ECSP045344A - USEFUL TROPANO DERIVATIVES IN THERAPY - Google Patents
USEFUL TROPANO DERIVATIVES IN THERAPYInfo
- Publication number
- ECSP045344A ECSP045344A ECSP045344A ECSP045344A EC SP045344 A ECSP045344 A EC SP045344A EC SP045344 A ECSP045344 A EC SP045344A EC SP045344 A ECSP045344 A EC SP045344A
- Authority
- EC
- Ecuador
- Prior art keywords
- useful
- tropano
- therapy
- derivatives
- treatment
- Prior art date
Links
- 238000002560 therapeutic procedure Methods 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 102100035875 C-C chemokine receptor type 5 Human genes 0.000 abstract 1
- 101710149870 C-C chemokine receptor type 5 Proteins 0.000 abstract 1
- 102000004274 CCR5 Receptors Human genes 0.000 abstract 1
- 108010017088 CCR5 Receptors Proteins 0.000 abstract 1
- 208000031886 HIV Infections Diseases 0.000 abstract 1
- 206010061218 Inflammation Diseases 0.000 abstract 1
- 239000005557 antagonist Substances 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 208000027866 inflammatory disease Diseases 0.000 abstract 1
- 230000004054 inflammatory process Effects 0.000 abstract 1
- 241001430294 unidentified retrovirus Species 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invención proporciona compuestos de la fórmula (I) en la que X, Y, R1, R2, R3, R4, R5 y R6 son como se definió anteriormente en la presente memoria. Los compuestos de la presente invención son moduladores, especialmente antagonistas, de la actividad de los receptores CCR5 de quimioquinas. Los moduladores del receptor CCR5 pueden ser útiles para el tratamiento de diversas enfermedades inflamatorias y situaciones con inflamaciones, y para el tratamiento de la infección por el HIV-1 y retrovirus genéticamente relacionados.The present invention provides compounds of the formula (I) in which X, Y, R1, R2, R3, R4, R5 and R6 are as defined hereinbefore. The compounds of the present invention are modulators, especially antagonists, of the activity of CCR5 chemokine receptors. CCR5 receptor modulators can be useful for the treatment of various inflammatory diseases and situations with inflammations, and for the treatment of HIV-1 infection and genetically related retroviruses.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP045344 ECSP045344A (en) | 2004-10-08 | 2004-10-08 | USEFUL TROPANO DERIVATIVES IN THERAPY |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP045344 ECSP045344A (en) | 2004-10-08 | 2004-10-08 | USEFUL TROPANO DERIVATIVES IN THERAPY |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP045344A true ECSP045344A (en) | 2004-11-26 |
Family
ID=40419304
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP045344 ECSP045344A (en) | 2004-10-08 | 2004-10-08 | USEFUL TROPANO DERIVATIVES IN THERAPY |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP045344A (en) |
-
2004
- 2004-10-08 EC ECSP045344 patent/ECSP045344A/en unknown
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