CA1034953A - Pyrazol-5-ones - Google Patents

Pyrazol-5-ones

Info

Publication number: CA1034953A
Authority: CA; Canada
Prior art keywords: pyrazol; ones
Prior art date: 1973-04-17
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired

Application number

CA197,660A

Other languages

English (en)

French (fr)

Inventor

Harald Horstmann

Eike Moller

Karl Meng

Egbert Wehinger

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Bayer AG

Original Assignee

Bayer AG

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1973-04-17

Filing date

1974-04-17

Publication date

1978-07-18

1973-04-17 Priority claimed from DE2319280A external-priority patent/DE2319280A1/de

1973-12-19 Priority claimed from DE2363139A external-priority patent/DE2363139A1/de

1974-04-17 Application filed by Bayer AG filed Critical Bayer AG

1978-07-18 Application granted granted Critical

1978-07-18 Publication of CA1034953A publication Critical patent/CA1034953A/en

Status Expired legal-status Critical Current

Links

JEXVQSWXXUJEMA-UHFFFAOYSA-N pyrazol-3-one Chemical class O=C1C=CN=N1 JEXVQSWXXUJEMA-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
- C07D231/20—One oxygen atom attached in position 3 or 5
- C07D231/22—One oxygen atom attached in position 3 or 5 with aryl radicals attached to ring nitrogen atoms
- C07D231/24—One oxygen atom attached in position 3 or 5 with aryl radicals attached to ring nitrogen atoms having sulfone or sulfonic acid radicals in the molecule
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/10—Antioedematous agents; Diuretics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
- C07D231/20—One oxygen atom attached in position 3 or 5
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/44—Oxygen and nitrogen or sulfur and nitrogen atoms
- C07D231/52—Oxygen atom in position 3 and nitrogen atom in position 5, or vice versa

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Hematology (AREA)
Diabetes (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Catalysts (AREA)

CA197,660A 1973-04-17 1974-04-17 Pyrazol-5-ones Expired CA1034953A (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE2319280A DE2319280A1 (de)	1973-04-17	1973-04-17	1-substituierte pyrazolone-(5), verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel
DE2363139A DE2363139A1 (de)	1973-12-19	1973-12-19	1-substituierte pyrazolone-(5), verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel

Publications (1)

Publication Number	Publication Date
CA1034953A true CA1034953A (en)	1978-07-18

Family

ID=25764996

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CA197,660A Expired CA1034953A (en)	1973-04-17	1974-04-17	Pyrazol-5-ones

Country Status (27)

Country	Link
US (1)	US3957814A (ro)
JP (1)	JPS5314071B2 (ro)
AR (5)	AR207444A1 (ro)
AT (1)	AT337176B (ro)
BG (5)	BG21405A3 (ro)
CA (1)	CA1034953A (ro)
CH (5)	CH603592A5 (ro)
DD (1)	DD113757A5 (ro)
DK (1)	DK136066C (ro)
EG (1)	EG11157A (ro)
ES (3)	ES425373A1 (ro)
FI (1)	FI57587C (ro)
FR (1)	FR2226172B1 (ro)
GB (1)	GB1429141A (ro)
HK (1)	HK70276A (ro)
HU (1)	HU168590B (ro)
IE (1)	IE39212B1 (ro)
IL (1)	IL44626A (ro)
LU (1)	LU69872A1 (ro)
NL (1)	NL177917C (ro)
NO (1)	NO138530C (ro)
PH (1)	PH14829A (ro)
PL (1)	PL96883B1 (ro)
RO (2)	RO69740A (ro)
SE (1)	SE408301B (ro)
SU (2)	SU541430A3 (ro)
YU (1)	YU104874A (ro)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4056533A (en) *	1973-04-17	1977-11-01	Bayer Aktiengesellschaft	Pyrazol-5-ones
DE2526467A1 (de) *	1975-06-13	1976-12-30	Bayer Ag	4-substituierte pyrazolderivate, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel
DE3306366A1 (de) *	1983-02-24	1984-08-30	Bayer Ag, 5090 Leverkusen	Muzolimin enthaltende arzneimittel, deren verwendung und verfahren zu deren herstellung
US4663327A (en) *	1984-05-23	1987-05-05	Bayer Aktiengesellschaft	1-heteroaryl-4-aryl-pyrazolin-5-ones
JPH0730031B2 (ja) *	1986-04-02	1995-04-05	日産化学工業株式会社	２―ピラゾリン―５―オン類の製造法
DE3738963A1 (de) *	1987-11-17	1989-05-24	Bayer Ag	3-aminopyrazolin-5-one
US5711929A (en) *	1989-05-06	1998-01-27	698638 Alberta Ltd.	Purification of elemental sulphur
GB8912861D0 (en) *	1989-06-05	1989-07-26	Sherritt Gordon Ltd	Purification of elemental sulphur
US5300514A (en) *	1990-07-17	1994-04-05	Eli Lilly And Company	Pyrazolidinone CCK and gastrin antagonists and pharmaceutical formulations thereof
US5399565A (en) *	1990-07-17	1995-03-21	Eli Lilly And Company	Pyrazolidinone CCK and gastrin antagonists and pharmaceutical formulations therof
DE69131268T2 (de) *	1990-09-21	1999-12-30	Rohm And Haas Co., Philadelphia	Dihydropyridazinone und Pyridazinone als Fungizide
CN1038249C (zh) *	1991-08-28	1998-05-06	罗姆和哈斯公司	含有二氢哒嗪酮及其相关化合物的杀菌组合物

