CL2008002541A1 - Formulacion topica local que comprende fipronil y un portador veterinariamente aceptable, en ausencia de un inhibidor de la cristalizacion de fipronil; y su uso para controlar ectoparasitos en animales domesticos. - Google Patents

Formulacion topica local que comprende fipronil y un portador veterinariamente aceptable, en ausencia de un inhibidor de la cristalizacion de fipronil; y su uso para controlar ectoparasitos en animales domesticos.

Info

Publication number
CL2008002541A1
CL2008002541A1 CL2008002541A CL2008002541A CL2008002541A1 CL 2008002541 A1 CL2008002541 A1 CL 2008002541A1 CL 2008002541 A CL2008002541 A CL 2008002541A CL 2008002541 A CL2008002541 A CL 2008002541A CL 2008002541 A1 CL2008002541 A1 CL 2008002541A1
Authority
CL
Chile
Prior art keywords
fipronil
absence
acceptable carrier
domestic animals
topical formulation
Prior art date
Application number
CL2008002541A
Other languages
English (en)
Inventor
Keith A Freehauf
Chen Chao Wang
Peter Andrew O'neill
Original Assignee
Schering Plough Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Plough Ltd filed Critical Schering Plough Ltd
Publication of CL2008002541A1 publication Critical patent/CL2008002541A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0014—Skin, i.e. galenical aspects of topical compositions
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/02—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having no bond to a nitrogen atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Dermatology (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Plant Substances (AREA)

Abstract

Formulación tópica local que comprende fipronil y un portador veterinariamente aceptable, en ausencia de un inhibidor de la cristalización de fipronil; y su uso para controlar ectoparásitos en animales domésticos.
CL2008002541A 2007-08-30 2008-08-28 Formulacion topica local que comprende fipronil y un portador veterinariamente aceptable, en ausencia de un inhibidor de la cristalizacion de fipronil; y su uso para controlar ectoparasitos en animales domesticos. CL2008002541A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US96912807P 2007-08-30 2007-08-30

Publications (1)

Publication Number Publication Date
CL2008002541A1 true CL2008002541A1 (es) 2009-01-16

Family

ID=40184969

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2008002541A CL2008002541A1 (es) 2007-08-30 2008-08-28 Formulacion topica local que comprende fipronil y un portador veterinariamente aceptable, en ausencia de un inhibidor de la cristalizacion de fipronil; y su uso para controlar ectoparasitos en animales domesticos.

Country Status (14)

Country Link
US (1) US20110288141A1 (es)
EP (1) EP2194967A2 (es)
JP (1) JP2010536935A (es)
KR (1) KR20100075440A (es)
AU (1) AU2008292070A1 (es)
BR (1) BRPI0815919A2 (es)
CA (1) CA2697943A1 (es)
CL (1) CL2008002541A1 (es)
MX (1) MX2010002270A (es)
NZ (1) NZ583581A (es)
PE (1) PE20090997A1 (es)
RU (1) RU2480197C2 (es)
TW (1) TW200924647A (es)
WO (1) WO2009027506A2 (es)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2010215542A (ja) * 2009-03-13 2010-09-30 Aasu Biochem Kk 非ヒト動物から外部寄生虫を駆除する、または非ヒト動物への外部寄生虫の接触を防ぐための組成物、および当該組成物の利用
GB0905365D0 (en) 2009-03-27 2009-05-13 Norbrook Lab Ltd A topical parasiticide composition
UA108641C2 (uk) 2010-04-02 2015-05-25 Паразитицидна композиція, яка містить чотири активних агенти, та спосіб її застосування
WO2012107585A1 (fr) 2011-02-11 2012-08-16 Ceva Sante Animale Sa Nouvelles compositions antiparasitaires topiques concentrees et stables
US9925167B2 (en) 2011-06-30 2018-03-27 Hansen-Ab Gmbh Agents for the control of parasites on animals
HUE042360T2 (hu) 2011-09-12 2019-06-28 Merial Inc Izoxazolin hatóanyagot tartalmazó parazitaellenes készítmények, ezek elõállítása és alkalmazása
MX374546B (es) * 2012-11-14 2025-03-06 Elanco Us Inc Composiciones farmacéuticas que comprende spinetoram, alcohol bencílico y carbonato de propileno y el uso de la misma como ectoparasiticida en gato.
WO2015017328A2 (en) 2013-07-29 2015-02-05 Spallitta Frank Anthony Organophosphates for treating afflictions of the skin
US11446241B2 (en) 2013-07-29 2022-09-20 Attillaps Holdings Inc. Treatment of ophthalmological conditions with acetylcholinesterase inhibitors
RU2567024C2 (ru) * 2014-01-09 2015-10-27 Федеральное государственное бюджетное научное учреждение "Всероссийский научно-исследовательский институт ветеринарной энтомологии и арахнологии" (ФГБНУ ВИИВЭА) Инсектицидное синергетическое средство
DK3157534T3 (da) 2014-06-19 2022-08-22 Attillaps Holdings Acetylcholinesterasehæmmere til behandling af dermatologiske tilstande
PT3319599T (pt) 2015-07-10 2022-01-28 Ceva Sante Animale Conjunto de partes que combinam uma combinação de dinotefurano/permetrina/piriproxifeno para uso tópico e milbemicina oxime oral para controlar a propagação da dirofilariose
EP3120846A1 (en) * 2015-07-24 2017-01-25 Ceva Sante Animale Compositions and uses thereof for controlling ectoparasites in non-human mammals
GB201520724D0 (en) 2015-11-24 2016-01-06 Merial Inc Veterinary formulations
RU2657752C1 (ru) * 2017-03-29 2018-06-15 Александр Анатольевич Хахалин Инсектоакарицидное средство для лечения и профилактики эктопаразитозов плотоядных животных
RU2692620C1 (ru) * 2018-04-13 2019-06-25 Федеральное государственное бюджетное учреждение науки Федеральный исследовательский центр Тюменский научный центр Сибирского отделения Российской академии наук (ТюмНЦ СО РАН) Способ снижения численности мух на объектах ветеринарно-санитарного надзора

