CA2761000C - Composition pour administration prolongee de medicaments comprenant un liant geopolymere - Google Patents
Composition pour administration prolongee de medicaments comprenant un liant geopolymere Download PDFInfo
- Publication number
- CA2761000C CA2761000C CA2761000A CA2761000A CA2761000C CA 2761000 C CA2761000 C CA 2761000C CA 2761000 A CA2761000 A CA 2761000A CA 2761000 A CA2761000 A CA 2761000A CA 2761000 C CA2761000 C CA 2761000C
- Authority
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- Prior art keywords
- composition
- api
- ddss
- active pharmaceutical
- pharmaceutical ingredient
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
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- 239000011163 secondary particle Substances 0.000 description 1
- 230000001624 sedative effect Effects 0.000 description 1
- 210000002966 serum Anatomy 0.000 description 1
- 229910021487 silica fume Inorganic materials 0.000 description 1
- 235000012239 silicon dioxide Nutrition 0.000 description 1
- 229910052814 silicon oxide Inorganic materials 0.000 description 1
- 208000019116 sleep disease Diseases 0.000 description 1
- 210000000813 small intestine Anatomy 0.000 description 1
- 239000000779 smoke Substances 0.000 description 1
- 230000000391 smoking effect Effects 0.000 description 1
- 238000002791 soaking Methods 0.000 description 1
- 229910001388 sodium aluminate Inorganic materials 0.000 description 1
- 239000011780 sodium chloride Substances 0.000 description 1
- 238000003980 solgel method Methods 0.000 description 1
- 239000012453 solvate Substances 0.000 description 1
- 239000000600 sorbitol Substances 0.000 description 1
- 210000000278 spinal cord Anatomy 0.000 description 1
- 239000008107 starch Substances 0.000 description 1
- 235000019698 starch Nutrition 0.000 description 1
- 229930002534 steroid glycoside Natural products 0.000 description 1
- 150000008143 steroidal glycosides Chemical class 0.000 description 1
- 150000003431 steroids Chemical class 0.000 description 1
- 238000003860 storage Methods 0.000 description 1
- 235000011149 sulphuric acid Nutrition 0.000 description 1
- 239000013589 supplement Substances 0.000 description 1
- 230000009747 swallowing Effects 0.000 description 1
- 230000001975 sympathomimetic effect Effects 0.000 description 1
- 229940064707 sympathomimetics Drugs 0.000 description 1
- 238000002636 symptomatic treatment Methods 0.000 description 1
- 230000001839 systemic circulation Effects 0.000 description 1
- 229960003188 temazepam Drugs 0.000 description 1
- IMCGHZIGRANKHV-AJNGGQMLSA-N tert-butyl (3s,5s)-2-oxo-5-[(2s,4s)-5-oxo-4-propan-2-yloxolan-2-yl]-3-propan-2-ylpyrrolidine-1-carboxylate Chemical compound O1C(=O)[C@H](C(C)C)C[C@H]1[C@H]1N(C(=O)OC(C)(C)C)C(=O)[C@H](C(C)C)C1 IMCGHZIGRANKHV-AJNGGQMLSA-N 0.000 description 1
- IQWYAQCHYZHJOS-UHFFFAOYSA-N tetrazepam Chemical compound N=1CC(=O)N(C)C2=CC=C(Cl)C=C2C=1C1=CCCCC1 IQWYAQCHYZHJOS-UHFFFAOYSA-N 0.000 description 1
- 229960005214 tetrazepam Drugs 0.000 description 1
- 229930003945 thebaine Natural products 0.000 description 1
- FQXXSQDCDRQNQE-VMDGZTHMSA-N thebaine Chemical compound C([C@@H](N(CC1)C)C2=CC=C3OC)C4=CC=C(OC)C5=C4[C@@]21[C@H]3O5 FQXXSQDCDRQNQE-VMDGZTHMSA-N 0.000 description 1
- 229940124597 therapeutic agent Drugs 0.000 description 1
- 229940126585 therapeutic drug Drugs 0.000 description 1
- 230000004797 therapeutic response Effects 0.000 description 1
- 229960001402 tilidine Drugs 0.000 description 1
- 210000001519 tissue Anatomy 0.000 description 1
- 230000009772 tissue formation Effects 0.000 description 1
