CN112409363B - 用于治疗认知损害的苯并二氮杂䓬衍生物、组合物和方法 - Google Patents

用于治疗认知损害的苯并二氮杂䓬衍生物、组合物和方法 Download PDF

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Publication number: CN112409363B
Authority: CN; China
Prior art keywords: alkyl; compound; cognitive impairment; pharmaceutically acceptable; acceptable salt
Prior art date: 2013-12-20
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Active

Application number

CN202010983158.0A

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English (en)

Chinese (zh)

Other versions

CN112409363A (zh

Inventor

B·梅克纳恩

J·A·巴特拉

黄建星

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Agenebio Inc

Original Assignee

Agenebio Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2013-12-20

Filing date

2014-12-19

Publication date

2023-11-14

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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=53403769&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CN112409363(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2014-12-19 Application filed by Agenebio Inc filed Critical Agenebio Inc

2014-12-19 Priority to CN202010983158.0A priority Critical patent/CN112409363B/zh

2021-02-26 Publication of CN112409363A publication Critical patent/CN112409363A/zh

2023-11-14 Application granted granted Critical

2023-11-14 Publication of CN112409363B publication Critical patent/CN112409363B/zh

Status Active legal-status Critical Current

2034-12-19 Anticipated expiration legal-status Critical

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Classifications

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- C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
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- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
- A61K31/5513—1,4-Benzodiazepines, e.g. diazepam or clozapine
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- C—CHEMISTRY; METALLURGY
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- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
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Hospice & Palliative Care (AREA)
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Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Quinoline Compounds (AREA)
Hydrogenated Pyridines (AREA)
Plural Heterocyclic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

CN202010983158.0A 2013-12-20 2014-12-19 用于治疗认知损害的苯并二氮杂䓬衍生物、组合物和方法 Active CN112409363B (zh)

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US201462075743P	2014-11-05	2014-11-05
US62/075,743		2014-11-05
PCT/US2014/071644 WO2015095783A1 (en)	2013-12-20	2014-12-19	Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment
CN201480073611.7A CN106068256B (zh)	2013-12-20	2014-12-19	用于治疗认知损害的苯并二氮杂*衍生物、组合物和方法
CN202010983158.0A CN112409363B (zh)	2013-12-20	2014-12-19	用于治疗认知损害的苯并二氮杂䓬衍生物、组合物和方法

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CA2934553C (en)	2023-10-31
US10329301B2 (en)	2019-06-25
US20190284196A1 (en)	2019-09-19
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EP3083569A4 (en)	2017-10-04
AU2014368961A2 (en)	2016-11-10
EP4032889A1 (en)	2022-07-27
JP6883988B2 (ja)	2021-06-09
MX2016007808A (es)	2016-09-07
US20170253603A2 (en)	2017-09-07
MX2019010577A (es)	2019-10-21
IL246261B (en)	2021-03-25
MX381561B (es)	2025-03-12
CA3123897C (en)	2024-02-06
CA3123897A1 (en)	2015-06-25
BR112016014564A2 (pt)	2017-08-08
US11142529B2 (en)	2021-10-12
JP2021080287A (ja)	2021-05-27
JP2020011998A (ja)	2020-01-23
EP3083569A1 (en)	2016-10-26
US20170022208A1 (en)	2017-01-26
CN112409363A (zh)	2021-02-26
CN106068256A8 (zh)	2018-10-30
AU2014368961A1 (en)	2016-08-04
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US12528819B2 (en)	2026-01-20	Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment
US12024525B2 (en)	2024-07-02	Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment
JP2021528427A (ja)	2021-10-21	認知障害を処置するためのベンゾジアゼピン誘導体、組成物および方法
HK40046882A (en)	2021-11-12	Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment
HK40057489A (en)	2022-04-14	Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment
HK40077472A (en)	2023-03-10	Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment
HK40049071A (en)	2021-12-10	Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment
HK1230171A1 (en)	2017-12-01	Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment
HK40016046B (en)	2024-02-02	Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment
HK40016046A (en)	2020-09-04	Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment
HK40016541A (en)	2020-09-11	Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment
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