CR10060A - 3-aminociclopentanocarboxamidas como moduladores de receptores de quimioquinas - Google Patents

3-aminociclopentanocarboxamidas como moduladores de receptores de quimioquinas

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Publication number
CR10060A
CR10060A CR10060A CR10060A CR10060A CR 10060 A CR10060 A CR 10060A CR 10060 A CR10060 A CR 10060A CR 10060 A CR10060 A CR 10060A CR 10060 A CR10060 A CR 10060A
Authority
CR
Costa Rica
Prior art keywords
chemiokin
aminociclopentanocarboxamids
receptors modulators
receptors
compounds
Prior art date
Application number
CR10060A
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English (en)
Inventor
Xue Chu-Biao
Original Assignee
Incyte Corp
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Publication date
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Application filed by Incyte Corp filed Critical Incyte Corp
Publication of CR10060A publication Critical patent/CR10060A/es

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
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  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Communicable Diseases (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Rheumatology (AREA)
  • Psychiatry (AREA)
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  • AIDS & HIV (AREA)
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  • Child & Adolescent Psychology (AREA)
  • Transplantation (AREA)

Abstract

La presente invención se refiere a compuestos de Fórmula I: que son moduladores de receptores de quimioquinas. Los compuestos de la invención, y las composiciones de los mismos, son útiles en el tratamiento de enfermedades relacionadas con la expresión y/o actividad de receptores de quimioquinas.
CR10060A 2005-12-21 2008-06-10 3-aminociclopentanocarboxamidas como moduladores de receptores de quimioquinas CR10060A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US75247705P 2005-12-21 2005-12-21
US75232005P 2005-12-21 2005-12-21

Publications (1)

Publication Number Publication Date
CR10060A true CR10060A (es) 2008-07-17

Family

ID=38126410

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Application Number Title Priority Date Filing Date
CR10060A CR10060A (es) 2005-12-21 2008-06-10 3-aminociclopentanocarboxamidas como moduladores de receptores de quimioquinas

Country Status (21)

Country Link
US (2) US7700624B2 (es)
EP (1) EP1971576A2 (es)
JP (1) JP2009520809A (es)
KR (1) KR20080070868A (es)
AP (1) AP2008004487A0 (es)
AR (1) AR058402A1 (es)
AU (1) AU2006327823A1 (es)
BR (1) BRPI0620073A2 (es)
CA (1) CA2634636A1 (es)
CR (1) CR10060A (es)
EA (1) EA200801220A1 (es)
EC (1) ECSP088527A (es)
IL (1) IL191602A0 (es)
MA (1) MA30077B1 (es)
ME (1) MEP1008A (es)
NL (1) NL2000380C2 (es)
NO (1) NO20082285L (es)
RS (1) RS20080246A (es)
TW (1) TW200734323A (es)
UY (1) UY30052A1 (es)
WO (1) WO2007072201A2 (es)

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US7910108B2 (en) 2006-06-05 2011-03-22 Incyte Corporation Sheddase inhibitors combined with CD30-binding immunotherapeutics for the treatment of CD30 positive diseases
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TW201613864A (en) 2014-02-20 2016-04-16 Takeda Pharmaceutical Novel compounds
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AU2020405446A1 (en) 2019-12-20 2022-05-26 Nuevolution A/S Compounds active towards nuclear receptors
BR112022012205A2 (pt) 2019-12-20 2022-09-13 Nuevolution As Compostos ativos para receptores nucleares
JP7713954B2 (ja) 2020-03-31 2025-07-28 ヌエヴォリューション・アクティーゼルスカブ 核内受容体に対して活性な化合物
CA3174252A1 (en) 2020-03-31 2021-10-07 Nuevolution A/S Compounds active towards nuclear receptors
EP4600242A1 (en) 2022-10-07 2025-08-13 Kissei Pharmaceutical Co., Ltd. Cyclopentane compound

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CN1950085A (zh) * 2004-05-11 2007-04-18 因赛特公司 作为趋化因子受体调节剂的3－(4－杂芳基环己基氨基)环戊烷羧酰胺
AU2005259983B2 (en) * 2004-06-28 2011-07-28 Incyte Corporation 3-aminocyclopentanecarboxamides as modulators of chemokine receptors
AP2006003849A0 (en) * 2004-06-28 2006-12-31 Incyte Corp 3-Aminocyclopentanecarboxamides as modulators of chemokine receptors
MEP1008A (xx) * 2005-12-21 2010-02-10 Incyte Corp 3-aminociklopentankarboksamidi kao modulatori receptora hemokina

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US20070149532A1 (en) 2007-06-28
EP1971576A2 (en) 2008-09-24
AU2006327823A1 (en) 2007-06-28
WO2007072201A2 (en) 2007-06-28
ECSP088527A (es) 2008-07-30
JP2009520809A (ja) 2009-05-28
AP2008004487A0 (en) 2008-06-30
KR20080070868A (ko) 2008-07-31
EA200801220A1 (ru) 2008-12-30
CA2634636A1 (en) 2007-06-28
US7700624B2 (en) 2010-04-20
NO20082285L (no) 2008-06-18
AR058402A1 (es) 2008-01-30
BRPI0620073A2 (pt) 2011-11-01
NL2000380C2 (nl) 2007-11-28
MA30077B1 (fr) 2008-12-01
WO2007072201A3 (en) 2007-10-04
IL191602A0 (en) 2009-02-11
US20100203039A1 (en) 2010-08-12
TW200734323A (en) 2007-09-16
MEP1008A (xx) 2010-02-10
NL2000380A1 (nl) 2007-06-25
UY30052A1 (es) 2007-07-31

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