CS505587A3 - 4-pyridone derivatives, process of their preparation and pharmaceuticalcompositions comprising them - Google Patents

4-pyridone derivatives, process of their preparation and pharmaceuticalcompositions comprising them

Info

Publication number: CS505587A3
Authority: CS; Czechoslovakia
Prior art keywords: pharmaceuticalcompositions; preparation; pyridone derivatives; pyridone; derivatives
Prior art date: 1986-07-04

Application number

CS875055A

Other languages

English (en)

Other versions

CS277415B6 (en

Inventor

Fritz Dr Sauter

Ulrich Dr Dipl Ing Jordis

Manfred Dr Dipl Ing Rudolf

Josef Dr Wieser

Karl Dr Baumann

Original Assignee

Chemie Linz Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1986-07-04

Filing date

1987-07-03

Publication date

1992-08-12

1987-07-03 Application filed by Chemie Linz Ag filed Critical Chemie Linz Ag

1992-08-12 Publication of CS505587A3 publication Critical patent/CS505587A3/cs

1993-03-17 Publication of CS277415B6 publication Critical patent/CS277415B6/cs

Links

MPOYBFYHRQBZPM-UHFFFAOYSA-N 3h-pyridin-4-one Chemical class O=C1CC=NC=C1 MPOYBFYHRQBZPM-UHFFFAOYSA-N 0.000 title 1
239000008194 pharmaceutical composition Substances 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/80—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D211/84—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen directly attached to ring carbon atoms
- C07D211/86—Oxygen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/08—Bridged systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Communicable Diseases (AREA)
Pharmacology & Pharmacy (AREA)
Oncology (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pyridine Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

CS875055A 1986-07-04 1987-07-03 4-pyridone derivatives, process of their preparation and pharmaceutical preparations comprising them CS277415B6 (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE3622509		1986-07-04

Publications (2)

Publication Number	Publication Date
CS505587A3 true CS505587A3 (en)	1992-08-12
CS277415B6 CS277415B6 (en)	1993-03-17

Family

ID=6304401

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CS875055A CS277415B6 (en)	1986-07-04	1987-07-03	4-pyridone derivatives, process of their preparation and pharmaceutical preparations comprising them

Country Status (24)

Country	Link
US (1)	US5045549A (cs)
EP (1)	EP0251308B1 (cs)
JP (1)	JPH07103123B2 (cs)
KR (1)	KR880001595A (cs)
AR (1)	AR245450A1 (cs)
AT (1)	ATE58538T1 (cs)
AU (1)	AU608515B2 (cs)
CS (1)	CS277415B6 (cs)
DD (1)	DD262428A1 (cs)
DE (1)	DE3766299D1 (cs)
DK (1)	DK342187A (cs)
ES (1)	ES2018667B3 (cs)
FI (1)	FI88506C (cs)
GR (1)	GR3001097T3 (cs)
HU (1)	HU197907B (cs)
IL (1)	IL83049A (cs)
MY (1)	MY101261A (cs)
NO (1)	NO166130C (cs)
NZ (1)	NZ220950A (cs)
PH (1)	PH24239A (cs)
PT (1)	PT85257B (cs)
SU (1)	SU1551248A3 (cs)
YU (1)	YU45039B (cs)
ZA (1)	ZA874849B (cs)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IN166416B (cs) *	1985-09-18	1990-05-05	Pfizer
YU46451B (sh) *	1987-04-08	1993-10-20	Chinoin Gyogyszer Es Vegyeszeti Ter Mekek Gyara Rt.	Postupak za dobivanje mešovitih anhidrida hinolin-karboksilne i borne kiseline
JPH02131453A (ja) *	1988-04-15	1990-05-21	Asahi Glass Co Ltd	２―クロロ―４，５―ジフルオロベンゾイルアクリル酸誘導体
JPH072679B2 (ja) *	1988-04-15	1995-01-18	旭硝子株式会社	２―クロロ―４，５―ジフルオロ安息香酸誘導体
WO1989012055A1 (fr) *	1988-06-08	1989-12-14	Kyorin Pharmaceutical Co., Ltd.	Agent antitumoral
JPH02298946A (ja) *	1989-05-15	1990-12-11	Johoku Seihan Center:Kk	製版・版下作製材および製版・版下作製における貼付方法
EP0449445A3 (en) *	1990-03-27	1993-08-25	Pfizer Inc.	Preparation of beta-ketoesters useful in preparing quinolone antibiotics
ES2147721T3 (es)	1990-04-18	2000-10-01	Procter & Gamble Pharma	Quinolonil lactamas antimicrobianas.
FR2692577B1 (fr) *	1992-05-26	1996-02-02	Bouchara Sa	Nouvelles quinolones fluorees, leur procede de preparation et les compositions pharmaceutiques en renfermant.
TW252107B (cs) *	1993-08-27	1995-07-21	Hokuriku Pharmacetical Co Ltd
ES2092963B1 (es) *	1995-04-12	1997-12-16	Sint Quimica Sa	Procedimiento para la preparacion del acido 1-ciclopropil-6-fluoro-1, 4-dihidro-7-(1s,4s)-5-metil-2,5-diazabiciclo(2.2.1) hept-2-il)-4-oxo-3-quinolincarboxilico y sus sales.
SE0003795D0 (sv)	2000-10-20	2000-10-20	Astrazeneca Ab	Pharmaceutically useful compounds
WO2011031745A1 (en)	2009-09-09	2011-03-17	Achaogen, Inc.	Antibacterial fluoroquinolone analogs

