CS204759B1 - 1-cinnamoyloxy-2-(4-/3-chlorpropionyl/phenoxy)ethane andprocess for preparing thereof - Google Patents

1-cinnamoyloxy-2-(4-/3-chlorpropionyl/phenoxy)ethane andprocess for preparing thereof Download PDF

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Publication number
CS204759B1
CS204759B1 CS538479A CS538479A CS204759B1 CS 204759 B1 CS204759 B1 CS 204759B1 CS 538479 A CS538479 A CS 538479A CS 538479 A CS538479 A CS 538479A CS 204759 B1 CS204759 B1 CS 204759B1
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Czechoslovakia
Prior art keywords
phenoxy
cinnamoyloxy
ethane
preparing
added
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CS538479A
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Czech (cs)
Slovak (sk)
Inventor
Ivan Zvara
Ivan Lukac
Pavol Hrdlovic
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Ivan Zvara
Ivan Lukac
Pavol Hrdlovic
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Application filed by Ivan Zvara, Ivan Lukac, Pavol Hrdlovic filed Critical Ivan Zvara
Priority to CS538479A priority Critical patent/CS204759B1/en
Publication of CS204759B1 publication Critical patent/CS204759B1/en

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Description

Vynález sa týká novej zlúčeniny l-einnamoyloxy-2-[4-/3-chlórpropionyl/fenoxý] etánu vzorcaThe present invention relates to a novel compound of 1-einnamoyloxy-2- [4- (3-chloropropionyl) phenoxy] ethane of the formula

Sp6sob přípravy novej zlúčeniny, ktorá nie je známa z literatúry je založený na tom, že na l-cinnamoyloxy-2-fenoxy etán sa pfisobí chloridom kyseliny 3-chlorpropiónovej za přítomnosti bezvodého chloridu hlinitého.A method for the preparation of a novel compound which is not known from the literature is based on the reaction of 1-cinnamoyloxy-2-phenoxy ethane with 3-chloropropionic chloride in the presence of anhydrous aluminum chloride.

Uvedená zlúčenina sa m6že využit na přípravu monoméru, na přípravu polymérov so 8®ft~ ciálnymi vlastnosťami.Said compound can be used for the preparation of the monomer, for the preparation of polymers with 8F-specific properties.

PříkladExample

Do trojhrdlej baňky opatrenej spatným chladičom, miešadlom a deliacim lievikom ša vložilo 11,2 g .(0,084 mol) chloridu hlinitého v 20 ml sírouhlíka, potom pri teplote vodného kúpeTa 15 °C, za miešania sa přidá roztok 7,1 g (0,056 mol) 3-chlórpropionylchloridu v 10 ml sírouhlíka a potom sa kúpeT odstavil a pri teplote miestnosti sa přidával roztok 15 g (0,056 mol) l-cinnamoyloxy-2-fenoxy etánu v 100 ml sírouhlíka. Po přidaní asi štvrti204 75911.2 g (0.084 mol) of aluminum chloride in 20 ml of carbon disulphide was added to a three-necked flask equipped with an inverted condenser, stirrer and separatory funnel, then at a bath temperature of 15 ° C, while stirring a solution of 7.1 g (0.056 mol) was added. 3-chloropropionyl chloride in 10 ml of carbon disulfide and then the bath was removed and a solution of 15 g (0.056 mol) of 1-cinnamoyloxy-2-phenoxy ethane in 100 ml of carbon disulfide was added at room temperature. After adding about a quarter of 204 759

204 7S9 ny roztoku sa reakčná zmes zahriala do mierneho refluxu a přidal sa zvyšok a reakčná zmes sa refluxovala ešte 30 minút. Potom sa rozložila na zmesi ladu a kyseliny chlorovodíkovej Produkt sa extrahoval chloroformom a štyrikřát premyl vodou. Potom sa chloroform vákuovo odpařil. Získala ea svetložltá tuhá látka, ktorá sa krystalizovala z benzénu. Získali sa kryštálý svetlohnedej farby o t.t. 93,5 °C až 95 °C. Výťažok 53,3 %.The solution was heated to gentle reflux and the residue was added and the reaction mixture was refluxed for a further 30 minutes. It was then decomposed into ice / hydrochloric acid. The product was extracted with chloroform and washed four times with water. The chloroform was then evaporated in vacuo. Obtained a light yellow solid which was crystallized from benzene. A pale brown crystalline color of m.p. 93.5 ° C to 95 ° C. Yield 53.3%.

Claims (2)

2 204 7S9 ny roztoku sa reakčně zmes zahriala do mierneho refluxu a přidal sa zvyšok a reakčná zmessa refluxovala ešte 30 minút. Potom sa rozložila na zmesi ladu a kyseliny chlorovodíkovéjProdukt sa extrahoval chloroformom a štyrikrát premyl vodou. Potom sa chloroform vákuovoodpařil. Získala sa svetložltě tuhá látka, ktorá sa krystalizovala z benzénu. Získali sakryStálý svetlohnedej farby o t.t. 93,5 °C až 95 °C. Výťažok 53,3 %· PBEDMET VYNÁLEZU 1/ l-cinnamoyloxy-2-£4-/3-chlorpropionyl/fenox3fJ etán vzorca:The solution was warmed to gentle reflux and the residue was added and the reaction mixture was refluxed for 30 minutes. It was then quenched with ice / hydrochloric acid and extracted with chloroform and washed four times with water. Then, the chloroform was evaporated in vacuo. A light yellow solid was obtained which crystallized from benzene. They got the hell of a steady light brown color with a melt. 93.5 ° C to 95 ° C. Yield 53.3% PBEDMET OF THE INVENTION 1-Cinnamoyloxy-2- [4- (3-chloropropionyl) phenoxy] ethane of formula: 2/ SpOsob přípravy l-cinnamoyloxy-2-£4--/3-chlorpropionyl/-fehoxýJ etánu podlá bodu 1, vy-značujúci sa tým, že na l-cinnamoyloxy-2-fenoXy-etán sa pfisobí chloridom kyseliny3-chlorpropionovej za přítomnosti bezvodáho chloridu hlinitého.2. A process for preparing 1-cinnamoyloxy-2- [4- (3-chloropropionyl) phenoxy] ethane according to claim 1, wherein 3-chloropropionic acid chloride is added to the 1-cinnamoyloxy-2-phenoxy-ethane at the presence of anhydrous aluminum chloride.
CS538479A 1979-08-06 1979-08-06 1-cinnamoyloxy-2-(4-/3-chlorpropionyl/phenoxy)ethane andprocess for preparing thereof CS204759B1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CS538479A CS204759B1 (en) 1979-08-06 1979-08-06 1-cinnamoyloxy-2-(4-/3-chlorpropionyl/phenoxy)ethane andprocess for preparing thereof

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CS538479A CS204759B1 (en) 1979-08-06 1979-08-06 1-cinnamoyloxy-2-(4-/3-chlorpropionyl/phenoxy)ethane andprocess for preparing thereof

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