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2753377B1 (fr) * 1996-09-19 1999-09-24 Rhone Merieux Nouvelle association parasiticide a base de 1-n-phenylpyra- zoles et de lactones macrocycliques endectocides
US6426333B1 (en) * 1996-09-19 2002-07-30 Merial Spot-on formulations for combating parasites
US5232940A (en) * 1985-12-20 1993-08-03 Hatton Leslie R Derivatives of N-phenylpyrazoles
FR2739255B1 (fr) * 1995-09-29 1998-09-04 Rhone Merieux Composition antiparasitaire pour le traitement et la protection des animaux de compagnie
US6010710A (en) * 1996-03-29 2000-01-04 Merial Direct pour-on skin solution for antiparasitic use in cattle and sheep
US20050192319A1 (en) * 1996-09-19 2005-09-01 Albert Boeckh Spot-on formulations for combating parasites
US6733767B2 (en) * 1998-03-19 2004-05-11 Merck & Co., Inc. Liquid polymeric compositions for controlled release of bioactive substances
KR100684055B1 (ko) * 1998-03-19 2007-02-16 머크 앤드 캄파니 인코포레이티드 생물활성 물질의 방출 조절용 액체 중합체성 조성물
JP2001139403A (ja) * 1999-11-10 2001-05-22 Sumika Life Tech Co Ltd 動物の外部寄生虫駆除剤
AUPQ441699A0 (en) * 1999-12-02 2000-01-06 Eli Lilly And Company Pour-on formulations
KR20040047962A (ko) 2001-10-25 2004-06-05 상꾜 라이프테크 가부시키가이샤 기생충 구제 조성물
JP2003201204A (ja) * 2001-10-25 2003-07-18 Sankyo Co Ltd 寄生虫駆除組成物
US7262214B2 (en) * 2003-02-26 2007-08-28 Merial Limited 1-N-arylpyrazole derivatives in prevention of arthropod-borne and mosquito-borne diseases
LT1610613T (lt) * 2003-04-04 2017-03-27 Merial, Inc. Vietinio taikymo antihelmintinės veterinarinės kompozicijos
AU2005284422A1 (en) * 2004-09-16 2006-03-23 Bayer Healthcare Ag Dermally applicable formulations for treating skin diseases in animals
SG172705A1 (en) * 2006-09-01 2011-07-28 Du Pont Local topical administration formulations containing indoxacarb

Also Published As

Publication number Publication date
JP2010536935A (ja) 2010-12-02
RU2480197C2 (ru) 2013-04-27
KR20100075440A (ko) 2010-07-02
MX2010002270A (es) 2010-03-17
WO2009027506A3 (en) 2010-02-18
EP2194967A2 (en) 2010-06-16
CA2697943A1 (en) 2009-03-05
PE20090997A1 (es) 2009-07-16
AU2008292070A1 (en) 2009-03-05
NZ583581A (en) 2012-07-27
US20110288141A1 (en) 2011-11-24
TW200924647A (en) 2009-06-16
BRPI0815919A2 (pt) 2015-02-18
RU2010111887A (ru) 2011-10-10
WO2009027506A2 (en) 2009-03-05

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