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CA1175836A (en) *	1977-09-20	1984-10-09	Marcel Pesson	Production of 1,4-dihydroquinoline-3-carboxylic acid derivatives
DE2808070A1 (de) *	1978-02-24	1979-08-30	Bayer Ag	Verfahren zur herstellung von 4-pyridon-3-carbonsaeuren und/oder deren derivaten
DE3267485D1 (en) *	1981-02-18	1986-01-02	Nippon Shinyaku Co Ltd	Substituted carboxylic acid derivatives
US4499091A (en) *	1982-03-31	1985-02-12	Sterling Drug Inc.	1-Amino (or substituted amino)-1,4-dihydro-4-oxo-6-fluoro-7-heterylquinoline-3-carboxylic acids and their use as antibacterial agents
EP0090424B1 (en) *	1982-03-31	1986-05-28	Sterling Drug Inc.	New quinolone compounds and preparation thereof
NZ208470A (en) *	1983-07-18	1988-06-30	Abbott Lab	6-fluoro-1,4-dihydro-4-oxo-quinoline-3-carboxylic acid derivatives and antibacterial compositions containing such
US4730000A (en) *	1984-04-09	1988-03-08	Abbott Laboratories	Quinoline antibacterial compounds
JPS6056959A (ja) *	1983-07-18	1985-04-02	アボツト　ラボラトリ−ズ	キノリン抗菌性化合物
US4571396A (en) *	1984-04-16	1986-02-18	Warner-Lambert Company	Antibacterial agents
EP0181521A1 (en) *	1984-10-19	1986-05-21	Otsuka Pharmaceutical Co., Ltd.	Antimicrobial 1-substituted Phenyl-4-oxoquinoline-3-carboxylic acid compounds
US4578473A (en) *	1985-04-15	1986-03-25	Warner-Lambert Company	Process for quinoline-3-carboxylic acid antibacterial agents
IN166416B (cs) *	1985-09-18	1990-05-05	Pfizer
DE3601567A1 (de) *	1986-01-21	1987-07-23	Bayer Ag	7-(azabicycloalkyl)-chinoloncarbonsaeure- und -naphthyridon-carbonsaeure-derivate
US4923879A (en) *	1987-07-31	1990-05-08	Warner-Lambert Company	1,8-Naphthyridines and their use as antibacterial agents
US4962108A (en) *	1987-07-31	1990-10-09	Warner-Lambert Company	Antibacterial quinoline compounds
US4962112A (en) *	1987-08-04	1990-10-09	Abbott Laboratories	7-(2-methyl-4-aminopyrrolidinyl)naphthryidine and quinoline compounds
US4780468A (en) *	1987-08-07	1988-10-25	Warner-Lambert Company	8-trifluoromethyl quinolones as antibacterial agents
US4851418A (en) *	1987-08-21	1989-07-25	Warner-Lambert Company	Naphthyridine antibacterial agents containing an α-amino acid in the side chain of the 7-substituent
WO1989005643A1 (en) *	1987-12-18	1989-06-29	Pfizer Inc.	Heterocyclic-substituted quinoline-carboxylic acids
US4920120A (en) *	1988-01-25	1990-04-24	Warner-Lambert Company	Antibacterial agents

