CA1083143A - Derives carba de la somatostatine et procede de preparation - Google Patents

Derives carba de la somatostatine et procede de preparation

Info

Publication number
CA1083143A
CA1083143A CA267,944A CA267944A CA1083143A CA 1083143 A CA1083143 A CA 1083143A CA 267944 A CA267944 A CA 267944A CA 1083143 A CA1083143 A CA 1083143A
Authority
CA
Canada
Prior art keywords
phe
thr
lys
trp
boc
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA267,944A
Other languages
English (en)
Inventor
Nedumparambil A. Abraham
Kazimir Sestanj
Hans U. Immer
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Wyeth Canada Inc
Original Assignee
Ayerst Mckenna and Harrison Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ayerst Mckenna and Harrison Inc filed Critical Ayerst Mckenna and Harrison Inc
Application granted granted Critical
Publication of CA1083143A publication Critical patent/CA1083143A/fr
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/655—Somatostatins
    • C07K14/6555—Somatostatins at least 1 amino acid in D-form
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biophysics (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Zoology (AREA)
  • Biochemistry (AREA)
  • Toxicology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Endocrinology (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
CA267,944A 1976-01-02 1976-12-15 Derives carba de la somatostatine et procede de preparation Expired CA1083143A (fr)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US64609676A 1976-01-02 1976-01-02
US646,096 1976-01-02
US74549376A 1976-11-26 1976-11-26
US745,493 1976-11-26

Publications (1)

Publication Number Publication Date
CA1083143A true CA1083143A (fr) 1980-08-05

Family

ID=27094853

Family Applications (1)

Application Number Title Priority Date Filing Date
CA267,944A Expired CA1083143A (fr) 1976-01-02 1976-12-15 Derives carba de la somatostatine et procede de preparation

Country Status (6)

Country Link
CA (1) CA1083143A (fr)
DE (1) DE2659758A1 (fr)
FR (2) FR2336943A1 (fr)
GB (1) GB1570210A (fr)
IL (1) IL51134A (fr)
SE (1) SE7614757L (fr)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2860734D1 (en) * 1977-06-08 1981-09-03 Merck & Co Inc Somatostatin analogs, process for their preparation and pharmaceutical compositions containing them
US4115554A (en) * 1977-08-29 1978-09-19 Merck & Co., Inc. Somatostatin analogs
US4140767A (en) * 1977-12-01 1979-02-20 Merck & Co., Inc. Somatostatin analogs
US4139526A (en) * 1977-12-01 1979-02-13 Merck & Co., Inc. Somatostatin analogs
US4369179A (en) * 1979-12-14 1983-01-18 Ciba-Geigy Corporation Acylpeptides
US5443815A (en) * 1991-11-27 1995-08-22 Diatech, Inc. Technetium-99m labeled peptides for imaging
US6183722B1 (en) 1991-11-27 2001-02-06 Diatide, Inc. Somatostatin analogs
US5620675A (en) 1992-06-23 1997-04-15 Diatech, Inc. Radioactive peptides
US5716596A (en) * 1992-06-23 1998-02-10 Diatide, Inc. Radioactively labeled somatostatin-derived peptides for imaging and therapeutic uses
US6017512A (en) * 1992-06-23 2000-01-25 Diatide, Inc. Radiolabeled peptides
US5871711A (en) * 1992-06-23 1999-02-16 Diatide, Inc. Radioactively-labeled somatostatin-derived peptides for imaging and therapeutic uses
DE69426673T2 (de) * 1993-06-23 2001-09-20 Diatide, Inc. Radiomarkierte somatostatin derivate zur abbildung und zur therapeutischen verwendung
US6051206A (en) * 1994-06-03 2000-04-18 Diatide, Inc Radiolabeled somatostatin-derived peptides for imaging and therapeutic uses

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2416048A1 (de) * 1974-04-03 1975-10-30 Hoechst Ag Neue peptide mit biologischer wirkung
US4011182A (en) * 1975-03-21 1977-03-08 American Home Products Corporation Cyclic undecapeptide analogs of somatostatin and intermediates
US4000259A (en) * 1975-06-16 1976-12-28 American Home Products Corporation Cyclic dodecapeptide analogs of somatostatin and intermediates

Also Published As

Publication number Publication date
FR2336943A1 (fr) 1977-07-29
FR2336943B1 (fr) 1980-04-18
DE2659758A1 (de) 1977-07-07
SE7614757L (sv) 1977-09-16
GB1570210A (en) 1980-06-25
IL51134A (en) 1980-02-29
FR2384745A1 (fr) 1978-10-20
IL51134A0 (en) 1977-02-28

Similar Documents

Publication Publication Date Title
CA1245217A (fr) Peptides inhibiteurs de la renine
CA1111841A (fr) Cyclopeptides
US4261886A (en) Peptides having thymopoietin-like activity
US4803261A (en) Method for synthesizing a peptide containing a non-peptide
CA1065856A (fr) Derives de la calcitonine du saumon
US4190646A (en) Polypeptide compositions and methods
AU598507B2 (en) Peptides with vasorelaxant, natriuretic and diuretic effects, a process for their preparation, agents containing them, and their use
US4002740A (en) Tridecapeptide compositions and methods
US4486415A (en) Cyclic hexapeptide somatostatin analogs
CA1107273A (fr) Analogues de la somatostatine ayant un residu tryptophyl substitue en position 8
GB1570210A (en) Peptides
US4703034A (en) Novel cyclic tetrapeptide
CA1255850A (fr) Peptides avec ponts disulfures et methode de preparation
US4115554A (en) Somatostatin analogs
US4612366A (en) Cyclic hexapeptide somatostatin analogs
EP0016612B1 (fr) Peptides à activité analogue à l'ubiquitine, procédé pour leur préparation, compositions thérapeutiques les contenant et leur utilisation
US4162248A (en) Somatostatin analogs
US4611054A (en) Cyclic hexapeptide somatostatin analogs
US4190647A (en) Polypeptides and methods
US3917581A (en) Derivatives of somatostatin and process therefor
US4133805A (en) Cyclic undecapeptides related to somatostatin and intermediates therefor
US4397842A (en) Peptides having thymopoietin-like activity
EP0018182B1 (fr) Peptides possédant une activité analogue à celle de la thymopoiétine, compositions pharmaceutiques qui les contiennent, et procédé pour les préparer
US4118380A (en) Decapeptide analogs of somatostatin
EP0113029B1 (fr) Hexapeptides dicycliques, leur procédé de préparation et leurs compositions pharmaceutiques

Legal Events

Date Code Title Description
MKEX Expiry