CN106029659B - 谷氨酰胺酶抑制剂 - Google Patents

谷氨酰胺酶抑制剂 Download PDF

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Publication number
CN106029659B
CN106029659B CN201580009614.9A CN201580009614A CN106029659B CN 106029659 B CN106029659 B CN 106029659B CN 201580009614 A CN201580009614 A CN 201580009614A CN 106029659 B CN106029659 B CN 106029659B
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Prior art keywords
acetamido
pyridin
acetamide
thiadiazol
piperidin
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Expired - Fee Related
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CN201580009614.9A
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Chinese (zh)
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CN106029659A (zh
Inventor
普拉尚特·卡希纳特·巴瓦
斯瓦鲁普·库马尔·文卡塔·萨蒂亚·瓦卡拉恩卡
斯里坎坦·维斯瓦纳德哈
买里卡普地·伽雅特里·斯瓦鲁普
戈文达拉朱卢·巴布
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Rhizen Pharmaceuticals AG
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Rhizen Pharmaceuticals AG
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Application filed by Rhizen Pharmaceuticals AG filed Critical Rhizen Pharmaceuticals AG
Priority to CN202010256915.4A priority Critical patent/CN111393431A/zh
Priority to CN202010671865.6A priority patent/CN111892589A/zh
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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