DD202557A5 - Verfahren zur herstellung von neuen benzoylphenylpiperidinderivaten - Google Patents

Verfahren zur herstellung von neuen benzoylphenylpiperidinderivaten Download PDF

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Publication number
DD202557A5
DD202557A5 DD82241202A DD24120282A DD202557A5 DD 202557 A5 DD202557 A5 DD 202557A5 DD 82241202 A DD82241202 A DD 82241202A DD 24120282 A DD24120282 A DD 24120282A DD 202557 A5 DD202557 A5 DD 202557A5
Authority
DD
German Democratic Republic
Prior art keywords
group
alkyl group
different
atoms
same
Prior art date
Application number
DD82241202A
Other languages
German (de)
English (en)
Inventor
Bernhard Majoie
Francois Bellamy
Pierre Dodey
Jacques Robin
Original Assignee
Sori Soc Rech Ind
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sori Soc Rech Ind filed Critical Sori Soc Rech Ind
Publication of DD202557A5 publication Critical patent/DD202557A5/de

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
    • C07D295/135—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/04—Immunostimulants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/10—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms
    • C07D211/14—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms with hydrocarbon or substituted hydrocarbon radicals attached to the ring nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40—Oxygen atoms
    • C07D211/44—Oxygen atoms attached in position 4
    • C07D211/46—Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Immunology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DD82241202A 1981-06-29 1982-06-29 Verfahren zur herstellung von neuen benzoylphenylpiperidinderivaten DD202557A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8112745A FR2508445A1 (fr) 1981-06-29 1981-06-29 Nouveaux derives de benzoyl-phenyl-piperidine, leur procede de preparation et leur application, notamment en therapeutique

Publications (1)

Publication Number Publication Date
DD202557A5 true DD202557A5 (de) 1983-09-21

Family

ID=9259970

Family Applications (1)

Application Number Title Priority Date Filing Date
DD82241202A DD202557A5 (de) 1981-06-29 1982-06-29 Verfahren zur herstellung von neuen benzoylphenylpiperidinderivaten

Country Status (26)

Country Link
US (2) US4528294A (2)
EP (1) EP0069012B1 (2)
JP (1) JPS588061A (2)
KR (1) KR880001298B1 (2)
AR (1) AR230048A1 (2)
AT (1) ATE9795T1 (2)
AU (1) AU550320B2 (2)
CA (1) CA1187501A (2)
CS (1) CS235542B2 (2)
DD (1) DD202557A5 (2)
DE (1) DE3260949D1 (2)
DK (1) DK152668C (2)
ES (1) ES513565A0 (2)
FI (1) FI77447C (2)
FR (1) FR2508445A1 (2)
GR (1) GR76401B (2)
HU (1) HU189150B (2)
IE (1) IE53189B1 (2)
IL (2) IL66123A (2)
NO (1) NO160136C (2)
OA (1) OA07133A (2)
PH (1) PH17368A (2)
PT (1) PT75135B (2)
SU (1) SU1147251A3 (2)
YU (1) YU43799B (2)
ZA (1) ZA824536B (2)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL82573A0 (en) * 1986-05-30 1987-11-30 Sori Soc Rech Ind Preparation of benzoylphenyl-piperidine derivatives
FR2620027A1 (fr) * 1987-09-09 1989-03-10 Fournier Innovation Synergie Nouvelle utilisation de la (5-amino-2-(4-methyl-1-piperidinyl)phenyl)-(4-chlorophenyl)-methanone
US6664271B1 (en) 1999-05-21 2003-12-16 Eli Lilly And Company Immunopotentiator agents
EP1286984A2 (en) * 2000-03-10 2003-03-05 Pharmacia Corporation Method for the preparation of tetrahydrobenzothiepines

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3202655A (en) * 1962-04-27 1965-08-24 Yvon G Perron 6-[alpha-substituted-alpha-(2-or 3-heterocyclic) acetamido] penicillanic acid and nontoxic salts thereof
FR1375300A (fr) * 1962-11-13 1964-10-16 Hoffmann La Roche Dérivés de benzophénone et leur préparation
BE637329A (2) * 1962-11-13
FR1403939A (fr) * 1963-06-07 1965-06-25 Hoffmann La Roche Procédé pour la préparation de dérivés de benzodiazépine
US3668199A (en) * 1966-06-13 1972-06-06 Upjohn Co 1,3-aminoalcohols
FR1526708A (fr) * 1966-06-13 1968-05-24 Upjohn Co 1.3-amino-alcools, leurs intermédiaires et dérivés et leur procédé de préparation
FR1530393A (fr) * 1966-07-11 1968-06-21 Hoffmann La Roche Procédé pour la préparation de dérivés de pipéridine
IE34545B1 (en) * 1969-10-01 1975-06-11 Continental Pharma Amino-alcohols,their salts and process for preparing the same
HU167949B (2) * 1973-07-26 1976-01-28
HU167950B (2) * 1973-07-26 1976-01-28
US4064121A (en) * 1973-07-26 1977-12-20 Richter Gedeon Vegyeszeti Gyar Rt. Substituted nitrobenzophenone derivatives and a process for the preparation thereof
US4021563A (en) * 1975-02-06 1977-05-03 Sven Eric Harry Hernestam Method of treating cardiac arrhythmia with γ-piperidino-butyrophenones
IE49998B1 (en) * 1979-08-06 1986-01-22 Merrell Dow Pharma 4-(naphthalenyloxy)piperidine derivatives

Also Published As

Publication number Publication date
OA07133A (fr) 1984-03-31
KR880001298B1 (ko) 1988-07-22
FI822215A0 (fi) 1982-06-21
NO822185L (no) 1982-12-30
KR840000514A (ko) 1984-02-22
CA1187501A (en) 1985-05-21
ES8304936A1 (es) 1983-03-16
IE53189B1 (en) 1988-08-17
AR230048A1 (es) 1984-02-29
DE3260949D1 (en) 1984-11-15
ES513565A0 (es) 1983-03-16
FR2508445B1 (2) 1984-02-10
JPH0127062B2 (2) 1989-05-26
FI77447C (fi) 1989-03-10
DK289382A (da) 1982-12-30
JPS588061A (ja) 1983-01-18
PH17368A (en) 1984-08-06
FI822215L (fi) 1982-12-30
GR76401B (2) 1984-08-10
DK152668C (da) 1988-09-19
AU8542982A (en) 1983-01-06
IL66123A0 (en) 1982-09-30
IE821475L (en) 1982-12-29
YU43799B (en) 1989-12-31
SU1147251A3 (ru) 1985-03-23
US4528294A (en) 1985-07-09
PT75135B (fr) 1984-05-25
EP0069012B1 (fr) 1984-10-10
AU550320B2 (en) 1986-03-20
FR2508445A1 (fr) 1982-12-31
ZA824536B (en) 1983-04-27
IL76287A0 (en) 1986-01-31
US4680402A (en) 1987-07-14
NO160136C (no) 1989-03-15
IL66123A (en) 1986-02-28
FI77447B (fi) 1988-11-30
NO160136B (no) 1988-12-05
DK152668B (da) 1988-04-11
CS235542B2 (en) 1985-05-15
ATE9795T1 (de) 1984-10-15
YU141582A (en) 1985-03-20
PT75135A (fr) 1982-07-01
EP0069012A1 (fr) 1983-01-05
HU189150B (en) 1986-06-30

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