CR10038A - Analogo de la diazonamida a - Google Patents

Analogo de la diazonamida a

Info

Publication number
CR10038A
CR10038A CR10038A CR10038A CR10038A CR 10038 A CR10038 A CR 10038A CR 10038 A CR10038 A CR 10038A CR 10038 A CR10038 A CR 10038A CR 10038 A CR10038 A CR 10038A
Authority
CR
Costa Rica
Prior art keywords
diazonamide
analog
conjugates
salts
effective
Prior art date
Application number
CR10038A
Other languages
English (en)
Inventor
Harran Patrick
Williams Noelle
Burgett Anthony
Original Assignee
Univ Texas
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US11/264,502 external-priority patent/US7517895B2/en
Application filed by Univ Texas filed Critical Univ Texas
Publication of CR10038A publication Critical patent/CR10038A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/22—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Un análogo específico de la diazonamida A y sus sales y conjugados, efectivos para el tratamiento de enfermedades proliferactivas.
CR10038A 2005-10-31 2008-05-30 Analogo de la diazonamida a CR10038A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US11/264,502 US7517895B2 (en) 2001-08-24 2005-10-31 Synthetic diazonamides
US81465106P 2006-06-16 2006-06-16

Publications (1)

Publication Number Publication Date
CR10038A true CR10038A (es) 2008-09-12

Family

ID=38006479

Family Applications (1)

Application Number Title Priority Date Filing Date
CR10038A CR10038A (es) 2005-10-31 2008-05-30 Analogo de la diazonamida a

Country Status (8)

Country Link
US (1) US7538129B2 (es)
EP (1) EP1948169A4 (es)
JP (1) JP2009513710A (es)
AU (1) AU2006308849A1 (es)
BR (1) BRPI0618136A2 (es)
CR (1) CR10038A (es)
EA (1) EA013692B1 (es)
WO (1) WO2007053650A2 (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2008154441A1 (en) * 2007-06-07 2008-12-18 Joyant Pharmaceuticals, Inc. Methods for preparing diazonamides
WO2009086170A1 (en) * 2007-12-21 2009-07-09 Joyant Pharmaceuticals, Inc. Diazonamide analogs with improved solubility
JP5123429B2 (ja) * 2008-04-29 2013-01-23 ジョイアント ファーマスーティカルズ、インク. インドリン抗癌剤
WO2009143485A1 (en) * 2008-05-22 2009-11-26 Joyant Pharmaceuticals, Inc. Diazonamide analogs
BR112013027089A2 (pt) 2011-04-22 2017-10-31 Joyant Pharmaceuticals Inc composto, composição farmacêutica e método para usar um composto
US10353032B2 (en) * 2015-10-27 2019-07-16 Halliburton Energy Services, Inc. Viscosity determination apparatus, systems, and methods

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7517895B2 (en) * 2001-08-24 2009-04-14 Board Of Regents, The University Of Texas System Synthetic diazonamides
US7022720B2 (en) * 2001-08-24 2006-04-04 Board Of Regents, The University Of Texas System Synthetic diazonamides as novel anti-mitotic agents

Also Published As

Publication number Publication date
WO2007053650A2 (en) 2007-05-10
US20070149583A1 (en) 2007-06-28
EA200801238A1 (ru) 2008-12-30
BRPI0618136A2 (pt) 2011-08-16
EA013692B1 (ru) 2010-06-30
EP1948169A4 (en) 2009-11-04
WO2007053650A3 (en) 2007-11-22
JP2009513710A (ja) 2009-04-02
EP1948169A2 (en) 2008-07-30
US7538129B2 (en) 2009-05-26
AU2006308849A1 (en) 2007-05-10

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal (granting procedure)