- OGIDPMRJRNCKJF-UHFFFAOYSA-N titanium oxide Inorganic materials [Ti]=O OGIDPMRJRNCKJF-UHFFFAOYSA-N 0.000 description 1
- 230000000699 topical effect Effects 0.000 description 1
- 239000011573 trace mineral Substances 0.000 description 1
- 235000013619 trace mineral Nutrition 0.000 description 1
- 229960004380 tramadol Drugs 0.000 description 1
- TVYLLZQTGLZFBW-GOEBONIOSA-N tramadol Natural products COC1=CC=CC([C@@]2(O)[C@@H](CCCC2)CN(C)C)=C1 TVYLLZQTGLZFBW-GOEBONIOSA-N 0.000 description 1
- 239000003204 tranquilizing agent Substances 0.000 description 1
- 230000002936 tranquilizing effect Effects 0.000 description 1
- QORWJWZARLRLPR-UHFFFAOYSA-H tricalcium bis(phosphate) Chemical class [Ca+2].[Ca+2].[Ca+2].[O-]P([O-])([O-])=O.[O-]P([O-])([O-])=O QORWJWZARLRLPR-UHFFFAOYSA-H 0.000 description 1
- 230000003424 uricosuric effect Effects 0.000 description 1
- 229960005486 vaccine Drugs 0.000 description 1
- 229940124549 vasodilator Drugs 0.000 description 1
- 239000003071 vasodilator agent Substances 0.000 description 1
- 229940088594 vitamin Drugs 0.000 description 1
- 239000011782 vitamin Substances 0.000 description 1
- 235000013343 vitamin Nutrition 0.000 description 1
- 229930003231 vitamin Natural products 0.000 description 1
- HUNXMJYCHXQEGX-UHFFFAOYSA-N zaleplon Chemical compound CCN(C(C)=O)C1=CC=CC(C=2N3N=CC(=C3N=CC=2)C#N)=C1 HUNXMJYCHXQEGX-UHFFFAOYSA-N 0.000 description 1
- 229960004010 zaleplon Drugs 0.000 description 1
- 229910001928 zirconium oxide Inorganic materials 0.000 description 1
- 229960005111 zolpidem tartrate Drugs 0.000 description 1
- 229960000820 zopiclone Drugs 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/02—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4468—Non condensed piperidines, e.g. piperocaine having a nitrogen directly attached in position 4, e.g. clebopride, fentanyl
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1611—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2121/00—Preparations for use in therapy
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Inorganic Chemistry (AREA)
- Neurosurgery (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Cette invention concerne une composition médicale à libération prolongée comprenant un principe pharmaceutique actif et un liant géopolymère. Le principe pharmaceutique actif est de préférence combiné au liant géopolymère pendant la formation dudit liant.
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE0900626 | 2009-05-08 | ||
| SE0900626-3 | 2009-05-08 | ||
| SE1000117 | 2010-02-08 | ||
| SE1000117-0 | 2010-02-08 | ||
| PCT/GB2010/000910 WO2010128300A1 (fr) | 2009-05-08 | 2010-05-07 | Composition pour administration prolongée de médicaments comprenant un liant géopolymère |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CA2761000A1 CA2761000A1 (fr) | 2010-11-11 |
| CA2761000C true CA2761000C (fr) | 2018-05-29 |
Family
ID=42638663
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2761000A Expired - Fee Related CA2761000C (fr) | 2009-05-08 | 2010-05-07 | Composition pour administration prolongee de medicaments comprenant un liant geopolymere |
Country Status (15)
| Country | Link |
|---|---|
| US (2) | US9486527B2 (fr) |
| EP (1) | EP2427177B1 (fr) |
| JP (1) | JP5691051B2 (fr) |
| KR (1) | KR101830080B1 (fr) |
| CN (1) | CN102421419B (fr) |
| AU (1) | AU2010244194B2 (fr) |
| BR (1) | BRPI1011412A8 (fr) |
| CA (1) | CA2761000C (fr) |
| DK (1) | DK2427177T3 (fr) |
| EA (1) | EA027618B1 (fr) |
| ES (1) | ES2673196T3 (fr) |
| IL (1) | IL215826A (fr) |
| MX (1) | MX2011011829A (fr) |
| PL (1) | PL2427177T3 (fr) |
| WO (1) | WO2010128300A1 (fr) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR101830080B1 (ko) * | 2009-05-08 | 2018-02-21 | 엠플리큐어 아베 | 지오폴리머성 결합제를 포함하는 지속형 약물 전달 조성물 |