1987
- 1987-07-01 IL IL83049A patent/IL83049A/xx not_active IP Right Cessation
- 1987-07-01 FI FI872897A patent/FI88506C/fi not_active IP Right Cessation
- 1987-07-01 AT AT87109461T patent/ATE58538T1/de not_active IP Right Cessation
- 1987-07-01 ES ES87109461T patent/ES2018667B3/es not_active Expired - Lifetime
- 1987-07-01 DE DE8787109461T patent/DE3766299D1/de not_active Expired - Lifetime
- 1987-07-01 EP EP87109461A patent/EP0251308B1/de not_active Expired - Lifetime
- 1987-07-02 NO NO872778A patent/NO166130C/no unknown
- 1987-07-02 YU YU1246/87A patent/YU45039B/xx unknown
- 1987-07-03 JP JP62165560A patent/JPH07103123B2/ja not_active Expired - Lifetime
- 1987-07-03 NZ NZ220950A patent/NZ220950A/xx unknown
- 1987-07-03 PT PT85257A patent/PT85257B/pt not_active IP Right Cessation
- 1987-07-03 ZA ZA874849A patent/ZA874849B/xx unknown
- 1987-07-03 AR AR87308059A patent/AR245450A1/es active
- 1987-07-03 PH PH35494A patent/PH24239A/en unknown
- 1987-07-03 MY MYPI87000937A patent/MY101261A/en unknown
- 1987-07-03 DK DK342187A patent/DK342187A/da not_active Application Discontinuation
- 1987-07-03 AU AU75080/87A patent/AU608515B2/en not_active Ceased
- 1987-07-03 CS CS875055A patent/CS277415B6/cs unknown
- 1987-07-03 SU SU874203001A patent/SU1551248A3/ru active
- 1987-07-03 HU HU873023A patent/HU197907B/hu not_active IP Right Cessation
- 1987-07-04 KR KR1019870007133A patent/KR880001595A/ko not_active Ceased
- 1987-07-06 US US07/070,351 patent/US5045549A/en not_active Expired - Fee Related
- 1987-07-06 DD DD87304673A patent/DD262428A1/de not_active IP Right Cessation
1990
- 1990-11-23 GR GR90400603T patent/GR3001097T3/el unknown

Also Published As

Publication number	Publication date
EP0251308B1 (de)	1990-11-22
NO166130B (no)	1991-02-25
YU45039B (en)	1991-06-30
GR3001097T3 (en)	1992-04-17
NO872778L (no)	1988-01-05
DK342187A (da)	1988-01-05
PT85257B (pt)	1990-03-30
PT85257A (en)	1987-08-01
PH24239A (en)	1990-05-04
MY101261A (en)	1991-08-17
SU1551248A3 (ru)	1990-03-15
FI88506C (fi)	1993-05-25
FI88506B (fi)	1993-02-15
YU124687A (en)	1988-12-31
FI872897A7 (fi)	1988-01-05
DD262428A1 (de)	1988-11-30
JPS6322580A (ja)	1988-01-30
IL83049A0 (en)	1987-12-31
AU608515B2 (en)	1991-04-11
ATE58538T1 (de)	1990-12-15
HUT45060A (en)	1988-05-30
NO166130C (no)	1991-06-05
US5045549A (en)	1991-09-03
CS277415B6 (en)	1993-03-17
ZA874849B (en)	1988-03-30
KR880001595A (ko)	1988-04-25
AU7508087A (en)	1988-01-07
JPH07103123B2 (ja)	1995-11-08
DK342187D0 (da)	1987-07-03
ES2018667B3 (es)	1991-05-01
IL83049A (en)	1991-12-12
DE3766299D1 (de)	1991-01-03
FI872897A0 (fi)	1987-07-01
EP0251308A1 (de)	1988-01-07
HU197907B (en)	1989-06-28
NO872778D0 (no)	1987-07-02
AR245450A1 (es)	1994-01-31
NZ220950A (en)	1990-07-26

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