CR7720A - Acetil 2-hidroxi-1,3- diaminoalcanos - Google Patents

Acetil 2-hidroxi-1,3- diaminoalcanos

Info

Publication number
CR7720A
CR7720A CR7720A CR7720A CR7720A CR 7720 A CR7720 A CR 7720A CR 7720 A CR7720 A CR 7720A CR 7720 A CR7720 A CR 7720A CR 7720 A CR7720 A CR 7720A
Authority
CR
Costa Rica
Prior art keywords
diaminoalcane
hydroxi
oil
compounds
disclosed
Prior art date
Application number
CR7720A
Other languages
English (en)
Inventor
Maillard Michel
T Baldwin Eric
P Beck James
Hughes Robert
Varghese John
R Pulley Shon
Tenbrink Ruth
Original Assignee
Elan Pharm Inc
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Elan Pharm Inc, Upjohn Co filed Critical Elan Pharm Inc
Publication of CR7720A publication Critical patent/CR7720A/es

Links

Landscapes

  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)

Abstract

Se divulgan compuestos de la Formula I. Donde las variables Z,X, R15, R2, R3, Rc son definidas aqui. Los compuestos divulgados aqui son inhibidores de la enzima beta secretasa y por lo tanto, son utiles para el tratamiento de la enfermedad del Alzheimer y otras enfermedades caracterizadas por la deposicion del peptido A beta en un mamifero.
CR7720A 2002-09-10 2005-03-09 Acetil 2-hidroxi-1,3- diaminoalcanos CR7720A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US40945302P 2002-09-10 2002-09-10

Publications (1)

Publication Number Publication Date
CR7720A true CR7720A (es) 2005-07-14

Family

ID=35353421

Family Applications (1)

Application Number Title Priority Date Filing Date
CR7720A CR7720A (es) 2002-09-10 2005-03-09 Acetil 2-hidroxi-1,3- diaminoalcanos

Country Status (5)

Country Link
CN (1) CN100384824C (es)
AP (1) AP2005003247A0 (es)
CR (1) CR7720A (es)
TN (1) TNSN05067A1 (es)
ZA (1) ZA200501991B (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102010030538A1 (de) * 2010-06-25 2011-12-29 Bayer Schering Pharma Aktiengesellschaft 6,7-Dihydro-5H-benzo[7]annulen-Derivate, Verfahren zu ihrer Herstellung, pharmazeutische Präparate die diese enthalten, sowie deren Verwendung zur Herstellung von Arzneimitteln
DE102011087987A1 (de) * 2011-12-08 2013-06-13 Bayer Intellectual Property Gmbh 6,7-Dihydro-5H-benzo[7]annulen-Derivate, Verfahren zu ihrer Herstellung, pharmazeutische Präparate die diese enthalten, sowie deren Verwendung zur Herstellung von Arzneimitteln
SG10202100751YA (en) 2016-07-29 2021-03-30 Sunovion Pharmaceuticals Inc Compounds and compositions and uses thereof
WO2018019291A1 (en) * 2016-07-29 2018-02-01 The Hong Kong University Of Science And Technology C(sp3)-c(sp2) cross-coupling reaction of organozinc reagents and heterocyclic (pseudo)halides
SG11202000669VA (en) 2017-08-02 2020-02-27 Sunovion Pharmaceuticals Inc Isochroman compounds and uses thereof
CN113189089B (zh) * 2021-03-19 2022-05-17 四川轻化工大学 一种臭氧检测试剂及其制备装置和制备方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5482947A (en) * 1990-11-19 1996-01-09 Talley; John J. Retroviral protease inhibitors
AU749281B2 (en) * 1997-02-04 2002-06-20 Regents Of The University Of California, The Nanomolar, non-peptide inhibitors of cathepsin D

Also Published As

Publication number Publication date
CN100384824C (zh) 2008-04-30
CN1694870A (zh) 2005-11-09
ZA200501991B (en) 2006-01-25
TNSN05067A1 (en) 2007-05-14
AP2005003247A0 (en) 2005-03-31

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal (granting procedure)