| DK3254676T3 (en) | 2009-10-30 | 2019-03-11 | Ix Biopharma Ltd | QUICK-SOLVING SOLID DOSAGE FORM |
| US12186426B2 (en) | 2009-10-30 | 2025-01-07 | Ix Biopharma Ltd. | Solid dosage form |
| UA102627C2 (uk) * | 2012-03-20 | 2013-07-25 | Общество С Ограниченной Ответственностью "Наномедтраст" | Нанокомпозит оксид церію-алюмосилікатні трубки та спосіб його отримання |
| IN2014DN09416A (fr) | 2012-04-25 | 2015-07-17 | Spi Pharma Inc | |
| BR112015000320B1 (pt) | 2012-07-12 | 2023-03-07 | SpecGx LLC | Composições farmacêuticas dissuasivas de abuso e seu processo de preparação |
| ES2821528T3 (es) | 2012-11-14 | 2021-04-26 | Grace W R & Co | Composiciones que contienen un material biológicamente activo y un óxido inorgánico no ordenado |
| US20140194328A1 (en) | 2013-01-07 | 2014-07-10 | Vince Alessi | Thermoset ceramic compositions and a method of preparation therefor |
| US20190046743A1 (en) | 2016-02-29 | 2019-02-14 | Emplicure Ab | Devices for evaporation and inhalation of nicotine |
| CN105997907A (zh) * | 2016-05-16 | 2016-10-12 | 胡小丽 | 高血压治疗药丸 |
| CN105769798A (zh) * | 2016-05-16 | 2016-07-20 | 张阳 | 一种高血压治疗药物的制备方法 |
| CN105997915A (zh) * | 2016-05-16 | 2016-10-12 | 张阳 | 一种高血压治疗用缓释片剂 |
| KR102007278B1 (ko) | 2017-01-19 | 2019-08-06 | 가톨릭대학교 산학협력단 | 바이러스 진단 및 치료를 위한 인지능 물질 및 이의 제조방법 |
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-
2010
- 2010-05-07 KR KR1020117029261A patent/KR101830080B1/ko not_active Expired - Fee Related
- 2010-05-07 WO PCT/GB2010/000910 patent/WO2010128300A1/fr not_active Ceased
- 2010-05-07 JP JP2012509085A patent/JP5691051B2/ja not_active Expired - Fee Related
- 2010-05-07 CN CN201080020128.4A patent/CN102421419B/zh not_active Expired - Fee Related
- 2010-05-07 ES ES10718263.6T patent/ES2673196T3/es active Active
- 2010-05-07 BR BRPI1011412A patent/BRPI1011412A8/pt not_active Application Discontinuation
- 2010-05-07 CA CA2761000A patent/CA2761000C/fr not_active Expired - Fee Related
- 2010-05-07 EP EP10718263.6A patent/EP2427177B1/fr active Active
- 2010-05-07 AU AU2010244194A patent/AU2010244194B2/en not_active Ceased
- 2010-05-07 US US13/319,201 patent/US9486527B2/en active Active
- 2010-05-07 PL PL10718263T patent/PL2427177T3/pl unknown
- 2010-05-07 MX MX2011011829A patent/MX2011011829A/es active IP Right Grant
- 2010-05-07 EA EA201101596A patent/EA027618B1/ru not_active IP Right Cessation
- 2010-05-07 DK DK10718263.6T patent/DK2427177T3/en active
-
2011
- 2011-10-23 IL IL215826A patent/IL215826A/en not_active IP Right Cessation
-
2016
- 2016-11-08 US US15/345,877 patent/US10092652B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| CN102421419A (zh) | 2012-04-18 |
| EP2427177A1 (fr) | 2012-03-14 |
| AU2010244194A1 (en) | 2011-11-10 |
| KR20120015344A (ko) | 2012-02-21 |
| BRPI1011412A8 (pt) | 2018-01-02 |
| IL215826A (en) | 2016-11-30 |
| US10092652B2 (en) | 2018-10-09 |
| WO2010128300A1 (fr) | 2010-11-11 |
| IL215826A0 (en) | 2012-01-31 |
| AU2010244194B2 (en) | 2014-12-04 |
| PL2427177T3 (pl) | 2018-09-28 |
| EA027618B1 (ru) | 2017-08-31 |
| CN102421419B (zh) | 2016-05-04 |
| MX2011011829A (es) | 2012-02-21 |
| EA201101596A1 (ru) | 2012-05-30 |
| KR101830080B1 (ko) | 2018-02-21 |
| ES2673196T3 (es) | 2018-06-20 |
| JP2012526091A (ja) | 2012-10-25 |
| BRPI1011412A2 (pt) | 2016-03-15 |
| JP5691051B2 (ja) | 2015-04-01 |
| DK2427177T3 (en) | 2018-06-18 |
| US20170112932A1 (en) | 2017-04-27 |
| US20120252845A1 (en) | 2012-10-04 |
| CA2761000A1 (fr) | 2010-11-11 |
| EP2427177B1 (fr) | 2018-03-28 |
| US9486527B2 (en) | 2016-11-08 |
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