CR8747A - Derivados de tetrahidronaftiridina - Google Patents

Derivados de tetrahidronaftiridina

Info

Publication number
CR8747A
CR8747A CR8747A CR8747A CR8747A CR 8747 A CR8747 A CR 8747A CR 8747 A CR8747 A CR 8747A CR 8747 A CR8747 A CR 8747A CR 8747 A CR8747 A CR 8747A
Authority
CR
Costa Rica
Prior art keywords
derivatives
tetrahydronaftiridine
disorders
preparation
conditions
Prior art date
Application number
CR8747A
Other languages
English (en)
Inventor
Lunn Graham
Paul Mathias John
Sinclair Strang Ross
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of CR8747A publication Critical patent/CR8747A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965—Non-condensed pyrazines
    • A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/16—Otologicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Child & Adolescent Psychology (AREA)
  • Reproductive Health (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Anesthesiology (AREA)
  • Rheumatology (AREA)
  • Otolaryngology (AREA)
  • Endocrinology (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pyridine Compounds (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

La invencion se refiere a derivados de tetrahidronaftiridina y a procedimientos para la preparacion de intermedios usados en la preparacion de composiciones que contienen y los usos de tales derivados. Dichos derivados de tetrahidronaftiridina son ligandos de H3 y son utiles en numerosas enfermedades, trastornos y afecciones, en particular enfermedades, trastornos y afecciones inflamatorias, alergicas y respiratorias.
CR8747A 2004-05-12 2006-11-10 Derivados de tetrahidronaftiridina CR8747A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP04291222A EP1595881A1 (en) 2004-05-12 2004-05-12 Tetrahydronaphthyridine derivates useful as histamine H3 receptor ligands

Publications (1)

Publication Number Publication Date
CR8747A true CR8747A (es) 2006-12-05

Family

ID=34931096

Family Applications (1)

Application Number Title Priority Date Filing Date
CR8747A CR8747A (es) 2004-05-12 2006-11-10 Derivados de tetrahidronaftiridina

Country Status (32)

Country Link
US (2) US7557121B2 (es)
EP (2) EP1595881A1 (es)
JP (1) JP4084410B2 (es)
KR (1) KR100908155B1 (es)
CN (2) CN101798305A (es)
AP (1) AP2006003786A0 (es)
AR (1) AR049092A1 (es)
AT (1) ATE491707T1 (es)
AU (1) AU2005243403B2 (es)
BR (1) BRPI0510762A (es)
CA (1) CA2564201C (es)
CR (1) CR8747A (es)
DE (1) DE602005025345D1 (es)
DK (1) DK1756104T3 (es)
EA (1) EA010487B1 (es)
EC (1) ECSP066984A (es)
ES (1) ES2355572T3 (es)
GE (1) GEP20084552B (es)
GT (1) GT200500112A (es)
IL (1) IL178882A (es)
MA (1) MA28579B1 (es)
MX (1) MXPA06013113A (es)
NL (1) NL1029016C2 (es)
NO (1) NO20064577L (es)
PA (1) PA8632801A1 (es)
PE (1) PE20060312A1 (es)
SV (1) SV2005002112A (es)
TN (1) TNSN06369A1 (es)
TW (1) TW200607506A (es)
UY (1) UY28895A1 (es)
WO (1) WO2005111036A1 (es)
ZA (1) ZA200609111B (es)

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Also Published As

Publication number Publication date
NO20064577L (no) 2006-11-06
AU2005243403B2 (en) 2010-10-07
AP2006003786A0 (en) 2006-10-31
KR20070014174A (ko) 2007-01-31
US7557121B2 (en) 2009-07-07
BRPI0510762A (pt) 2007-11-20
MXPA06013113A (es) 2007-02-28
JP4084410B2 (ja) 2008-04-30
NL1029016C2 (nl) 2006-05-30
EA010487B1 (ru) 2008-10-30
ATE491707T1 (de) 2011-01-15
TNSN06369A1 (fr) 2008-02-22
WO2005111036A1 (en) 2005-11-24
GEP20084552B (en) 2008-11-25
ZA200609111B (en) 2008-08-27
DK1756104T3 (da) 2011-02-21
EA200601897A1 (ru) 2007-02-27
CN101798305A (zh) 2010-08-11
DE602005025345D1 (de) 2011-01-27
CN1950371B (zh) 2011-01-12
NL1029016A1 (nl) 2005-11-15
JP2007536374A (ja) 2007-12-13
IL178882A (en) 2011-03-31
AR049092A1 (es) 2006-06-28
UY28895A1 (es) 2005-12-30
US20090258861A1 (en) 2009-10-15
TW200607506A (en) 2006-03-01
CN1950371A (zh) 2007-04-18
EP1756104B1 (en) 2010-12-15
AU2005243403A1 (en) 2005-11-24
IL178882A0 (en) 2007-03-08
GT200500112A (es) 2005-12-12
SV2005002112A (es) 2005-12-13
MA28579B1 (fr) 2007-05-02
EP1595881A1 (en) 2005-11-16
US20050256135A1 (en) 2005-11-17
CA2564201A1 (en) 2005-11-24
CA2564201C (en) 2011-01-18
PA8632801A1 (es) 2006-06-02
PE20060312A1 (es) 2006-05-03
KR100908155B1 (ko) 2009-07-16
ES2355572T3 (es) 2011-03-29
ECSP066984A (es) 2006-12-29
EP1756104A1 (en) 2007-02-28

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