CA2149147A1 - Derives de pyrimidineamine pharmacologiquement actifs ainsi que leurs procedes de preparation - Google Patents

Derives de pyrimidineamine pharmacologiquement actifs ainsi que leurs procedes de preparation

Info

Publication number: CA2149147A1
Authority: CA; Canada
Prior art keywords: substituted; lower alkyl; processes; preparation; pharmacologically active
Prior art date: 1993-10-01
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Granted

Application number

CA002149147A

Other languages

English (en)

Other versions

CA2149147C (fr

Inventor

Jurg Zimmermann

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Novartis AG

Original Assignee

Individual

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1993-10-01

Filing date

1994-09-21

Publication date

1995-04-13

1994-09-21 Application filed by Individual filed Critical Individual

1994-09-21 Priority claimed from PCT/EP1994/003148 external-priority patent/WO1995009851A1/fr

1995-04-13 Publication of CA2149147A1 publication Critical patent/CA2149147A1/fr

2006-05-02 Application granted granted Critical

2006-05-02 Publication of CA2149147C publication Critical patent/CA2149147C/fr

2014-09-21 Anticipated expiration legal-status Critical

Status Expired - Fee Related legal-status Critical Current

Links

LJXQPZWIHJMPQQ-UHFFFAOYSA-N pyrimidin-2-amine Chemical class NC1=NC=CC=N1 LJXQPZWIHJMPQQ-UHFFFAOYSA-N 0.000 title 1
125000000217 alkyl group Chemical group 0.000 abstract 4
UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 2
125000003282 alkyl amino group Chemical group 0.000 abstract 2
-1 cyano, carbamoyl Chemical group 0.000 abstract 2
229910052736 halogen Inorganic materials 0.000 abstract 2
150000002367 halogens Chemical class 0.000 abstract 2
229910052739 hydrogen Inorganic materials 0.000 abstract 2
239000001257 hydrogen Substances 0.000 abstract 2
206010028980 Neoplasm Diseases 0.000 abstract 1
229910052799 carbon Inorganic materials 0.000 abstract 1
125000004432 carbon atom Chemical group C* 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
125000002883 imidazolyl group Chemical group 0.000 abstract 1
XGXNTJHZPBRBHJ-UHFFFAOYSA-N n-phenylpyrimidin-2-amine Chemical class N=1C=CC=NC=1NC1=CC=CC=C1 XGXNTJHZPBRBHJ-UHFFFAOYSA-N 0.000 abstract 1
125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
125000003373 pyrazinyl group Chemical group 0.000 abstract 1
125000002098 pyridazinyl group Chemical group 0.000 abstract 1
125000004076 pyridyl group Chemical group 0.000 abstract 1
125000000714 pyrimidinyl group Chemical group 0.000 abstract 1
125000001424 substituent group Chemical group 0.000 abstract 1
125000000335 thiazolyl group Chemical group 0.000 abstract 1

Landscapes

Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

CA002149147A 1993-10-01 1994-09-21 Derives de pyrimidineamine pharmacologiquement actifs ainsi que leurs procedes de preparation Expired - Fee Related CA2149147C (fr)

Applications Claiming Priority (5)

Application Number	Priority Date	Filing Date	Title
CH2968/93-9		1993-10-01
CH296893		1993-10-01
CH228094		1994-07-18
CH2280/94-0		1994-07-18
PCT/EP1994/003148 WO1995009851A1 (fr)	1993-10-01	1994-09-21	Derives de pyrimidineamine pharmacologiquement actifs ainsi que leurs procedes de preparation

Publications (2)

Publication Number	Publication Date
CA2149147A1 true CA2149147A1 (fr)	1995-04-13
CA2149147C CA2149147C (fr)	2006-05-02

Family

ID=36283829

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CA002149147A Expired - Fee Related CA2149147C (fr)	1993-10-01	1994-09-21	Derives de pyrimidineamine pharmacologiquement actifs ainsi que leurs procedes de preparation

Country Status (1)

Country	Link
CA (1)	CA2149147C (fr)

1994
- 1994-09-21 CA CA002149147A patent/CA2149147C/fr not_active Expired - Fee Related

Also Published As

Publication number	Publication date
CA2149147C (fr)	2006-05-02

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Legal Events

Date	Code	Title	Description
2001-08-17	EEER	Examination request
2010-09-21	MKLA	Lapsed