CR10169A - "uso de derivados de sulfamida heterociclica benzo-fusionada para disminuir lipidos y disminuir niveles de glucosa en la sangre" - Google Patents

"uso de derivados de sulfamida heterociclica benzo-fusionada para disminuir lipidos y disminuir niveles de glucosa en la sangre"

Info

Publication number
CR10169A
CR10169A CR10169A CR10169A CR10169A CR 10169 A CR10169 A CR 10169A CR 10169 A CR10169 A CR 10169A CR 10169 A CR10169 A CR 10169A CR 10169 A CR10169 A CR 10169A
Authority
CR
Costa Rica
Prior art keywords
decrease
benzo
heterociclic
fusion
blood
Prior art date
Application number
CR10169A
Other languages
English (en)
Inventor
L Smith-Swintosky Virginia
B Reitz Allen
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of CR10169A publication Critical patent/CR10169A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/357—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having two or more oxygen atoms in the same ring, e.g. crown ethers, guanadrel
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A61K31/353—3,4-Dihydrobenzopyrans, e.g. chroman, catechin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Hematology (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Obesity (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Thiazole And Isothizaole Compounds (AREA)

Abstract

La presente invención es un método para los trastornos relacionados con glucosa y trastornos relacionados con lípidos que comprende la administración a un sujeto que lo necesita de una cantidad terapeuticamente efectiva de uno o mas derivados de sulfamida heterocíclica benzo-fusionada novedosos de fórmula (I) o fórmula (II) como se define aquí; la presente invención se refiere además a métodos de tratamiento que comprende la co-terapia con un agente anti-diabético, y agente anti-lipídico y/o un agente anti-obesidad.
CR10169A 2005-12-19 2008-07-21 "uso de derivados de sulfamida heterociclica benzo-fusionada para disminuir lipidos y disminuir niveles de glucosa en la sangre" CR10169A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US75167705P 2005-12-19 2005-12-19
US11/611,961 US8497298B2 (en) 2005-12-19 2006-12-18 Use of benzo-fused heterocycle sulfamide derivatives for lowering lipids and lowering blood glucose levels

Publications (1)

Publication Number Publication Date
CR10169A true CR10169A (es) 2009-01-14

Family

ID=38225368

Family Applications (1)

Application Number Title Priority Date Filing Date
CR10169A CR10169A (es) 2005-12-19 2008-07-21 "uso de derivados de sulfamida heterociclica benzo-fusionada para disminuir lipidos y disminuir niveles de glucosa en la sangre"

Country Status (24)

Country Link
US (1) US8497298B2 (es)
EP (1) EP1973541B1 (es)
JP (1) JP5190374B2 (es)
KR (1) KR101363332B1 (es)
CN (1) CN101365441B (es)
AT (1) ATE486595T1 (es)
AU (1) AU2006337617B8 (es)
BR (1) BRPI0620011A2 (es)
CA (1) CA2634419C (es)
CR (1) CR10169A (es)
CY (1) CY1111161T1 (es)
DE (1) DE602006018066D1 (es)
DK (1) DK1973541T3 (es)
EA (2) EA016892B1 (es)
HR (1) HRP20110008T1 (es)
IL (1) IL192101A (es)
MY (1) MY148866A (es)
NO (1) NO20083003L (es)
NZ (1) NZ569043A (es)
PL (1) PL1973541T3 (es)
PT (1) PT1973541E (es)
RS (1) RS51521B (es)
SI (1) SI1973541T1 (es)
WO (1) WO2007092086A2 (es)

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US8691867B2 (en) 2005-12-19 2014-04-08 Janssen Pharmaceutica Nv Use of benzo-fused heterocycle sulfamide derivatives for the treatment of substance abuse and addiction
US8937096B2 (en) 2005-12-19 2015-01-20 Janssen Pharmaceutica Nv Use of benzo-fused heterocyle sulfamide derivatives for the treatment of mania and bipolar disorder
JP2009537635A (ja) 2006-05-19 2009-10-29 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ 癲癇の処置のための共同−療法
US20090247617A1 (en) * 2008-03-26 2009-10-01 Abdel-Magid Ahmed F Process for the preparation of benzo-fused heteroaryl sulfamates
US20090247616A1 (en) * 2008-03-26 2009-10-01 Smith-Swintosky Virginia L Use of benzo-fused heterocyle sulfamide derivatives for the treatment of anxiety
PE20110060A1 (es) 2008-06-23 2011-01-31 Janssen Pharmaceutica Nv Forma cristalina de (2s)-(-)-n-(6-cloro-2,3-dihidro-benzo[1,4]dioxin-2-ilmetil)-sulfamida
US8815939B2 (en) * 2008-07-22 2014-08-26 Janssen Pharmaceutica Nv Substituted sulfamide derivatives
CA2850513A1 (en) 2011-09-29 2013-04-04 Janssen Pharmaceutica Nv Process for the preparation of sulfamide derivatives
KR20140082762A (ko) 2011-09-29 2014-07-02 얀센 파마슈티카 엔.브이. 설파미드 유도체의 개선된 제조 방법
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CN105232543A (zh) * 2015-11-11 2016-01-13 朱忠良 一种抗糖尿病的口服药物组合物

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HRP20110008T1 (hr) 2011-02-28
EA015606B1 (ru) 2011-10-31
US20070155821A1 (en) 2007-07-05
RS51521B (sr) 2011-06-30
WO2007092086A3 (en) 2007-09-27
JP5190374B2 (ja) 2013-04-24
CA2634419C (en) 2014-10-14
IL192101A0 (en) 2009-08-03
CA2634419A1 (en) 2007-08-16
MY148866A (en) 2013-06-14
EP1973541B1 (en) 2010-11-03
PL1973541T3 (pl) 2011-04-29
HK1125287A1 (en) 2009-08-07
BRPI0620011A2 (pt) 2011-10-25
PT1973541E (pt) 2010-12-14
KR20080089408A (ko) 2008-10-06
CN101365441A (zh) 2009-02-11
NZ569043A (en) 2011-03-31
DE602006018066D1 (de) 2010-12-16
ATE486595T1 (de) 2010-11-15
AU2006337617A1 (en) 2007-08-16
SI1973541T1 (sl) 2011-02-28
KR101363332B1 (ko) 2014-02-19
JP2009520032A (ja) 2009-05-21
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AU2006337617B8 (en) 2013-05-30
CY1111161T1 (el) 2015-06-11
EA016892B1 (ru) 2012-08-30
DK1973541T3 (da) 2011-02-14
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