CL2012001073A1 - Compuestos derivados de pirido[4,3-d]pirimidin-5-ona, sus composiciones farmaceuticas y su uso como inhibidores de quinasa para tratar asma, epoc, colitis ulcerante, bronquitis, lupus, cancer de mamas, enfermedad de alzheimer, enfermedad de parkinson, osteoporosis, esclerosis multiple, diabetes, trastornos oculares, restenosis, enfermedades inflamatorias. - Google Patents

Compuestos derivados de pirido[4,3-d]pirimidin-5-ona, sus composiciones farmaceuticas y su uso como inhibidores de quinasa para tratar asma, epoc, colitis ulcerante, bronquitis, lupus, cancer de mamas, enfermedad de alzheimer, enfermedad de parkinson, osteoporosis, esclerosis multiple, diabetes, trastornos oculares, restenosis, enfermedades inflamatorias.

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Publication number
CL2012001073A1
CL2012001073A1 CL2012001073A CL2012001073A CL2012001073A1 CL 2012001073 A1 CL2012001073 A1 CL 2012001073A1 CL 2012001073 A CL2012001073 A CL 2012001073A CL 2012001073 A CL2012001073 A CL 2012001073A CL 2012001073 A1 CL2012001073 A1 CL 2012001073A1
Authority
CL
Chile
Prior art keywords
alzheimer
disease
pyrido
copd
bronchitis
Prior art date
Application number
CL2012001073A
Other languages
English (en)
Inventor
Hong Woo Kim
Jong Sung Koh
Jaekyoo Lee
Youngsam Kim
Hee Kyu Lee
Jang-Sik Choi
Sun-Hee Lim
Ho-Juhn Song
Original Assignee
Genosco
Oscotec Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43922599&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2012001073(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Genosco, Oscotec Inc filed Critical Genosco
Publication of CL2012001073A1 publication Critical patent/CL2012001073A1/es

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
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    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

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Abstract

Compuestos derivados de pirido[4,3-d]pirimidin-5-ona, como inhibidores de quinasa, útiles para el tratamiento del asma, epoc, colitis ulcerante, bronquitis, lupus, cáncer de mamas, enfermedad de Alzheimer, enfermedad de Parkinson, osteoporosis, entre otras.
CL2012001073A 2009-10-29 2012-04-26 Compuestos derivados de pirido[4,3-d]pirimidin-5-ona, sus composiciones farmaceuticas y su uso como inhibidores de quinasa para tratar asma, epoc, colitis ulcerante, bronquitis, lupus, cancer de mamas, enfermedad de alzheimer, enfermedad de parkinson, osteoporosis, esclerosis multiple, diabetes, trastornos oculares, restenosis, enfermedades inflamatorias. CL2012001073A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US25622209P 2009-10-29 2009-10-29

Publications (1)

Publication Number Publication Date
CL2012001073A1 true CL2012001073A1 (es) 2012-10-26

Family

ID=43922599

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2012001073A CL2012001073A1 (es) 2009-10-29 2012-04-26 Compuestos derivados de pirido[4,3-d]pirimidin-5-ona, sus composiciones farmaceuticas y su uso como inhibidores de quinasa para tratar asma, epoc, colitis ulcerante, bronquitis, lupus, cancer de mamas, enfermedad de alzheimer, enfermedad de parkinson, osteoporosis, esclerosis multiple, diabetes, trastornos oculares, restenosis, enfermedades inflamatorias.

Country Status (18)

Country Link
US (1) US8404677B2 (es)
EP (1) EP2493313B1 (es)
JP (1) JP5993742B2 (es)
KR (1) KR101690358B1 (es)
CN (1) CN102695416B (es)
BR (1) BR112012010085B1 (es)
CA (1) CA2779105C (es)
CL (1) CL2012001073A1 (es)
EA (1) EA029273B1 (es)
ES (1) ES2658290T3 (es)
IL (1) IL219447A (es)
MX (1) MX2012004846A (es)
MY (1) MY173494A (es)
NZ (2) NZ599040A (es)
SG (1) SG10201407012XA (es)
TR (1) TR201802464T4 (es)
WO (1) WO2011053861A1 (es)
ZA (1) ZA201203842B (es)

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