2004-06-05 2006-01-01 Astrazeneca Ab Chemical compound
TW200714597A (en) * 2005-05-27 2007-04-16 Astrazeneca Ab Chemical compounds
TW200825060A (en) * 2006-10-26 2008-06-16 Astrazeneca Ab Chemical compounds
MX2011001333A (es) * 2008-08-04 2011-03-15 Astrazeneca Ab Derivados de pirazolo [3, 4] pirimidin-4-ilo y sus usos para tratar la diabetes y obesidad.
GB0902434D0 (en) * 2009-02-13 2009-04-01 Astrazeneca Ab Chemical process
WO2010116176A1 (en) * 2009-04-09 2010-10-14 Astrazeneca Ab Pyrazolo [4, 5-e] pyrimidine derivative and its use to treat diabetes and obesity
AR076220A1 (es) 2009-04-09 2011-05-26 Astrazeneca Ab Derivados de pirazol [4,5 - e] pirimidina
CN118265703A (zh) 2021-09-02 2024-06-28 康杜英国管理有限公司 3-{[5-(氮杂环丁烷-1-基羰基)吡嗪-2-基]氧基}-5-{[(1s)-1-甲基-2-(甲氧基)乙基]氧基)-n-(5-甲基吡嗪-2-基)苯甲酰胺的治疗性共晶

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GB0902434D0 (en) 2009-02-13 2009-04-01 Astrazeneca Ab Chemical process
AR076220A1 (es) 2009-04-09 2011-05-26 Astrazeneca Ab Derivados de pirazol [4,5 - e] pirimidina

Also Published As

Publication number Publication date
EP2396317A1 (en) 2011-12-21
US8093252B2 (en) 2012-01-10
AR075418A1 (es) 2011-03-30
CN102395580A (zh) 2012-03-28
MX2011008576A (es) 2011-09-06
CA2749994A1 (en) 2010-08-19
UY32446A (es) 2010-09-30
RU2011135628A (ru) 2013-03-20
CN102395580B (zh) 2014-03-12
WO2010092386A1 (en) 2010-08-19
JP2012517990A (ja) 2012-08-09
GB0902406D0 (en) 2009-04-01
KR20110120941A (ko) 2011-11-04
US20100210621A1 (en) 2010-08-19
TW201040161A (en) 2010-11-16
AU2010212605A1 (en) 2011-08-04

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