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US2376380A (en) *		1945-05-22		Preparation of amino pyrazolones
GB636988A (en) *	1947-12-24	1950-05-10	Gevaert Photo Producten Naamlo	Improvements in and relating to the production of colour photographic images
US2511231A (en) *	1949-03-26	1950-06-13	Eastman Kodak Co	1-cyanophenyl-3-acylamino-5-pyrazolone couplers for color photography
US2600788A (en) *	1949-06-07	1952-06-17	Eastman Kodak Co	Halogen-substituted pyrazolone couplers for color photography
US2672417A (en) *	1949-12-31	1954-03-16	Gevaert Photo Prod Nv	Production of color photographic images
NL279140A (ro) *	1961-05-31

1974
- 1974-01-01 AR AR253331A patent/AR207444A1/es active
- 1974-03-29 FR FR7411495A patent/FR2226172B1/fr not_active Expired
- 1974-04-09 HU HUBA3058A patent/HU168590B/hu unknown
- 1974-04-11 FI FI1105/74A patent/FI57587C/fi active
- 1974-04-12 BG BG027980A patent/BG21405A3/xx unknown
- 1974-04-12 BG BG026395A patent/BG21217A3/xx unknown
- 1974-04-12 BG BG027979A patent/BG22821A3/xx unknown
- 1974-04-12 BG BG027977A patent/BG21857A3/xx unknown
- 1974-04-12 IL IL44626A patent/IL44626A/xx unknown
- 1974-04-12 BG BG027978A patent/BG21218A3/xx unknown
- 1974-04-15 YU YU01048/74A patent/YU104874A/xx unknown
- 1974-04-15 RO RO7485201A patent/RO69740A/ro unknown
- 1974-04-15 US US05/461,282 patent/US3957814A/en not_active Expired - Lifetime
- 1974-04-15 JP JP4111274A patent/JPS5314071B2/ja not_active Expired
- 1974-04-15 RO RO7400078420A patent/RO63749A/ro unknown
- 1974-04-15 PH PH15730A patent/PH14829A/en unknown
- 1974-04-15 DD DD177913A patent/DD113757A5/xx unknown
- 1974-04-16 NO NO741365A patent/NO138530C/no unknown
- 1974-04-16 ES ES425373A patent/ES425373A1/es not_active Expired
- 1974-04-16 PL PL1974170378A patent/PL96883B1/pl unknown
- 1974-04-16 NL NLAANVRAGE7405115,A patent/NL177917C/xx not_active IP Right Cessation
- 1974-04-16 CH CH524274A patent/CH603592A5/xx not_active IP Right Cessation
- 1974-04-16 DK DK208074A patent/DK136066C/da not_active IP Right Cessation
- 1974-04-16 LU LU69872A patent/LU69872A1/xx unknown
- 1974-04-16 CH CH156477A patent/CH605801A5/xx not_active IP Right Cessation
- 1974-04-16 EG EG119/74A patent/EG11157A/xx active
- 1974-04-16 SE SE7405078A patent/SE408301B/sv not_active IP Right Cessation
- 1974-04-16 CH CH156577A patent/CH605800A5/xx not_active IP Right Cessation
- 1974-04-16 CH CH156377A patent/CH596172A5/xx not_active IP Right Cessation
- 1974-04-16 AT AT313274A patent/AT337176B/de not_active IP Right Cessation
- 1974-04-16 CH CH156677A patent/CH605797A5/xx not_active IP Right Cessation
- 1974-04-16 GB GB1650774A patent/GB1429141A/en not_active Expired
- 1974-04-17 CA CA197,660A patent/CA1034953A/en not_active Expired
- 1974-04-17 IE IE798/74A patent/IE39212B1/xx unknown
1975
- 1975-01-01 AR AR258508A patent/AR205272A1/es active
- 1975-01-01 AR AR258506A patent/AR208192A1/es active
- 1975-01-01 AR AR258507A patent/AR205271A1/es active
- 1975-03-19 SU SU2114308A patent/SU541430A3/ru active
- 1975-03-19 SU SU2115103A patent/SU539525A3/ru active
- 1975-04-25 AR AR258505A patent/AR204951A1/es active
1976
- 1976-04-15 ES ES447064A patent/ES447064A1/es not_active Expired
- 1976-04-15 ES ES447063A patent/ES447063A1/es not_active Expired
- 1976-11-11 HK HK702/76*UA patent/HK70276A/xx unknown

