CN1314906A - 帕罗西汀的盐 - Google Patents

帕罗西汀的盐 Download PDF

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Publication number
CN1314906A
CN1314906A CN99810197A CN99810197A CN1314906A CN 1314906 A CN1314906 A CN 1314906A CN 99810197 A CN99810197 A CN 99810197A CN 99810197 A CN99810197 A CN 99810197A CN 1314906 A CN1314906 A CN 1314906A
Authority
CN
China
Prior art keywords
acid
methyl
phenyl
benzoic
amino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CN99810197A
Other languages
English (en)
Chinese (zh)
Inventor
V·W·雅赛维茨
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SmithKline Beecham Ltd
Original Assignee
SmithKline Beecham Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by SmithKline Beecham Ltd filed Critical SmithKline Beecham Ltd
Publication of CN1314906A publication Critical patent/CN1314906A/zh
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Psychology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyridine Compounds (AREA)
CN99810197A 1998-07-02 1999-06-30 帕罗西汀的盐 Pending CN1314906A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9814316.7A GB9814316D0 (en) 1998-07-02 1998-07-02 Novel compounds
GB9814316.7 1998-07-02

Publications (1)

Publication Number Publication Date
CN1314906A true CN1314906A (zh) 2001-09-26

Family

ID=10834803

Family Applications (1)

Application Number Title Priority Date Filing Date
CN99810197A Pending CN1314906A (zh) 1998-07-02 1999-06-30 帕罗西汀的盐

Country Status (21)

Country Link
EP (1) EP1091958A1 (cs)
JP (1) JP2002519421A (cs)
KR (1) KR20010053337A (cs)
CN (1) CN1314906A (cs)
AP (1) AP2000002017A0 (cs)
AU (2) AU4903999A (cs)
BG (1) BG105204A (cs)
BR (1) BR9911679A (cs)
CA (1) CA2336470A1 (cs)
CZ (1) CZ20004923A3 (cs)
EA (1) EA200100098A1 (cs)
GB (1) GB9814316D0 (cs)
HU (1) HUP0103712A3 (cs)
ID (1) ID27766A (cs)
IL (1) IL140385A0 (cs)
NO (1) NO20006547L (cs)
PL (1) PL345365A1 (cs)
SK (1) SK20242000A3 (cs)
TR (1) TR200100055T2 (cs)
WO (1) WO2000001692A1 (cs)
ZA (2) ZA992899B (cs)

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN109212055A (zh) * 2018-08-19 2019-01-15 丁立平 一种测定饮用水中四种痕量单卤代苯乙酸的气相色谱-质谱联用法
CN109342633A (zh) * 2018-11-27 2019-02-15 北京市化工职业病防治院 尿液中苯、甲苯和二甲苯代谢物的检测方法
CN116283778A (zh) * 2023-02-23 2023-06-23 江苏理工学院 一种吡唑羧酸类化合物及其制备方法和应用

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4354984B2 (ja) 2003-05-07 2009-10-28 オステオロジックス エイ／エス 水溶性ストロンチウム塩を用いる軟骨／骨症状の治療
EP2266584B1 (en) 2003-05-07 2012-09-05 Osteologix A/S Composition with strontium and vitamin D for the prophylaxis and/or treatment of cartilage and/or bone conditions
EP1732575B1 (en) 2004-02-26 2010-12-29 Osteologix A/S Strontium-containing compounds for use in the prevention or treatment of necrotic bone conditions
JP4954867B2 (ja) 2004-05-06 2012-06-20 オステオロジックス エイ／エス 有機金属塩類を製造するための高収率で迅速な合成法
KR100672184B1 (ko) * 2004-09-21 2007-01-19 주식회사종근당 파록세틴의 콜린산 또는 콜린산 유도체 염
US9873667B2 (en) 2006-07-27 2018-01-23 Emisphere Technologies Inc. Arylsulfanyl compounds and compositions for delivering active agents
CN111337460B (zh) * 2018-12-18 2021-09-17 中国科学院大连化学物理研究所 一种高稳定性Halo-tag探针及其合成和生物应用
US20250091996A1 (en) 2023-09-15 2025-03-20 King Faisal University 2-(1h-imidazole-1-carbonyl)benzoic acid as an anticancer compound

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8430581D0 (en) * 1984-12-04 1985-01-09 Ferrosan As Treatment
DE3688827T2 (de) * 1985-10-25 1994-03-31 Beecham Group Plc Piperidinderivat, seine Herstellung und seine Verwendung als Arzneimittel.
CA2206592A1 (en) * 1996-05-30 1997-11-30 Shu-Zhong Wang Method of producing amorphous paroxetine hydrochloride
HU221921B1 (hu) * 1996-07-08 2003-02-28 Richter Gedeon Vegyészeti Gyár Rt. N-benzil-piperidin- és tetrahidropiridinszármazékok és eljárás azok előállítására
CZ295301B6 (cs) * 1997-06-10 2005-07-13 Synthon B. V. Deriváty 4-fenylpiperidinu, způsob jejich přípravy, jejich použití a lék je obsahující
CA2319652A1 (en) * 1998-02-06 1999-08-12 Michael Urquhart Salts of paroxetine

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN109212055A (zh) * 2018-08-19 2019-01-15 丁立平 一种测定饮用水中四种痕量单卤代苯乙酸的气相色谱-质谱联用法
CN109212055B (zh) * 2018-08-19 2021-05-07 丁立平 一种测定饮用水中四种痕量单卤代苯乙酸的气相色谱-质谱联用法
CN109342633A (zh) * 2018-11-27 2019-02-15 北京市化工职业病防治院 尿液中苯、甲苯和二甲苯代谢物的检测方法
CN116283778A (zh) * 2023-02-23 2023-06-23 江苏理工学院 一种吡唑羧酸类化合物及其制备方法和应用

Also Published As

Publication number Publication date
NO20006547D0 (no) 2000-12-21
EP1091958A1 (en) 2001-04-18
TR200100055T2 (tr) 2001-07-23
BR9911679A (pt) 2002-01-29
GB9814316D0 (en) 1998-09-02
IL140385A0 (en) 2002-02-10
ID27766A (id) 2001-04-26
PL345365A1 (en) 2001-12-17
AU2002100370A4 (en) 2002-06-06
HUP0103712A2 (hu) 2002-05-29
NO20006547L (no) 2001-02-12
ZA200100020B (en) 2002-03-25
EA200100098A1 (ru) 2001-08-27
AU4903999A (en) 2000-01-24
AP2000002017A0 (en) 2000-12-31
CZ20004923A3 (cs) 2001-08-15
WO2000001692A1 (en) 2000-01-13
KR20010053337A (ko) 2001-06-25
CA2336470A1 (en) 2000-01-13
BG105204A (en) 2001-11-30
SK20242000A3 (sk) 2001-07-10
ZA992899B (en) 2000-03-29
HUP0103712A3 (en) 2002-09-30
JP2002519421A (ja) 2002-07-02

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C06 Publication
C10 Entry into substantive examination
PB01 Publication
SE01 Entry into force of request for substantive examination
C02 Deemed withdrawal of patent application after publication (patent law 2001)
WD01 Invention patent application deemed withdrawn after publication