CH530415A - Verfahren zur Herstellung von Pyrimidinderivaten - Google Patents

Verfahren zur Herstellung von Pyrimidinderivaten

Info

Publication number: CH530415A
Authority: CH; Switzerland
Prior art keywords: preparation; pyrimidine derivatives; pyrimidine; derivatives
Prior art date: 1969-08-13

Application number

CH1215970A

Other languages

English (en)

Inventor

Rudolf Dr Albrecht

Eberhard Dr Schroeder

Hans-Joachim Dr Kessler

Original Assignee

Schering Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1969-08-13

Filing date

1970-08-13

Publication date

1972-11-15

1969-08-16 Priority claimed from DE19691941761 external-priority patent/DE1941761C3/de

1970-08-13 Application filed by Schering Ag filed Critical Schering Ag

1972-11-15 Publication of CH530415A publication Critical patent/CH530415A/de

Links

229940083082 pyrimidine derivative acting on arteriolar smooth muscle Drugs 0.000 title 1
150000003230 pyrimidines Chemical class 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61C—DENTISTRY; APPARATUS OR METHODS FOR ORAL OR DENTAL HYGIENE
- A61C19/00—Dental auxiliary appliances
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
- G—PHYSICS
- G03—PHOTOGRAPHY; CINEMATOGRAPHY; ANALOGOUS TECHNIQUES USING WAVES OTHER THAN OPTICAL WAVES; ELECTROGRAPHY; HOLOGRAPHY
- G03B—APPARATUS OR ARRANGEMENTS FOR TAKING PHOTOGRAPHS OR FOR PROJECTING OR VIEWING THEM; APPARATUS OR ARRANGEMENTS EMPLOYING ANALOGOUS TECHNIQUES USING WAVES OTHER THAN OPTICAL WAVES; ACCESSORIES THEREFOR
- G03B17/00—Details of cameras or camera bodies; Accessories therefor
- G03B17/02—Bodies

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Oral & Maxillofacial Surgery (AREA)
Dentistry (AREA)
Epidemiology (AREA)
Physics & Mathematics (AREA)
Animal Behavior & Ethology (AREA)
General Physics & Mathematics (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Heterocyclic Compounds Containing Sulfur Atoms (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

CH1215970A 1969-08-13 1970-08-13 Verfahren zur Herstellung von Pyrimidinderivaten CH530415A (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE19691941575 DE1941575A1 (de)	1969-08-13	1969-08-13	Neue Nitrofurylpyrimidinderivate
DE19691941761 DE1941761C3 (de)		1969-08-16	2-(Thienyl-3 '-amino) -1.3-diazacyclopentene und Verfahren zu ihrer Herstellung

Publications (1)

Publication Number	Publication Date
CH530415A true CH530415A (de)	1972-11-15

Family

ID=25757797

Family Applications (4)

Application Number	Title	Priority Date	Filing Date
CH611473A CH544116A (de)	1969-08-13	1970-08-13	Verfahren zur Herstellung von 2-(Thienyl-3 -amino)-1,3-diazacycloalkenen-(2)
CH611573A CH554894A (de)	1969-08-13	1970-08-13	Verfahren zur herstellung von 2-(thienyl-3'-amino)-1,3diazacycloalkenen-(2).
CH1214570A CH555358A (de)	1969-08-13	1970-08-13	Verfahren zur herstellung von 2-(thienyl-3'-amino)-1,3diazacycloalkenen-(2).
CH1215970A CH530415A (de)	1969-08-13	1970-08-13	Verfahren zur Herstellung von Pyrimidinderivaten

Family Applications Before (3)

Application Number	Title	Priority Date	Filing Date
CH611473A CH544116A (de)	1969-08-13	1970-08-13	Verfahren zur Herstellung von 2-(Thienyl-3 -amino)-1,3-diazacycloalkenen-(2)
CH611573A CH554894A (de)	1969-08-13	1970-08-13	Verfahren zur herstellung von 2-(thienyl-3'-amino)-1,3diazacycloalkenen-(2).
CH1214570A CH555358A (de)	1969-08-13	1970-08-13	Verfahren zur herstellung von 2-(thienyl-3'-amino)-1,3diazacycloalkenen-(2).

