CR7429A - Composiciones de actuacion prolongada que contienen un compuesto de salicilanilida, una especie de polimero y al menos otro compuesto anti-parasiticida - Google Patents

Composiciones de actuacion prolongada que contienen un compuesto de salicilanilida, una especie de polimero y al menos otro compuesto anti-parasiticida

Info

Publication number
CR7429A
CR7429A CR7429A CR7429A CR7429A CR 7429 A CR7429 A CR 7429A CR 7429 A CR7429 A CR 7429A CR 7429 A CR7429 A CR 7429A CR 7429 A CR7429 A CR 7429A
Authority
CR
Costa Rica
Prior art keywords
compound
salicilanilide
polymer species
compositions containing
another anti
Prior art date
Application number
CR7429A
Other languages
English (en)
Inventor
Lillian Cromie
Sean Duffy
William Blakely
Original Assignee
Norbrook Lab Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Norbrook Lab Ltd filed Critical Norbrook Lab Ltd
Publication of CR7429A publication Critical patent/CR7429A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/275Nitriles; Isonitriles
    • A61K31/277Nitriles; Isonitriles having a ring, e.g. verapamil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/32Macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. carbomers, poly(meth)acrylates, or polyvinyl pyrrolidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Dermatology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Pain & Pain Management (AREA)
  • Inorganic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

Una composicion preparada para el tratamiento de animales con parasitos, parasitos que se saben susceptibles al menos una entre avermectinas, milbemicinas o salicilanilidas, comprende por ejemplo ivermectina en una cantidad comprendida entre el 0,1 y el 10% (p/v), un solvente seleccionado dentro del grupo consistente en glicerol formal, propilenglicol, polietilenglicol y combinaciones de los mismos, y una salicilanilida tal como closantel en una dosis requerida por el animal a ser tratado, habitualmente de alrededor de 2,5 mg/kg vivo de peso del animal a ser tratado, una especie polimerica seleccionada dentro del grupo consistente en polivinilpirrolidona y copolimeros de bloque de polioxipropileno/ polioxietileno, dichas especies polimericas mejoran la biodisponibilidad del closantel en la medida que pueden lograrse niveles en plasma sanguineo de dicho compuesto de mas de alrededor de 20 ppm a lo largo de un periodo de tratamiento.
CR7429A 2002-02-28 2004-08-24 Composiciones de actuacion prolongada que contienen un compuesto de salicilanilida, una especie de polimero y al menos otro compuesto anti-parasiticida CR7429A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB0204712A GB2386066A (en) 2002-02-28 2002-02-28 Long-acting parasiticidal composition with improved bioavailability comprising a salicylanilide, a further anti-parasitic compound & a polymeric species

Publications (1)

Publication Number Publication Date
CR7429A true CR7429A (es) 2006-02-06

Family

ID=9931978

Family Applications (1)

Application Number Title Priority Date Filing Date
CR7429A CR7429A (es) 2002-02-28 2004-08-24 Composiciones de actuacion prolongada que contienen un compuesto de salicilanilida, una especie de polimero y al menos otro compuesto anti-parasiticida

Country Status (23)

Country Link
US (1) US9289380B2 (es)
EP (1) EP1478372B1 (es)
JP (1) JP4480400B2 (es)
AP (1) AP1977A (es)
AR (1) AR038852A1 (es)
AT (1) ATE347897T1 (es)
AU (1) AU2003205887B2 (es)
BR (1) BR0307974B1 (es)
CA (1) CA2476520C (es)
CO (1) CO5611154A2 (es)
CR (1) CR7429A (es)
CY (1) CY1107530T1 (es)
DE (1) DE60310377T2 (es)
DK (1) DK1478372T3 (es)
EC (1) ECSP045320A (es)
ES (1) ES2275076T3 (es)
GB (1) GB2386066A (es)
MX (1) MXPA04007996A (es)
NZ (1) NZ534704A (es)
PT (1) PT1478372E (es)
SI (1) SI1478372T1 (es)
WO (1) WO2003072113A1 (es)
ZA (1) ZA200406782B (es)

