CR8323A - DERIVATIVES OF TROPANO - Google Patents
DERIVATIVES OF TROPANOInfo
- Publication number
- CR8323A CR8323A CR8323A CR8323A CR8323A CR 8323 A CR8323 A CR 8323A CR 8323 A CR8323 A CR 8323A CR 8323 A CR8323 A CR 8323A CR 8323 A CR8323 A CR 8323A
- Authority
- CR
- Costa Rica
- Prior art keywords
- treatment
- modular
- conditions
- inflammatory diseases
- present
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 abstract 2
- 208000027866 inflammatory disease Diseases 0.000 abstract 2
- 102100035875 C-C chemokine receptor type 5 Human genes 0.000 abstract 1
- 101710149870 C-C chemokine receptor type 5 Proteins 0.000 abstract 1
- 102000004274 CCR5 Receptors Human genes 0.000 abstract 1
- 108010017088 CCR5 Receptors Proteins 0.000 abstract 1
- 208000031886 HIV Infections Diseases 0.000 abstract 1
- 208000037357 HIV infectious disease Diseases 0.000 abstract 1
- 239000005557 antagonist Substances 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 208000033519 human immunodeficiency virus infectious disease Diseases 0.000 abstract 1
- 241001430294 unidentified retrovirus Species 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invencion proporciona compuestos de formula ( I ) en la que R1 y R2 son como se definen anteriormente en la presente memoria. Los compuestos de la presente invencion son modulares, especialmente antagonistas, de la actividad de receptores CCR5 de quimioquinas. Los modulares de receptor CCR5 pueden ser utiles en el tratamiento de diversas enfermedades y afecciones inflamatorias y en el tratamiento de diversas enfermedades y afecciones inflamatorias y en el tratamiento de infeccion por VIH y retrovirus geneticamente relacionados.The present invention provides compounds of formula (I) in which R1 and R2 are as defined hereinbefore. The compounds of the present invention are modular, especially antagonists, of the activity of CCR5 chemokine receptors. The CCR5 receptor modular can be useful in the treatment of various inflammatory diseases and conditions and in the treatment of various inflammatory diseases and conditions and in the treatment of HIV infection and genetically related retroviruses.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0323236.0A GB0323236D0 (en) | 2003-10-03 | 2003-10-03 | Chemical compounds |
| GB0325020A GB0325020D0 (en) | 2003-10-27 | 2003-10-27 | Chemical compounds |
| GB0418556A GB0418556D0 (en) | 2004-08-19 | 2004-08-19 | The treatment of pain |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CR8323A true CR8323A (en) | 2007-12-04 |
Family
ID=44839334
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CR8323A CR8323A (en) | 2003-10-03 | 2006-04-03 | DERIVATIVES OF TROPANO |
Country Status (1)
| Country | Link |
|---|---|
| CR (1) | CR8323A (en) |
-
2006
- 2006-04-03 CR CR8323A patent/CR8323A/en unknown
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