CA2658200A1 - Inhibiteurs de naaladase utiles comme composes et compositions pharmaceutiques - Google Patents

Inhibiteurs de naaladase utiles comme composes et compositions pharmaceutiques Download PDF

Info

Publication number: CA2658200A1
Authority: CA; Canada
Prior art keywords: formula; pentanedioic acid; moiety; compound; acid
Prior art date: 1998-07-06
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Abandoned

Application number

CA002658200A

Other languages

English (en)

Inventor

Paul F. Jackson

Keith M. Maclin

Eric Wang

Barbara S. Slusher

Rena S. Lapidus

Pavel Majer

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Eisai Inc

Original Assignee

Individual

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-07-06

Filing date

1999-07-02

Publication date

2000-01-13

1998-07-06 Priority claimed from US09/110,262 external-priority patent/US6395718B1/en

1999-01-12 Priority claimed from US09/228,391 external-priority patent/US6265609B1/en

1999-07-02 Application filed by Individual filed Critical Individual

1999-07-02 Priority claimed from CA002337797A external-priority patent/CA2337797C/fr

2000-01-13 Publication of CA2658200A1 publication Critical patent/CA2658200A1/fr

Status Abandoned legal-status Critical Current

Links

239000003112 inhibitor Substances 0.000 title claims abstract description 93
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Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Compounds Containing Sulfur Atoms (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

CA002658200A 1998-07-06 1999-07-02 Inhibiteurs de naaladase utiles comme composes et compositions pharmaceutiques Abandoned CA2658200A1 (fr)

Applications Claiming Priority (7)

Application Number	Priority Date	Filing Date	Title
US11018698A	1998-07-06	1998-07-06
US09/110,262 US6395718B1 (en)	1998-07-06	1998-07-06	Pharmaceutical compositions and methods of inhibiting angiogenesis using naaladase inhibitors
US09/228,391		1999-01-12
US09/110,262		1999-01-12
US09/110,186		1999-01-12
US09/228,391 US6265609B1 (en)	1998-07-06	1999-01-12	Thio-substituted pentanedioic acid derivatives
CA002337797A CA2337797C (fr)	1998-07-06	1999-07-02	Inhibiteurs de naaladase utiles comme composes et compositions pharmaceutiques

Related Parent Applications (1)

Application Number	Title	Priority Date	Filing Date
CA002337797A Division CA2337797C (fr)	1998-07-06	1999-07-02	Inhibiteurs de naaladase utiles comme composes et compositions pharmaceutiques

Publications (1)

Publication Number	Publication Date
CA2658200A1 true CA2658200A1 (fr)	2000-01-13

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ID=40639568

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CA002658200A Abandoned CA2658200A1 (fr)	1998-07-06	1999-07-02	Inhibiteurs de naaladase utiles comme composes et compositions pharmaceutiques

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JP (1)	JP2010001312A (fr)
CA (1)	CA2658200A1 (fr)
IL (1)	IL140499A (fr)

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Publication number	Priority date	Publication date	Assignee	Title
JPS5142175B2 (fr) *	1973-07-04	1976-11-13
JPS57116045A (en) *	1981-01-13	1982-07-19	Tokyo Organ Chem Ind Ltd	Dithiocarbamate, its preparation and injurious organism exterminatory agent consisting of said dithiocarbamate
JPS5810565A (ja) *	1981-07-09	1983-01-21	Tanabe Seiyaku Co Ltd	トリプトフアン誘導体及びその製法
JPS5810558A (ja) *	1981-07-09	1983-01-21	Tanabe Seiyaku Co Ltd	新規アミノ酸誘導体及びその製法
JPS6153285A (ja) *	1984-08-24	1986-03-17	Kyowa Hakko Kogyo Co Ltd	β−ラクタム化合物
JPH01206338A (ja) *	1988-02-15	1989-08-18	Konica Corp	ハロゲン化銀カラー写真感光材料
US5807884A (en) *	1992-10-30	1998-09-15	Emory University	Treatment for atherosclerosis and other cardiovascular and inflammatory diseases
CN1057907C (zh) *	1995-06-13	2000-11-01	北京医科大学	驱镉药物及其合成方法和应用
ID18382A (id) *	1996-09-27	1998-04-02	Guilford Pharm Inc	Komposisi sediaan farmasi dan metoda pengobatan gangguan kompulsif dengan menggunakan inhibitor naaladase

1999
- 1999-07-02 CA CA002658200A patent/CA2658200A1/fr not_active Abandoned
2000
- 2000-12-22 IL IL140499A patent/IL140499A/en not_active IP Right Cessation
2009
- 2009-09-30 JP JP2009228198A patent/JP2010001312A/ja active Pending

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IL140499A (en)	2006-12-31

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2009-03-17	EEER	Examination request
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Publication	Publication Date	Title
RU2268881C2 (ru)	2006-01-27	Производные пентадикарбоновой кислоты, фармацевтическая композиция на их основе и способы лечения
US6458775B1 (en)	2002-10-01	NAALADase inhibitors useful as pharmaceutical compounds and compositions
US6384022B1 (en)	2002-05-07	Prodrugs of NAALAdase inhibitors
AU733880B2 (en)	2001-05-31	Naaladase compositions and methods for treating glutamate abnormality and effecting neuronal activity in animals
US6265609B1 (en)	2001-07-24	Thio-substituted pentanedioic acid derivatives
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