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US7666444B2 (en) 2004-02-02 2010-02-23 Wyeth Antiparasitic composition
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WO2006083761A2 (en) 2005-02-03 2006-08-10 Alza Corporation Solvent/polymer solutions as suspension vehicles
US11246913B2 (en) 2005-02-03 2022-02-15 Intarcia Therapeutics, Inc. Suspension formulation comprising an insulinotropic peptide
US20070027105A1 (en) 2005-07-26 2007-02-01 Alza Corporation Peroxide removal from drug delivery vehicle
WO2007140416A2 (en) 2006-05-30 2007-12-06 Intarcia Therapeutics, Inc. Two-piece, internal-channel osmotic delivery system flow modulator
PT2359808E (pt) 2006-08-09 2013-08-28 Intarcia Therapeutics Inc Sistemas de entrega osmótica e montagens de pistão
ES2402172T3 (es) 2007-04-23 2013-04-29 Intarcia Therapeutics, Inc Formulación en suspensión de péptidos insulinotrópicos y usos de los mismos
WO2009102467A2 (en) 2008-02-13 2009-08-20 Intarcia Therapeutics, Inc. Devices, formulations, and methods for delivery of multiple beneficial agents
EP3735944A1 (en) 2009-09-28 2020-11-11 Intarcia Therapeutics, Inc. Rapid establishment and/or termination of substantial steady-state drug delivery
US20120208755A1 (en) 2011-02-16 2012-08-16 Intarcia Therapeutics, Inc. Compositions, Devices and Methods of Use Thereof for the Treatment of Cancers
FR2991173B1 (fr) 2012-06-04 2015-11-06 Virbac Composition veterinaire a administration cutanee a base d'oxyclozanide
HRP20250874T1 (hr) * 2013-09-30 2025-09-26 Zoetis Services Llc Dugodjelujuće formulacije spiro‑izoksazolina
MX385843B (es) 2014-09-12 2025-03-18 Antibiotx Aps Uso antibacteriano de salicilanilidas halogenadas.
US9889085B1 (en) 2014-09-30 2018-02-13 Intarcia Therapeutics, Inc. Therapeutic methods for the treatment of diabetes and related conditions for patients with high baseline HbA1c
GB201509326D0 (en) 2015-05-29 2015-07-15 Antibio Tx Aps Novel use
KR102650751B1 (ko) 2015-06-03 2024-03-22 인타르시아 세라퓨틱스 인코포레이티드 임플란트 배치 및 제거 시스템들
GB201604484D0 (en) * 2016-03-16 2016-04-27 Antibiotx Aps And Københavns Uni University Of Copenhagen Topical antibacterial compositions
CN109310743A (zh) 2016-05-16 2019-02-05 因塔西亚制药公司 胰高血糖素受体选择性多肽及其使用方法
USD860451S1 (en) 2016-06-02 2019-09-17 Intarcia Therapeutics, Inc. Implant removal tool
USD840030S1 (en) 2016-06-02 2019-02-05 Intarcia Therapeutics, Inc. Implant placement guide
AU2018206539A1 (en) 2017-01-03 2019-07-18 Intarcia Therapeutics, Inc. Methods comprising continuous administration of a GLP-1 receptor agonist and co-administration of a drug
US11419834B2 (en) 2019-02-25 2022-08-23 Rhode Island Hospital Methods for treating diseases or infections caused by or associated with H. pylori using a halogenated salicylanilide
EP4090353A4 (en) 2020-01-13 2023-08-09 Durect Corporation DELAYED-RELEASE DRUG DELIVERY SYSTEMS WITH REDUCED IMPURITIES AND RELATED PROCEDURES
JP2024503402A (ja) 2021-01-12 2024-01-25 デュレクト コーポレーション 徐放性薬物送達システム及び関連の方法

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Also Published As

Publication number Publication date
PT1478372E (pt) 2007-01-31
EP1478372A1 (en) 2004-11-24
AU2003205887A1 (en) 2003-09-09
DE60310377T2 (de) 2007-10-31
AU2003205887B2 (en) 2007-02-15
AP2004003142A0 (en) 2004-09-30
DK1478372T3 (da) 2007-04-10
DE60310377D1 (de) 2007-01-25
JP2005525355A (ja) 2005-08-25
AR038852A1 (es) 2005-01-26
NZ534704A (en) 2007-02-23
MXPA04007996A (es) 2004-11-26
CY1107530T1 (el) 2013-03-13
ZA200406782B (en) 2005-07-27
US20050118221A1 (en) 2005-06-02
AP1977A (en) 2009-03-19
CA2476520C (en) 2009-08-11
ATE347897T1 (de) 2007-01-15
GB2386066A (en) 2003-09-10
US9289380B2 (en) 2016-03-22
CA2476520A1 (en) 2003-09-04
CO5611154A2 (es) 2006-02-28
EP1478372B1 (en) 2006-12-13
JP4480400B2 (ja) 2010-06-16
GB0204712D0 (en) 2002-04-17
ES2275076T3 (es) 2007-06-01
ECSP045320A (es) 2004-11-26
BR0307974A (pt) 2004-12-21
BR0307974B1 (pt) 2014-10-21
WO2003072113A1 (en) 2003-09-04
SI1478372T1 (sl) 2007-04-30

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