Country Status (10)

Country	Link
US (2)	US3758476A (de)
AT (3)	AT310158B (de)
BE (2)	BE754820R (de)
CA (1)	CA1011738A (de)
CH (4)	CH544116A (de)
DE (1)	DE1941575A1 (de)
FR (2)	FR2068493B2 (de)
GB (2)	GB1324646A (de)
NL (2)	NL164859C (de)
SE (1)	SE368406B (de)

Families Citing this family (34)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4036972A (en) *	1973-02-23	1977-07-19	Boehringer Ingelheim Gmbh	2-(N-thienylmethyl-phenylamino)-imidazolines-(2) and salts thereof
DE2308883C3 (de) *	1973-02-23	1978-05-24	C.H. Boehringer Sohn, 6507 Ingelheim	2-Phenylamino-thienylmethyl-imidazoline-(2), Verfahren zur Herstellung derselben und diese enthaltene Arzneimittel
US3919225A (en) *	1974-04-26	1975-11-11	Universal Oil Prod Co	Preparation of N-vinyl substituted amidines
US3919231A (en) *	1974-06-17	1975-11-11	Morton Norwich Products Inc	Series of 5-aryl-2-furamidines
US3970648A (en) *	1974-09-06	1976-07-20	Diamond Shamrock Corporation	2-[2-(5-Nitro-2-furyl)vinyl]-4-(anilino)quinazolines
US4379926A (en) *	1978-05-08	1983-04-12	Ayerst, Mckenna & Harrison Ltd.	1,4,5,6-Tetrahydropyrimidine derivatives
EP0025269B1 (de) *	1979-08-23	1985-11-13	Beecham Group Plc	Veterinärzusammensetzung gegen Diarrhöe
DE19514579A1 (de) *	1995-04-20	1996-10-24	Boehringer Ingelheim Kg	Verwendung von alpha¶1¶¶L¶-Agonisten zur Behandlung der Harninkontinenz
DE10224892A1 (de) *	2002-06-04	2003-12-18	Aventis Pharma Gmbh	Substituierte Thiophene, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament
US7049333B2 (en) *	2002-06-04	2006-05-23	Sanofi-Aventis Deutschland Gmbh	Substituted thiophenes: compositions, processes of making, and uses in disease treatment and diagnosis
US7763280B2 (en) *	2002-11-28	2010-07-27	Boehringer Ingelheim Pharma Gmbh & Co. Kg	Tiotropium containing powder formulation for inhalation
DE10341240A1 (de)	2003-09-08	2005-04-07	Aventis Pharma Deutschland Gmbh	Substituierte Thienoimidazole, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament
CN101027299A (zh) *	2004-09-23	2007-08-29	尤利塞斯药品公司	碳－和杂－环硝基呋喃抗生素及其应用
CA2637292A1 (en) *	2006-01-27	2007-08-16	F. Hoffmann-La Roche Ag	Use of 2-imidazoles for the treatment of cns disorders
AU2007312389B2 (en) *	2006-10-19	2012-02-23	F. Hoffmann-La Roche Ag	Aminomethyl-2-imidazoles with affinity with the trace amine associated receptors
RU2009112496A (ru) *	2006-10-19	2010-11-27	Ф. Хоффманн-Ля Рош Аг (Ch)	Аминометил-4-имидазолы
CA2668454A1 (en) *	2006-11-02	2008-05-08	F. Hoffmann-La Roche Ag	Substituted 2-imidazoles
JP2010510184A (ja) *	2006-11-16	2010-04-02	エフ．ホフマン−ラロシュアーゲー	置換４−イミダゾール類
CA2672617A1 (en) *	2006-12-13	2008-06-19	F. Hoffmann-La Roche Ag	Novel 2-imidazoles as ligands for trace amine associated receptors (taar)
US20080146523A1 (en) *	2006-12-18	2008-06-19	Guido Galley	Imidazole derivatives
CN101600700B (zh) *	2007-02-02	2013-08-21	弗·哈夫曼-拉罗切有限公司	作为taar1配体用于cns病症的新的2-氨基噁唑啉
KR101222412B1 (ko)	2007-02-15	2013-01-15	에프. 호프만-라 로슈 아게	Ｔａａｒ1 리간드로서의 2-아미노옥사졸린
CN101687812A (zh)	2007-07-02	2010-03-31	弗·哈夫曼-拉罗切有限公司	对痕量胺相关受体(taar)具有良好亲和性的2-咪唑啉化合物
CA2691704A1 (en) *	2007-07-03	2009-01-08	F. Hoffmann-La Roche Ag	4-imidazolines and their use as antidepressants
CA2694362A1 (en) *	2007-07-27	2009-02-05	F. Hoffmann-La Roche Ag	2-azetidinemethaneamines and 2-pyrrolidinemethaneamines as taar-ligands
CN101765425A (zh) *	2007-08-02	2010-06-30	弗·哈夫曼-拉罗切有限公司	苯甲酰胺衍生物用于治疗cns障碍的用途
JP5341084B2 (ja) *	2007-08-03	2013-11-13	エフ．ホフマン−ラロシュアーゲー	Ｔａａｒ１リガンドとしてのピリジンカルボキシアミド及びベンズアミド誘導体
CN102083805A (zh) *	2008-07-24	2011-06-01	弗·哈夫曼-拉罗切有限公司	4,5-二氢-唑-2-基衍生物
US8242153B2 (en) *	2008-07-24	2012-08-14	Hoffmann-La Roche Inc.	4,5-dihydro-oxazol-2YL derivatives
US20100311798A1 (en) *	2009-06-05	2010-12-09	Decoret Guillaume	2-aminooxazolines as taar1 ligands
US8354441B2 (en) *	2009-11-11	2013-01-15	Hoffmann-La Roche Inc.	Oxazoline derivatives
US9452980B2 (en)	2009-12-22	2016-09-27	Hoffmann-La Roche Inc.	Substituted benzamides
CN108713019B (zh)	2016-03-17	2021-06-15	豪夫迈·罗氏有限公司	具有作为taar的激动剂的活性的5-乙基-4-甲基-吡唑-3-甲酰胺衍生物
CN111686806B (zh) *	2020-05-29	2022-09-30	黑龙江大学	一种聚[2-(3-噻吩基)乙醇]/石墨相氮化碳复合可见光催化剂的制备方法及应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR5402E (fr) *	1905-06-10	1906-03-27	Camille Durey	Compteur automatique de mouvements d'organes chez les etres animés
DE1695849A1 (de) *	1967-06-23	1971-05-13	Schering Ag	Verfahren zur Herstellung neuer Pyrimidinderivate

