CA2572990A1 - Use of substituted 2-thio-3,5-dicyano-4-phenyl-6-aminopyridines in the treatment of nausea and vomiting - Google Patents

Use of substituted 2-thio-3,5-dicyano-4-phenyl-6-aminopyridines in the treatment of nausea and vomiting Download PDF

Info

Publication number: CA2572990A1
Authority: CA; Canada
Prior art keywords: salts; vomiting; hydrates; nausea; treatment
Prior art date: 2004-07-06
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Abandoned

Application number

CA002572990A

Other languages

English (en)

French (fr)

Inventor

Thomas Krahn

Wolfgang Thielemann

Ulrich Rosentreter

Nicole Diedrichs

Thomas Kraemer

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Bayer Pharma AG

Original Assignee

Individual

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2004-07-06

Filing date

2005-06-23

Publication date

2006-01-12

2005-06-23 Application filed by Individual filed Critical Individual

2006-01-12 Publication of CA2572990A1 publication Critical patent/CA2572990A1/en

Status Abandoned legal-status Critical Current

Links

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238000011282 treatment Methods 0.000 title claims abstract description 17
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150000003839 salts Chemical class 0.000 claims description 21
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Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
General Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
Bioinformatics & Cheminformatics (AREA)
Hospice & Palliative Care (AREA)
Otolaryngology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Pyridine Compounds (AREA)
Hydrogenated Pyridines (AREA)
Plural Heterocyclic Compounds (AREA)

CA002572990A 2004-07-06 2005-06-23 Use of substituted 2-thio-3,5-dicyano-4-phenyl-6-aminopyridines in the treatment of nausea and vomiting Abandoned CA2572990A1 (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
DE102004032651.7		2004-07-06
DE102004032651A DE102004032651A1 (de)	2004-07-06	2004-07-06	Verwendung von substituierten 2-Thio-3,5-dicyano-4-phenyl-6-aminopyriden bei der Behandlung von Übelkeit und Erbrechen
PCT/EP2005/006779 WO2006002823A1 (de)	2004-07-06	2005-06-23	Verwendung von substituierten 2-thio-3,5-dicyano-4-phenyl-6-aminopyridinen bei der behandlung von übelkeit und erbrechen

Publications (1)

Publication Number	Publication Date
CA2572990A1 true CA2572990A1 (en)	2006-01-12

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ID=34970906

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CA002572990A Abandoned CA2572990A1 (en)	2004-07-06	2005-06-23	Use of substituted 2-thio-3,5-dicyano-4-phenyl-6-aminopyridines in the treatment of nausea and vomiting

Country Status (18)

Country	Link
US (1)	US7709504B2 (de)
EP (1)	EP1765343B1 (de)
JP (1)	JP2008505139A (de)
KR (1)	KR20070041561A (de)
CN (1)	CN101014342A (de)
AT (1)	ATE446753T1 (de)
AU (1)	AU2005259506A1 (de)
BR (1)	BRPI0513149A (de)
CA (1)	CA2572990A1 (de)
DE (2)	DE102004032651A1 (de)
EC (1)	ECSP077130A (de)
ES (1)	ES2333805T3 (de)
IL (1)	IL180551A0 (de)
MA (1)	MA28707B1 (de)
MX (1)	MX2007000224A (de)
NO (1)	NO20070608L (de)
RU (1)	RU2007104234A (de)
WO (1)	WO2006002823A1 (de)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE10110747A1 (de) *	2001-03-07	2002-09-12	Bayer Ag	Substituierte 2,6-Diamino-3,5-dicyano-4-aryl-pyridine und ihre Verwendung
DE102004042607A1 (de) *	2004-09-03	2006-03-09	Bayer Healthcare Ag	Substituierte Phenylaminothiazole und ihre Verwendung
DE102006042143A1 (de) *	2006-09-08	2008-03-27	Bayer Healthcare Aktiengesellschaft	Neue substituierte Bipyridin-Derivate und ihre Verwendung
DE102006056740A1 (de) *	2006-12-01	2008-06-05	Bayer Healthcare Ag	Cyclisch substituierte 3,5-Dicyano-2-thiopyridine und ihre Verwendung
DE102006056739A1 (de) *	2006-12-01	2008-06-05	Bayer Healthcare Ag	Substituierte 4-Amino-3,5-dicyano-2-thiopyridine und ihre Verwendung
DE102007035367A1 (de)	2007-07-27	2009-01-29	Bayer Healthcare Ag	Substituierte Aryloxazole und ihre Verwendung
DE102007036076A1 (de)	2007-08-01	2009-02-05	Bayer Healthcare Aktiengesellschaft	Dipeptoid-Produgs und ihre Verwendung
DE102007061764A1 (de) *	2007-12-20	2009-06-25	Bayer Healthcare Ag	Anellierte Cyanopyridine und ihre Verwendung
DE102007061763A1 (de) *	2007-12-20	2009-06-25	Bayer Healthcare Ag	Substituierte azabicyclische Verbindungen und ihre Verwendung
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- 2005-06-23 AU AU2005259506A patent/AU2005259506A1/en not_active Abandoned
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- 2005-06-23 KR KR1020077002837A patent/KR20070041561A/ko not_active Withdrawn
- 2005-06-23 DE DE502005008416T patent/DE502005008416D1/de not_active Expired - Lifetime
- 2005-06-23 EP EP05753010A patent/EP1765343B1/de not_active Expired - Lifetime
- 2005-06-23 CN CNA2005800299192A patent/CN101014342A/zh active Pending
- 2005-06-23 JP JP2007519663A patent/JP2008505139A/ja active Pending
- 2005-06-23 ES ES05753010T patent/ES2333805T3/es not_active Expired - Lifetime
- 2005-06-23 WO PCT/EP2005/006779 patent/WO2006002823A1/de not_active Ceased
- 2005-06-23 CA CA002572990A patent/CA2572990A1/en not_active Abandoned
- 2005-06-23 BR BRPI0513149-9A patent/BRPI0513149A/pt not_active Application Discontinuation
- 2005-06-23 RU RU2007104234/15A patent/RU2007104234A/ru unknown
2006
- 2006-12-29 MA MA29597A patent/MA28707B1/fr unknown
2007
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Publication number	Publication date
US20080249133A1 (en)	2008-10-09
RU2007104234A (ru)	2008-08-20
BRPI0513149A (pt)	2008-04-29
JP2008505139A (ja)	2008-02-21
IL180551A0 (en)	2008-03-20
DE502005008416D1 (de)	2009-12-10
MX2007000224A (es)	2007-06-15
EP1765343A1 (de)	2007-03-28
ECSP077130A (es)	2007-02-28
WO2006002823A1 (de)	2006-01-12
ES2333805T3 (es)	2010-03-01
AU2005259506A1 (en)	2006-01-12
MA28707B1 (fr)	2007-06-01
DE102004032651A1 (de)	2006-02-16
NO20070608L (no)	2007-02-01
KR20070041561A (ko)	2007-04-18
EP1765343B1 (de)	2009-10-28
US7709504B2 (en)	2010-05-04
ATE446753T1 (de)	2009-11-15
CN101014342A (zh)	2007-08-08

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2012-06-26	FZDE	Discontinued

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