CN1364159A - 丙酸3－氨基－3－芳基酯的合成 - Google Patents

丙酸3－氨基－3－芳基酯的合成 Download PDF

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Publication number
CN1364159A
CN1364159A CN00807449A CN00807449A CN1364159A CN 1364159 A CN1364159 A CN 1364159A CN 00807449 A CN00807449 A CN 00807449A CN 00807449 A CN00807449 A CN 00807449A CN 1364159 A CN1364159 A CN 1364159A
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CN
China
Prior art keywords
formula
compound
aryl
heteroaryl
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CN00807449A
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English (en)
Chinese (zh)
Inventor
A·F·阿布德尔-马吉德
J·H·科亨
C·A·马亚诺夫
小F·J·维拉尼
H·M·钟
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
3 Dimensional Pharmaceuticals Inc
Original Assignee
3 Dimensional Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 3 Dimensional Pharmaceuticals Inc filed Critical 3 Dimensional Pharmaceuticals Inc
Publication of CN1364159A publication Critical patent/CN1364159A/zh
Pending legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/30—Preparation of optical isomers
    • C07C227/32—Preparation of optical isomers by stereospecific synthesis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07—Optical isomers

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
CN00807449A 1999-03-22 2000-03-21 丙酸3－氨基－3－芳基酯的合成 Pending CN1364159A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US12566999P 1999-03-22 1999-03-22
US60/125,669 1999-03-22

Publications (1)

Publication Number Publication Date
CN1364159A true CN1364159A (zh) 2002-08-14

Family

ID=22420854

Family Applications (1)

Application Number Title Priority Date Filing Date
CN00807449A Pending CN1364159A (zh) 1999-03-22 2000-03-21 丙酸3－氨基－3－芳基酯的合成

Country Status (17)

Country Link
US (3) US6258956B1 (2)
EP (1) EP1163223A1 (2)
JP (1) JP2002540101A (2)
KR (1) KR20020015031A (2)
CN (1) CN1364159A (2)
AU (1) AU776300B2 (2)
BR (1) BR0009856A (2)
CA (1) CA2367971A1 (2)
HR (1) HRP20010768A2 (2)
HU (1) HUP0201263A3 (2)
MX (1) MXPA01009617A (2)
NZ (1) NZ514379A (2)
RU (1) RU2225859C2 (2)
SK (1) SK13592001A3 (2)
UA (1) UA72755C2 (2)
WO (1) WO2000056716A1 (2)
YU (1) YU74501A (2)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20020015031A (ko) 1999-03-22 2002-02-27 오르토-맥네일 파마슈티칼, 인코퍼레이티드 3-아미노-3-아릴 프로파노에이트의 합성
US7907988B2 (en) * 2002-04-01 2011-03-15 Ilan Elias Method and device for generating a passive movement in a diagnostic device
EP2100875B1 (en) 2003-09-18 2016-11-16 Takasago International Corporation Asymmetric reductive amination of keto acid derivatives for producing amino acid derivatives
CA2608845A1 (en) * 2005-05-19 2006-11-23 The Hong Kong Polytechnic University Method for asymmetric alkynylation of alpha-imino esters
CN107879963A (zh) * 2016-09-29 2018-04-06 中国科学院上海药物研究所 新型手性配体、金属螯合物、多种非天然氨基酸、马拉维诺及其关键中间体的合成方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE58243B1 (en) 1983-12-07 1993-08-11 Lonza Ag A process for the preparation of optically-active 3-amino carboxylic acids
US5254573A (en) * 1991-10-15 1993-10-19 Monsanto Company Substituted heterocyclic derivatives useful as platelet aggregation inhibitors
EP0923555B1 (en) * 1996-05-01 2005-06-15 Ortho-McNeil Pharmaceutical, Inc. Carboxamide derivatives of pyrrolidine, piperidine and hexahydroazepine for the treatment of thrombosis disorders
JP2000514809A (ja) 1996-07-12 2000-11-07 ジー．ディー．サール アンド カンパニー キラルβ―アミノ酸の不斉合成
NZ514383A (en) 1999-03-22 2004-01-30 Ortho Mcneil Pharm Inc Process of preparing 3S-3-amino-3-aryl propionic acid and derivatives thereof
CA2368024A1 (en) 1999-03-22 2000-09-28 Ortho-Mcneil Pharmaceutical, Inc. Process for preparing [s-(r*,s*)]-.beta.-[[[1-[1-oxo-3-(4-piperidinyl)propyl]-3-piperidinyl]carbonyl]amino]-3-pyridinepropanoic acid and derivatives
KR20020015031A (ko) 1999-03-22 2002-02-27 오르토-맥네일 파마슈티칼, 인코퍼레이티드 3-아미노-3-아릴 프로파노에이트의 합성

Also Published As

Publication number Publication date
HUP0201263A3 (en) 2003-05-28
YU74501A (sh) 2004-07-15
AU776300B2 (en) 2004-09-02
US20020198400A1 (en) 2002-12-26
MXPA01009617A (es) 2003-07-21
UA72755C2 (en) 2005-04-15
JP2002540101A (ja) 2002-11-26
RU2225859C2 (ru) 2004-03-20
SK13592001A3 (sk) 2002-11-06
NZ514379A (en) 2003-10-31
WO2000056716A1 (en) 2000-09-28
HU0201263D0 (2) 2002-05-29
US6258956B1 (en) 2001-07-10
KR20020015031A (ko) 2002-02-27
HUP0201263A2 (en) 2002-09-28
US20010029300A1 (en) 2001-10-11
EP1163223A1 (en) 2001-12-19
US6610855B2 (en) 2003-08-26
BR0009856A (pt) 2002-02-05
CA2367971A1 (en) 2000-09-28
AU3906400A (en) 2000-10-09
HRP20010768A2 (en) 2002-12-31

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