CU20130031A7 - Sistemas terapéuticos transdérmicos con lámina de protección inhibidora de la cristalización - Google Patents

Sistemas terapéuticos transdérmicos con lámina de protección inhibidora de la cristalización

Info

Publication number
CU20130031A7
CU20130031A7 CUP2013000031A CU20130031A CU20130031A7 CU 20130031 A7 CU20130031 A7 CU 20130031A7 CU P2013000031 A CUP2013000031 A CU P2013000031A CU 20130031 A CU20130031 A CU 20130031A CU 20130031 A7 CU20130031 A7 CU 20130031A7
Authority
CU
Cuba
Prior art keywords
protection sheet
transdermal therapeutic
therapeutic systems
crystallization inhibiting
inhibiting protection
Prior art date
Application number
CUP2013000031A
Other languages
English (en)
Other versions
CU24172B1 (es
Inventor
Estefan Bracht
Ildiko Terebesi
Thomas Langguth
Original Assignee
Bayer Ip Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44653285&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CU20130031(A7) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Ip Gmbh filed Critical Bayer Ip Gmbh
Publication of CU20130031A7 publication Critical patent/CU20130031A7/es
Publication of CU24172B1 publication Critical patent/CU24172B1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
    • A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
    • A61K9/7053—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/30—Oestrogens

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Dermatology (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Gynecology & Obstetrics (AREA)
  • Reproductive Health (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La invención se refiere a formulaciones farmacéuticas, en especial a sistemas terapéuticos transdérmicos, caracterizados porque en la superficie límite entre la lámina de protección desprendible (Release Liner) y la matriz con contenido de principios activos no recristaliza ningún principio activo. En el caso del principio activo, se trata de gestodeno o de un éster de gestodeno en el polímero de matriz sobresaturado y/o de etinilestradiol. La matriz está libre de solubilizantes, inhibidores de la cristalización y dispersantes.
CU20130031A 2010-09-06 2011-09-02 Sistemas terapéuticos transdérmicos con lámina de protección inhibidora de la cristalización CU24172B1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102010040299A DE102010040299A1 (de) 2010-09-06 2010-09-06 Transdermale therapeutische Systeme mit kristallisationsinhibierender Schutzfolie (Release Liner)
PCT/EP2011/065204 WO2012031985A1 (de) 2010-09-06 2011-09-02 Transdermale therapeutische systeme mit kristallisationsinhibierender schutzfolie (release liner)

Publications (2)

Publication Number Publication Date
CU20130031A7 true CU20130031A7 (es) 2013-05-31
CU24172B1 CU24172B1 (es) 2016-04-25

Family

ID=44653285

Family Applications (1)

Application Number Title Priority Date Filing Date
CU20130031A CU24172B1 (es) 2010-09-06 2011-09-02 Sistemas terapéuticos transdérmicos con lámina de protección inhibidora de la cristalización

Country Status (33)

Country Link
US (2) US8557279B2 (es)
EP (1) EP2613771A1 (es)
JP (2) JP6104800B2 (es)
KR (1) KR20130114127A (es)
CN (1) CN103079549B (es)
AP (1) AP3586A (es)
AR (1) AR082907A1 (es)
AU (1) AU2011298892B2 (es)
BR (1) BR112013005305A2 (es)
CA (1) CA2810103C (es)
CL (1) CL2013000636A1 (es)
CO (1) CO6690753A2 (es)
CR (1) CR20130098A (es)
CU (1) CU24172B1 (es)
DE (1) DE102010040299A1 (es)
DO (1) DOP2013000053A (es)
EA (1) EA032575B1 (es)
EC (1) ECSP13012477A (es)
GT (1) GT201300062A (es)
IL (2) IL224980A (es)
MA (1) MA34581B1 (es)
MX (1) MX2013002602A (es)
MY (1) MY162768A (es)
NZ (1) NZ607630A (es)
PE (2) PE20131138A1 (es)
PH (1) PH12013500429A1 (es)
SG (2) SG187941A1 (es)
TN (1) TN2013000087A1 (es)
TW (1) TWI576245B (es)
UA (1) UA110217C2 (es)
UY (1) UY33590A (es)
WO (1) WO2012031985A1 (es)
ZA (1) ZA201301389B (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI630208B (zh) 2008-12-08 2018-07-21 歐陸斯迪公司 二氫羥戊甲嗎啡
GB201309654D0 (en) 2013-05-30 2013-07-17 Euro Celtique Sa Method

