CR8759A - 3-aminociclopentanocarboxamidas como moduladores de receptores quimioquinas - Google Patents

3-aminociclopentanocarboxamidas como moduladores de receptores quimioquinas

Info

Publication number
CR8759A
CR8759A CR8759A CR8759A CR8759A CR 8759 A CR8759 A CR 8759A CR 8759 A CR8759 A CR 8759A CR 8759 A CR8759 A CR 8759A CR 8759 A CR8759 A CR 8759A
Authority
CR
Costa Rica
Prior art keywords
receptors
modulators
chemiokin
aminociclopentanocarboxamids
compounds
Prior art date
Application number
CR8759A
Other languages
English (en)
Inventor
Xue Chu-Biao
Zheng Changsheng
Feng Hao
Xia Michael
Glenn Joseph
Cao Ganfeng
W Metcalf Brian
Original Assignee
Incyte Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Incyte Corp filed Critical Incyte Corp
Publication of CR8759A publication Critical patent/CR8759A/es

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    • C07D309/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D309/08—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/14—Nitrogen atoms not forming part of a nitro radical
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/453—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with oxygen as a ring hetero atom
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
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    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
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    • A61P19/00—Drugs for skeletal disorders
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    • A61P25/00—Drugs for disorders of the nervous system
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    • A61P31/18—Antivirals for RNA viruses for HIV
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
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Abstract

La presente invencion se refiere a compuestos de formula (I): los cuales son moduladores de receptores de quimioquinas.Los compuestos de la invencion, y composiciones de los mismos son utiles en el tratamiento de enfermedades relacionadas con expresion y/o actividad de receptores de quimioquinas.
CR8759A 2004-06-28 2006-11-21 3-aminociclopentanocarboxamidas como moduladores de receptores quimioquinas CR8759A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US58348204P 2004-06-28 2004-06-28
US62448104P 2004-11-01 2004-11-01

Publications (1)

Publication Number Publication Date
CR8759A true CR8759A (es) 2006-12-13

Family

ID=35783315

Family Applications (1)

Application Number Title Priority Date Filing Date
CR8759A CR8759A (es) 2004-06-28 2006-11-21 3-aminociclopentanocarboxamidas como moduladores de receptores quimioquinas

Country Status (22)

Country Link
US (2) US7618970B2 (es)
EP (1) EP1763347A4 (es)
JP (2) JP4116671B2 (es)
KR (1) KR100856155B1 (es)
CN (1) CN102382088A (es)
AP (1) AP2006003848A0 (es)
AR (1) AR052215A1 (es)
AU (1) AU2005259983B2 (es)
BR (1) BRPI0512634A (es)
CA (1) CA2571397C (es)
CR (1) CR8759A (es)
EA (1) EA012649B1 (es)
EC (1) ECSP067121A (es)
GE (1) GEP20094844B (es)
IL (1) IL179735A0 (es)
MA (1) MA28681B1 (es)
MX (1) MXPA06014673A (es)
NO (1) NO20070489L (es)
NZ (1) NZ551673A (es)
TW (1) TWI366458B (es)
UA (1) UA83311C2 (es)
WO (1) WO2006004741A2 (es)

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US20090208485A1 (en) 2009-08-20
BRPI0512634A (pt) 2008-03-25
JP4116671B2 (ja) 2008-07-09
CN102382088A (zh) 2012-03-21
AR052215A1 (es) 2007-03-07
EP1763347A4 (en) 2009-05-20
US8563582B2 (en) 2013-10-22
NO20070489L (no) 2007-03-07
ECSP067121A (es) 2007-01-26
JP2008504298A (ja) 2008-02-14
EA200602243A1 (ru) 2007-04-27
GEP20094844B (en) 2009-11-25
AU2005259983B2 (en) 2011-07-28
CA2571397A1 (en) 2006-01-12
US20060020133A1 (en) 2006-01-26
CA2571397C (en) 2012-05-22
TW200608960A (en) 2006-03-16
EP1763347A2 (en) 2007-03-21
EA012649B1 (ru) 2009-12-30
NZ551673A (en) 2010-11-26
MXPA06014673A (es) 2007-03-26
KR20070024659A (ko) 2007-03-02
AP2006003848A0 (en) 2006-12-31
WO2006004741A3 (en) 2006-05-04
IL179735A0 (en) 2007-05-15
UA83311C2 (en) 2008-06-25
JP2008074878A (ja) 2008-04-03
MA28681B1 (fr) 2007-06-01
KR100856155B1 (ko) 2008-09-03
WO2006004741A2 (en) 2006-01-12
TWI366458B (en) 2012-06-21
US7618970B2 (en) 2009-11-17
AU2005259983A1 (en) 2006-01-12

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