CY2429B1 - Substituted 3,5-diphenyl-1,2,4-triazoles and theiruse as pharmaceutical metal chelators. - Google Patents

Substituted 3,5-diphenyl-1,2,4-triazoles and theiruse as pharmaceutical metal chelators.

Info

Publication number
CY2429B1
CY2429B1 CY0400016A CY0400016A CY2429B1 CY 2429 B1 CY2429 B1 CY 2429B1 CY 0400016 A CY0400016 A CY 0400016A CY 0400016 A CY0400016 A CY 0400016A CY 2429 B1 CY2429 B1 CY 2429B1
Authority
CY
Cyprus
Prior art keywords
theiruse
triazoles
diphenyl
substituted
metal chelators
Prior art date
Application number
CY0400016A
Other languages
English (en)
Inventor
Rene Lattmann
Pierre Acklin
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=4214048&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY2429(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of CY2429B1 publication Critical patent/CY2429B1/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P39/00General protective or antinoxious agents
    • A61P39/04Chelating agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Toxicology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CY0400016A 1996-06-25 2004-02-27 Substituted 3,5-diphenyl-1,2,4-triazoles and theiruse as pharmaceutical metal chelators. CY2429B1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH159396 1996-06-25

Publications (1)

Publication Number Publication Date
CY2429B1 true CY2429B1 (en) 2004-11-12

Family

ID=4214048

Family Applications (2)

Application Number Title Priority Date Filing Date
CY0400016A CY2429B1 (en) 1996-06-25 2004-02-27 Substituted 3,5-diphenyl-1,2,4-triazoles and theiruse as pharmaceutical metal chelators.
CY2007005C CY2007005I2 (el) 1996-06-25 2007-02-09 Υποκατεστημενες 3,5-διφαινυλ-1,2,4-τριαζολες και η χρηση τους ως φαρμακευτικων χηλικων σκευασματων για μεταλλα

Family Applications After (1)

Application Number Title Priority Date Filing Date
CY2007005C CY2007005I2 (el) 1996-06-25 2007-02-09 Υποκατεστημενες 3,5-διφαινυλ-1,2,4-τριαζολες και η χρηση τους ως φαρμακευτικων χηλικων σκευασματων για μεταλλα

Country Status (36)

Country Link
US (3) US6465504B1 (fr)
EP (1) EP0914118B1 (fr)
JP (1) JP3541042B2 (fr)
KR (1) KR100616378B1 (fr)
CN (1) CN1146415C (fr)
AP (1) AP1127A (fr)
AR (1) AR007479A1 (fr)
AT (1) ATE226435T1 (fr)
AU (1) AU718037B2 (fr)
BG (1) BG64248B1 (fr)
BR (1) BR9709973A (fr)
CA (1) CA2255951C (fr)
CY (2) CY2429B1 (fr)
CZ (1) CZ291470B6 (fr)
DE (3) DE122007000020I1 (fr)
DK (1) DK0914118T3 (fr)
ES (1) ES2187785T3 (fr)
FR (1) FR06C0049I2 (fr)
GE (1) GEP20084355B (fr)
HU (1) HU226232B1 (fr)
IL (1) IL127212A0 (fr)
LT (1) LTC0914118I2 (fr)
LU (1) LU91291I2 (fr)
MY (1) MY129541A (fr)
NL (1) NL300248I2 (fr)
NO (3) NO317180B1 (fr)
NZ (1) NZ333308A (fr)
OA (1) OA10946A (fr)
PL (1) PL194758B1 (fr)
PT (1) PT914118E (fr)
RU (1) RU2208010C2 (fr)
SI (1) SI0914118T1 (fr)
SK (1) SK284319B6 (fr)
TR (1) TR199802693T2 (fr)
TW (1) TW533205B (fr)
WO (1) WO1997049395A1 (fr)

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