Also Published As

Publication number	Publication date
DD113757A5 (ro)	1975-06-20
AR204951A1 (es)	1976-03-19
NO741365L (no)	1974-10-18
RO63749A (fr)	1979-01-15
CH605801A5 (ro)	1978-10-13
DK136066B (da)	1977-08-08
AR207444A1 (es)	1976-10-08
IL44626A (en)	1980-01-31
SE408301B (sv)	1979-06-05
RO69740A (ro)	1982-09-09
NL177917C (nl)	1985-12-16
CH605797A5 (ro)	1978-10-13
AT337176B (de)	1977-06-10
PH14829A (en)	1981-12-16
ATA313274A (de)	1976-10-15
JPS5018466A (ro)	1975-02-26
AR205272A1 (es)	1976-04-21
DK136066C (da)	1978-01-16
FI57587B (fi)	1980-05-30
IL44626A0 (en)	1974-06-30
ES425373A1 (es)	1976-09-01
PL96883B1 (pl)	1978-01-31
JPS5314071B2 (ro)	1978-05-15
BG21405A3 (bg)	1976-05-20
CH596172A5 (ro)	1978-02-28
SU541430A3 (ru)	1976-12-30
CH605800A5 (ro)	1978-10-13
NO138530C (no)	1978-09-20
US3957814A (en)	1976-05-18
FI57587C (fi)	1980-09-10
BG21857A3 (bg)	1976-09-20
NO138530B (no)	1978-05-12
ES447063A1 (es)	1977-06-16
LU69872A1 (ro)	1974-11-28
GB1429141A (en)	1976-03-24
AU6817474A (en)	1975-10-23
BG21218A3 (bg)	1976-03-20
ES447064A1 (es)	1977-09-16
IE39212B1 (en)	1978-08-30
BG21217A3 (bg)	1976-03-20
BG22821A3 (bg)	1977-04-20
HK70276A (en)	1976-11-19
CH603592A5 (ro)	1978-08-31
FR2226172A1 (ro)	1974-11-15
EG11157A (en)	1978-03-29
AR208192A1 (es)	1976-12-09
SU539525A3 (ru)	1976-12-15
YU104874A (en)	1982-02-28
HU168590B (ro)	1976-06-28
IE39212L (en)	1974-10-17
AR205271A1 (es)	1976-04-21
NL7405115A (ro)	1974-10-21
NL177917B (nl)	1985-07-16
FR2226172B1 (ro)	1978-07-28

Publication	Publication Date	Title
AU474137B2 (en)	1976-07-15	Auto-refractometer
AU468964B2 (en)	1976-01-29	Melik
CA1000682A (en)	1976-11-30	Sillcock
AU498889B2 (en)	1979-03-29	Piperidylene benzocycloheptathiophenes
CA1033713A (en)	1978-06-27	D-homo-steroids
CA1034592A (en)	1978-07-11	Amidinoureas
CA1031258A (en)	1978-05-16	Para-influenza-3-virus
AU476397B2 (en)	1976-09-16	A-cycloalkylbenzyl lactamimides
AU476505B2 (en)	1976-09-23	Alkylbenxyl lactamimides
AU472907B2 (en)	1976-06-10	Firecheck
CA971440A (en)	1975-07-22	Headgate
CA998215A (en)	1976-10-12	Warmhouse
AU476386B2 (en)	1976-09-16	Dibenzocycloheptenyl lactamimides
CA1007225A (en)	1977-03-22	Polycycloanilines
CA1031349A (en)	1978-05-16	Thiadiazolylimidazolidinones
AU471241B2 (en)	1976-04-15	Benzothiazolylureas
AU484993B2 (en)	1975-07-17	Polyhydroxyphenylchromanones
AU482530B2 (en)	1974-07-25	Benzocycloheptathiophenes
AU489559B2 (en)	1976-01-15	Amidinoureas
AU479426B2 (en)	1975-08-21	Carbothiolates
AU481998B2 (en)	1975-11-06	Benzenedisulfonamides
AU492165B2 (en)	1976-01-15	2-hydroxyphenyl-1-oxa-4 azaspiro-alkan-derivatives
AU482276B2 (en)	1976-04-08	Spiro-cyclopropanes
AU489560B2 (en)	1976-01-15	Amidinoureas
AU492033B2 (en)	1976-06-03	D-homo-20-keto-pregnanes