CO2017005357A2 - Un proceso para la fabricación de idalopirdina - Google Patents

Un proceso para la fabricación de idalopirdina

Info

Publication number: CO2017005357A2
Authority: CO; Colombia
Prior art keywords: idalopirdine; manufacture; describes; preparation; pharmaceutically acceptable
Prior art date: 2014-12-12

Application number

CONC2017/0005357A

Other languages

English (en)

Spanish (es)

Inventor

Mikkel Fog Jacobsen

Ole Nielsen

Original Assignee

H Lundbeck As

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2014-12-12

Filing date

2017-05-26

Publication date

2017-09-20

2015-12-10 Priority claimed from PCT/EP2015/079209 external-priority patent/WO2016091997A1/fr

2017-05-26 Application filed by H Lundbeck As filed Critical H Lundbeck As

2017-09-20 Publication of CO2017005357A2 publication Critical patent/CO2017005357A2/es

Links

YBAWYTYNMZWMMJ-UHFFFAOYSA-N 2-(6-fluoro-1h-indol-3-yl)-n-[[3-(2,2,3,3-tetrafluoropropoxy)phenyl]methyl]ethanamine Chemical compound FC(F)C(F)(F)COC1=CC=CC(CNCCC=2C3=CC=C(F)C=C3NC=2)=C1 YBAWYTYNMZWMMJ-UHFFFAOYSA-N 0.000 title abstract 3
229950005109 idalopirdine Drugs 0.000 title abstract 3
238000000034 method Methods 0.000 title abstract 3
238000004519 manufacturing process Methods 0.000 title abstract 2
150000003839 salts Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
- C07D209/16—Tryptamines
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
- A61K31/405—Indole-alkanecarboxylic acids; Derivatives thereof, e.g. tryptophan, indomethacin
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Indole Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

CONC2017/0005357A 2014-12-12 2017-05-26 Un proceso para la fabricación de idalopirdina CO2017005357A2 (es)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DKPA201400721		2014-12-12
PCT/EP2015/079209 WO2016091997A1 (fr)	2014-12-12	2015-12-10	Procédé de fabrication d'idalopirdine

Publications (1)

Publication Number	Publication Date
CO2017005357A2 true CO2017005357A2 (es)	2017-09-20

Family

ID=59011415

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CONC2017/0005357A CO2017005357A2 (es)	2014-12-12	2017-05-26	Un proceso para la fabricación de idalopirdina

Country Status (13)

Country	Link
EP (1)	EP3230265A1 (fr)
JP (1)	JP2017537128A (fr)
KR (1)	KR20170093821A (fr)
CN (1)	CN107001266A (fr)
AU (1)	AU2015359347A1 (fr)
BR (1)	BR112017012021A2 (fr)
CA (1)	CA2968770A1 (fr)
CL (1)	CL2017001466A1 (fr)
CO (1)	CO2017005357A2 (fr)
IL (1)	IL252471A0 (fr)
MA (1)	MA41148A (fr)
MX (1)	MX2017007510A (fr)
RU (1)	RU2017120216A (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
SG10202010291VA (en)	2014-12-12	2020-11-27	Japan Tobacco Inc	Dihydropyrimidin-2-one compounds and medical use thereof

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3042685A (en) *		1962-07-03		Process of making g-fluoro tryptamine
PE20081889A1 (es) *	2007-03-23	2009-03-05	Smithkline Beecham Corp	Indol carboxamidas como inhibidores de ikk2
TW201139370A (en) *	2009-12-23	2011-11-16	Lundbeck & Co As H	Processes for the manufacture of a pharmaceutically active agent

2015
- 2015-12-09 MA MA041148A patent/MA41148A/fr unknown
- 2015-12-10 MX MX2017007510A patent/MX2017007510A/es unknown
- 2015-12-10 EP EP15821029.4A patent/EP3230265A1/fr not_active Withdrawn
- 2015-12-10 RU RU2017120216A patent/RU2017120216A/ru not_active Application Discontinuation
- 2015-12-10 CN CN201580065028.6A patent/CN107001266A/zh active Pending
- 2015-12-10 KR KR1020177015206A patent/KR20170093821A/ko not_active Withdrawn
- 2015-12-10 JP JP2017531139A patent/JP2017537128A/ja active Pending
- 2015-12-10 AU AU2015359347A patent/AU2015359347A1/en not_active Abandoned
- 2015-12-10 BR BR112017012021A patent/BR112017012021A2/pt not_active Application Discontinuation
- 2015-12-10 CA CA2968770A patent/CA2968770A1/fr not_active Abandoned
2017
- 2017-05-23 IL IL252471A patent/IL252471A0/en unknown
- 2017-05-26 CO CONC2017/0005357A patent/CO2017005357A2/es unknown
- 2017-06-08 CL CL2017001466A patent/CL2017001466A1/es unknown

Also Published As

Publication number	Publication date
CL2017001466A1 (es)	2018-01-05
JP2017537128A (ja)	2017-12-14
CA2968770A1 (fr)	2016-06-16
AU2015359347A1 (en)	2017-06-08
IL252471A0 (en)	2017-07-31
MA41148A (fr)	2017-10-17
BR112017012021A2 (pt)	2018-03-13
CN107001266A (zh)	2017-08-01
KR20170093821A (ko)	2017-08-16
MX2017007510A (es)	2017-08-22
RU2017120216A (ru)	2019-01-15
EP3230265A1 (fr)	2017-10-18

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