0
- BE BE754935D patent/BE754935A/xx not_active IP Right Cessation
- BE BE754820D patent/BE754820R/xx active
1969
- 1969-08-13 DE DE19691941575 patent/DE1941575A1/de active Pending
1970
- 1970-08-06 US US00061853A patent/US3758476A/en not_active Expired - Lifetime
- 1970-08-07 NL NL7011708.A patent/NL164859C/xx not_active IP Right Cessation
- 1970-08-12 FR FR7029657A patent/FR2068493B2/fr not_active Expired
- 1970-08-12 US US00063336A patent/US3814758A/en not_active Expired - Lifetime
- 1970-08-12 NL NL7011933A patent/NL7011933A/xx unknown
- 1970-08-13 CH CH611473A patent/CH544116A/de not_active IP Right Cessation
- 1970-08-13 GB GB3899770A patent/GB1324646A/en not_active Expired
- 1970-08-13 CH CH611573A patent/CH554894A/de not_active IP Right Cessation
- 1970-08-13 CH CH1214570A patent/CH555358A/de not_active IP Right Cessation
- 1970-08-13 CH CH1215970A patent/CH530415A/de not_active IP Right Cessation
- 1970-08-14 AT AT167772A patent/AT310158B/de not_active IP Right Cessation
- 1970-08-14 GB GB3930370A patent/GB1312133A/en not_active Expired
- 1970-08-14 AT AT741970A patent/AT304535B/de not_active IP Right Cessation
- 1970-08-14 CA CA090,785A patent/CA1011738A/en not_active Expired
- 1970-08-14 AT AT167672A patent/AT310157B/de not_active IP Right Cessation
- 1970-08-14 SE SE11112/70A patent/SE368406B/xx unknown
- 1970-08-17 FR FR707030143A patent/FR2068505B1/fr not_active Expired

