DD145533A5 - Verfahren zur herstellung von benzodiazepin-derivaten - Google Patents

Verfahren zur herstellung von benzodiazepin-derivaten Download PDF

Info

Publication number
DD145533A5
DD145533A5 DD79214920A DD21492079A DD145533A5 DD 145533 A5 DD145533 A5 DD 145533A5 DD 79214920 A DD79214920 A DD 79214920A DD 21492079 A DD21492079 A DD 21492079A DD 145533 A5 DD145533 A5 DD 145533A5
Authority
DD
German Democratic Republic
Prior art keywords
dihydro
methyl
fluorophenyl
general formula
benzodiazepin
Prior art date
Application number
DD79214920A
Other languages
German (de)
English (en)
Inventor
Albert E Fischli
Andre Szente
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of DD145533A5 publication Critical patent/DD145533A5/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24—Oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DD79214920A 1978-08-11 1979-08-10 Verfahren zur herstellung von benzodiazepin-derivaten DD145533A5 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CH856378 1978-08-11
CH527079 1979-06-06
CH629679 1979-07-05

Publications (1)

Publication Number Publication Date
DD145533A5 true DD145533A5 (de) 1980-12-17

Family

ID=27175157

Family Applications (1)

Application Number Title Priority Date Filing Date
DD79214920A DD145533A5 (de) 1978-08-11 1979-08-10 Verfahren zur herstellung von benzodiazepin-derivaten

Country Status (19)

Country Link
US (3) US4281188A (fr)
EP (1) EP0008421B1 (fr)
AR (1) AR226541A1 (fr)
AU (1) AU528800B2 (fr)
BR (1) BR7905173A (fr)
CA (1) CA1114373A (fr)
CU (1) CU21116A (fr)
DD (1) DD145533A5 (fr)
DE (1) DE2966639D1 (fr)
DK (1) DK336379A (fr)
FI (1) FI68816C (fr)
GR (1) GR72263B (fr)
HU (1) HU182499B (fr)
IL (1) IL57989A (fr)
MC (1) MC1279A1 (fr)
NO (1) NO792615L (fr)
NZ (1) NZ191224A (fr)
PH (1) PH16128A (fr)
PT (1) PT70056A (fr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1163266A (fr) * 1980-07-31 1984-03-06 Albert E. Fischli Derives de benzodiazepine
CA1157855A (fr) * 1980-07-31 1983-11-29 Albert E. Fischli Derives de benzodiazepine
CA1202023A (fr) * 1982-01-19 1986-03-18 Jean-Marie Cassal Benzodiazepines
US5432700A (en) * 1992-12-21 1995-07-11 Ford Motor Company Adaptive active vehicle suspension system
WO2000034267A1 (fr) * 1998-12-04 2000-06-15 Takeda Chemical Industries, Ltd. Procede de production d'un compose d'amide cyclique

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3329701A (en) * 1962-06-14 1967-07-04 Hoffmann La Roche Cyanobenzophenones
BE787117A (fr) * 1971-08-04 1973-02-05 Hoffmann La Roche Derives de benzodiazepine
JPS5418269B2 (fr) * 1972-07-20 1979-07-06
JPS5084590A (fr) * 1973-11-28 1975-07-08
US4141895A (en) * 1977-06-16 1979-02-27 E. I. Du Pont De Nemours And Company Hydroxyquinazolines and their use as intermediates for pharmaceutical agents

Also Published As

Publication number Publication date
PT70056A (en) 1979-09-01
FI68816B (fi) 1985-07-31
EP0008421A3 (en) 1980-05-28
HU182499B (en) 1984-01-30
AR226541A1 (es) 1982-07-30
AU4956979A (en) 1980-02-14
IL57989A (en) 1982-11-30
US4296031A (en) 1981-10-20
US4281188A (en) 1981-07-28
GR72263B (fr) 1983-10-10
MC1279A1 (fr) 1980-05-23
CU21116A (es) 1982-08-24
BR7905173A (pt) 1980-04-22
PH16128A (en) 1983-07-08
AU528800B2 (en) 1983-05-12
CA1114373A (fr) 1981-12-15
FI792482A7 (fi) 1980-02-12
DK336379A (da) 1980-02-12
FI68816C (fi) 1985-11-11
NO792615L (no) 1980-02-12
NZ191224A (en) 1984-07-06
IL57989A0 (en) 1979-12-30
US4294758A (en) 1981-10-13
EP0008421A2 (fr) 1980-03-05
EP0008421B1 (fr) 1984-02-08
DE2966639D1 (en) 1984-03-15

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