CR10060A - 3-aminociclopentanocarboxamidas como moduladores de receptores de quimioquinas - Google Patents

3-aminociclopentanocarboxamidas como moduladores de receptores de quimioquinas

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Publication number
CR10060A
CR10060A CR10060A CR10060A CR10060A CR 10060 A CR10060 A CR 10060A CR 10060 A CR10060 A CR 10060A CR 10060 A CR10060 A CR 10060A CR 10060 A CR10060 A CR 10060A
Authority
CR
Costa Rica
Prior art keywords
chemiokin
aminociclopentanocarboxamids
receptors modulators
receptors
compounds
Prior art date
Application number
CR10060A
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English (en)
Inventor
Xue Chu-Biao
Original Assignee
Incyte Corp
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Publication date
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Application filed by Incyte Corp filed Critical Incyte Corp
Publication of CR10060A publication Critical patent/CR10060A/es

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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  • Obesity (AREA)
  • Urology & Nephrology (AREA)
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  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
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Abstract

La presente invención se refiere a compuestos de Fórmula I: que son moduladores de receptores de quimioquinas. Los compuestos de la invención, y las composiciones de los mismos, son útiles en el tratamiento de enfermedades relacionadas con la expresión y/o actividad de receptores de quimioquinas.
CR10060A 2005-12-21 2008-06-10 3-aminociclopentanocarboxamidas como moduladores de receptores de quimioquinas CR10060A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US75232005P 2005-12-21 2005-12-21
US75247705P 2005-12-21 2005-12-21

Publications (1)

Publication Number Publication Date
CR10060A true CR10060A (es) 2008-07-17

Family

ID=38126410

Family Applications (1)

Application Number Title Priority Date Filing Date
CR10060A CR10060A (es) 2005-12-21 2008-06-10 3-aminociclopentanocarboxamidas como moduladores de receptores de quimioquinas

Country Status (21)

Country Link
US (2) US7700624B2 (es)
EP (1) EP1971576A2 (es)
JP (1) JP2009520809A (es)
KR (1) KR20080070868A (es)
AP (1) AP2008004487A0 (es)
AR (1) AR058402A1 (es)
AU (1) AU2006327823A1 (es)
BR (1) BRPI0620073A2 (es)
CA (1) CA2634636A1 (es)
CR (1) CR10060A (es)
EA (1) EA200801220A1 (es)
EC (1) ECSP088527A (es)
IL (1) IL191602A0 (es)
MA (1) MA30077B1 (es)
ME (1) MEP1008A (es)
NL (1) NL2000380C2 (es)
NO (1) NO20082285L (es)
RS (1) RS20080246A (es)
TW (1) TW200734323A (es)
UY (1) UY30052A1 (es)
WO (1) WO2007072201A2 (es)

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US7910108B2 (en) 2006-06-05 2011-03-22 Incyte Corporation Sheddase inhibitors combined with CD30-binding immunotherapeutics for the treatment of CD30 positive diseases
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WO2012171863A1 (en) * 2011-06-16 2012-12-20 Boehringer Ingelheim International Gmbh New selective ccr2 antagonists
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CR20170077A (es) 2014-08-04 2017-06-26 Nuevolution As Derivados de heterociclilo opcionalmente condensados de pirimidina útiles para el tratamiento de enfermedades inflamatorias, metabólicas, oncológicas y autoinmunitarias
UY38994A (es) 2019-12-20 2021-07-30 Nuevolution As Compuestos activos frente a receptores nucleares
MX2022007265A (es) 2019-12-20 2022-09-09 Nuevolution As Compuestos activos frente a receptores nucleares.
AU2021245397A1 (en) 2020-03-31 2022-10-20 Nuevolution A/S Compounds active towards nuclear receptors
WO2021198956A1 (en) 2020-03-31 2021-10-07 Nuevolution A/S Compounds active towards nuclear receptors
AR130709A1 (es) 2022-10-07 2025-01-08 Kissei Pharmaceutical Compuesto de ciclopentano

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AU2006327823A1 (en) 2007-06-28
WO2007072201A3 (en) 2007-10-04
EA200801220A1 (ru) 2008-12-30
ECSP088527A (es) 2008-07-30
IL191602A0 (en) 2009-02-11
NL2000380A1 (nl) 2007-06-25
EP1971576A2 (en) 2008-09-24
TW200734323A (en) 2007-09-16
NO20082285L (no) 2008-06-18
JP2009520809A (ja) 2009-05-28
AR058402A1 (es) 2008-01-30
KR20080070868A (ko) 2008-07-31
BRPI0620073A2 (pt) 2011-11-01
MA30077B1 (fr) 2008-12-01
CA2634636A1 (en) 2007-06-28
NL2000380C2 (nl) 2007-11-28
UY30052A1 (es) 2007-07-31
MEP1008A (xx) 2010-02-10
AP2008004487A0 (en) 2008-06-30
US20070149532A1 (en) 2007-06-28
WO2007072201A2 (en) 2007-06-28
US7700624B2 (en) 2010-04-20
US20100203039A1 (en) 2010-08-12
RS20080246A (sr) 2009-07-15

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