Also Published As

Publication number	Publication date
CH555358A (de)	1974-10-31
SE368406B (de)	1974-07-01
CA1011738A (en)	1977-06-07
DE1941761A1 (de)	1971-02-25
US3758476A (en)	1973-09-11
BE754935A (fr)	1971-02-17
FR2068493A2 (de)	1971-08-27
FR2068505A1 (de)	1971-08-27
NL7011933A (de)	1971-02-16
US3814758A (en)	1974-06-04
DE1941575A1 (de)	1971-03-04
GB1324646A (en)	1973-07-25
DE1941761B2 (de)	1976-01-08
CH544116A (de)	1973-12-28
NL164859B (nl)	1980-09-15
FR2068505B1 (de)	1973-08-10
FR2068493B2 (de)	1973-12-21
BE754820R (fr)	1971-02-15
AT310157B (de)	1973-09-25
AT310158B (de)	1973-09-25
GB1312133A (en)	1973-04-04
AT304535B (de)	1973-01-10
CH554894A (de)	1974-10-15
NL164859C (nl)	1981-02-16
NL7011708A (de)	1971-02-18

Legal Events

Date	Code	Title	Description
1976-03-15	PL	Patent ceased

Publication	Publication Date	Title
CH530415A (de)	1972-11-15	Verfahren zur Herstellung von Pyrimidinderivaten
AT298508B (de)	1972-05-10	Verfahren zur Herstellung von Mercaptoalkylalkoxysilanen
AT315384B (de)	1974-05-27	Verfahren zur Herstellung von Pyrimidinnucleosiden
CH539642A (de)	1973-09-14	Verfahren zur Herstellung von Pyrimidinylpyrazolderivaten
AT302277B (de)	1972-10-10	Verfahren zur Herstellung von Chinondiiminen
CH552593A (de)	1974-08-15	Verfahren zur herstellung von pyridinthioacetamidderivaten.
CH521934A (de)	1972-04-30	Verfahren zur Herstellung von Buten-2-ol-4-Derivaten
CH529147A (de)	1972-10-15	Verfahren zur Herstellung von s-Triazinderivaten
CH552631A (de)	1974-08-15	Verfahren zur herstellung von n-acylderivaten von phosphoramidothioaten.
AT304774B (de)	1973-01-25	Verfahren zur Herstellung von 16β-Methyl-9α-fluor-steroiden
CH527845A (de)	1972-09-15	Verfahren zur Herstellung von Adenosinderivaten
CH531480A (de)	1972-12-15	Verfahren zur Herstellung von Aminoadamantanen
CH533120A (de)	1973-01-31	Verfahren zur Herstellung von Pyrimidinderivaten
CH532061A (de)	1972-12-31	Verfahren zur Herstellung von Benzodiazepinderivaten
AT296961B (de)	1972-03-10	Verfahren zur Herstellung von Alkyldihydroxybenzolen
AT296995B (de)	1972-03-10	Verfahren zur Herstellung von neuen Aminopyrimidinderivaten
AT300789B (de)	1972-08-10	Verfahren zur Herstellung von Nitroimidazolderivaten
CH544794A (de)	1974-01-15	Verfahren zur Herstellung von 1-Alkoxy-anthrachinonen
CH543486A (de)	1973-10-31	Verfahren zur Herstellung von Malononitrilderivaten
CH533629A (de)	1973-02-15	Verfahren zur Herstellung von Benzodiazepinderivaten
CH523903A (de)	1972-06-15	Verfahren zur Herstellung von substituierten 3-Amino-benzothiophenen
CH538469A (de)	1973-06-30	Verfahren zur Herstellung von substituierten Tetralonen
AT296297B (de)	1972-02-10	Verfahren zur Herstellung von N-Tritylimidazolen und -triazolen
CH532069A (de)	1972-12-31	Verfahren zur Herstellung von 3-Hydroxyisoxazolderivaten
CH523262A (de)	1972-05-31	Verfahren zur Herstellung von Pyrimidinderivaten