Family Cites Families (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH674618A5 (es) 1987-04-02 1990-06-29 Ciba Geigy Ag
ATE132751T1 (de) 1988-10-27 1996-01-15 Schering Ag Mittel zur transdermalen applikation enthaltend gestoden
PT99338A (pt) 1990-10-29 1992-10-30 Alza Corp Processo para a preparacao de composicoes de farmacos anticoncepcionais administradas transdermicamente contendo uma mistura dum estrogeno e gestodeno e dispositivos para a sua administracao transdermica
US5512292A (en) 1990-10-29 1996-04-30 Alza Corporation Transdermal contraceptive formulations methods and devices
DE4210711A1 (de) 1991-10-31 1993-05-06 Schering Ag Berlin Und Bergkamen, 1000 Berlin, De Transdermale therapeutische systeme mit kristallisationsinhibitoren
DE4336557C2 (de) 1993-05-06 1997-07-17 Lohmann Therapie Syst Lts Estradiolhaltiges transdermales therapeutisches System, Verfahren zu seiner Herstellung und seine Verwendung
DE4405898A1 (de) 1994-02-18 1995-08-24 Schering Ag Transdermale therapeutische Systeme enthaltend Sexualsteroide
DE4405899A1 (de) * 1994-02-18 1995-08-24 Schering Ag Mittel zur transdermalen Applikation enthaltend Desogestrel
US5762956A (en) 1996-04-24 1998-06-09 Rutgers, The State University Of New Jersey Transdermal contraceptive delivery system and process
DE19629468A1 (de) * 1996-07-11 1998-01-15 Schering Ag Transdermale therapeutische Systeme
DE19827732A1 (de) * 1998-06-22 1999-12-23 Rottapharm Bv Transdermales System vom Matrix-Typ zur Abgabe von Wirkstoffen mit einer hohen Abgaberate von Steroid-Hormonen und die Verwendung eines derartigen Systems zur Hormonersatztherapie
DE19906152B4 (de) 1999-02-10 2005-02-10 Jenapharm Gmbh & Co. Kg Wirkstoffhaltige Laminate für Transdermalsysteme
JP4841781B2 (ja) 1999-11-24 2011-12-21 アジル・セラピューティクス・インコーポレイテッド 改良された経皮的避妊薬送達系および方法
DE10053375C1 (de) * 2000-10-27 2002-01-24 Lohmann Therapie Syst Lts Transdermale therapeutische Systeme mit lichtempfindlichen Wirkstoffen
AU2002235155A1 (en) 2000-12-05 2002-06-18 Noven Pharmaceuticals, Inc. Crystallization inhibition of drugs in transdermal drug delivery systems
EP1216699A1 (de) 2000-12-21 2002-06-26 Schering Aktiengesellschaft Transdermalsystem enthaltend ein hochpotentes Gestagen
US20030165547A1 (en) * 2001-05-18 2003-09-04 Elisabeth Picard-Lesboueyries Cosmetic uses of 3beta-acetoxy-7-oxo-DHEA
DE10261696A1 (de) * 2002-12-30 2004-07-15 Schwarz Pharma Ag Vorrichtung zur transdermalen Verabreichung von Rotigotin-Base
ATE333271T1 (de) * 2003-02-21 2006-08-15 Schering Ag Uv-stabiles transdermales pflaster
UA89766C2 (en) * 2003-12-12 2010-03-10 Байер Шеринг Фарма Акциенгезельшафт Transdermal delivery system of gestodene
US8668925B2 (en) * 2003-12-12 2014-03-11 Bayer Intellectual Property Gmbh Transdermal delivery of hormones without the need of penetration enhancers
MXPA06006682A (es) 2003-12-12 2006-08-11 Schering Ag Hormonas de administracion transdermica que no necesitan potenciadores de penetracion.
US20060078604A1 (en) * 2004-10-08 2006-04-13 Noven Pharmaceuticals, Inc. Transdermal drug delivery device including an occlusive backing
DE102004062182B4 (de) 2004-12-20 2007-06-06 Bayer Schering Pharma Ag Transdermales Pflaster mit Progesteron A-Spezifische Liganden (PRASL) als Wirkstoff
US8962013B2 (en) * 2005-05-02 2015-02-24 Bayer Intellectual Property Gmbh Multi-layered transdermal system with triazine UV absorber
DE102005050729A1 (de) 2005-10-19 2007-04-26 Schering Ag Verfahren zur präventiven bedarfsweisen hormonalen Kontrazeption
KR20110082142A (ko) * 2008-10-06 2011-07-18 밀란 테크놀로지즈 인코포레이티드 비정질 로티고틴 경피 시스템

Also Published As

Publication number Publication date
PE20131138A1 (es) 2013-10-26
CU24172B1 (es) 2016-04-25
AP2013006787A0 (en) 2013-04-30
WO2012031985A1 (de) 2012-03-15
US20140018751A1 (en) 2014-01-16
CO6690753A2 (es) 2013-06-17
US8557279B2 (en) 2013-10-15
EA032575B1 (ru) 2019-06-28
GT201300062A (es) 2015-01-16
CN103079549A (zh) 2013-05-01
MA34581B1 (fr) 2013-10-02
JP2016216500A (ja) 2016-12-22
JP2013536828A (ja) 2013-09-26
JP6104800B2 (ja) 2017-03-29
TWI576245B (zh) 2017-04-01
AR082907A1 (es) 2013-01-16
MY162768A (en) 2017-07-14
AU2011298892A1 (en) 2013-03-28
CR20130098A (es) 2013-05-15
CA2810103C (en) 2019-06-18
CA2810103A1 (en) 2012-03-15
EP2613771A1 (de) 2013-07-17
DE102010040299A1 (de) 2012-03-08
SG10201506927TA (en) 2015-10-29
NZ607630A (en) 2015-02-27
US20120082714A1 (en) 2012-04-05
IL251124A0 (en) 2017-04-30
MX2013002602A (es) 2013-04-08
TN2013000087A1 (en) 2014-06-25
KR20130114127A (ko) 2013-10-16
PH12013500429A1 (en) 2019-10-07
CN103079549B (zh) 2016-11-02
IL251124B (en) 2020-07-30
ECSP13012477A (es) 2013-04-30
US9060955B2 (en) 2015-06-23
TW201217165A (en) 2012-05-01
UA110217C2 (en) 2015-12-10
BR112013005305A2 (pt) 2016-08-16
PE20180198A1 (es) 2018-01-26
SG187941A1 (en) 2013-04-30
ZA201301389B (en) 2021-05-26
CL2013000636A1 (es) 2013-09-13
DOP2013000053A (es) 2013-07-15
UY33590A (es) 2011-10-31
EA201390246A1 (ru) 2013-09-30
IL224980A (en) 2017-07-31
AU2011298892B2 (en) 2015-03-12
AP3586A (en) 2016-02-10

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