DK0503844T3 - Thienopyridinderivater og farmaceutiske præparater indeholdende disse - Google Patents

Thienopyridinderivater og farmaceutiske præparater indeholdende disse

Info

Publication number: DK0503844T3
Authority: DK; Denmark
Prior art keywords: pharmaceutical compositions; compositions containing; thienopyridine derivatives; lower alkyl; thienopyridine
Prior art date: 1991-03-12

Application number

DK92301901.2T

Other languages

English (en)

Inventor

Akio Ishii

Fumio Suzuki

Yoshikazu Miwa

Ichiro Miki

Hiroaki Hayashi

Shunji Ichikawa

Original Assignee

Kyowa Hakko Kogyo Kk

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1991-03-12

Filing date

1992-03-05

Publication date

1994-11-28

1992-03-05 Application filed by Kyowa Hakko Kogyo Kk filed Critical Kyowa Hakko Kogyo Kk

1994-11-28 Application granted granted Critical

1994-11-28 Publication of DK0503844T3 publication Critical patent/DK0503844T3/da

Links

DBDCNCCRPKTRSD-UHFFFAOYSA-N thieno[3,2-b]pyridine Chemical class C1=CC=C2SC=CC2=N1 DBDCNCCRPKTRSD-UHFFFAOYSA-N 0.000 title abstract 2
239000008194 pharmaceutical composition Substances 0.000 title 1
125000000217 alkyl group Chemical group 0.000 abstract 2
UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
208000019695 Migraine disease Diseases 0.000 abstract 1
230000003474 anti-emetic effect Effects 0.000 abstract 1
239000002111 antiemetic agent Substances 0.000 abstract 1
229940125683 antiemetic agent Drugs 0.000 abstract 1
229910052739 hydrogen Inorganic materials 0.000 abstract 1
239000001257 hydrogen Substances 0.000 abstract 1
206010027599 migraine Diseases 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Psychiatry (AREA)
Pain & Pain Management (AREA)
Hospice & Palliative Care (AREA)
Anesthesiology (AREA)
Addiction (AREA)
Otolaryngology (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

DK92301901.2T 1991-03-12 1992-03-05 Thienopyridinderivater og farmaceutiske præparater indeholdende disse DK0503844T3 (da)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
JP4626691		1991-03-12

Publications (1)

Publication Number	Publication Date
DK0503844T3 true DK0503844T3 (da)	1994-11-28

Family

ID=12742417

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK92301901.2T DK0503844T3 (da)	1991-03-12	1992-03-05	Thienopyridinderivater og farmaceutiske præparater indeholdende disse

Country Status (7)

Country	Link
US (1)	US5155115A (da)
EP (1)	EP0503844B1 (da)
JP (1)	JP3117777B2 (da)
AT (1)	ATE109484T1 (da)
DE (1)	DE69200290T2 (da)
DK (1)	DK0503844T3 (da)
ES (1)	ES2057959T3 (da)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPH05310732A (ja) *	1992-03-12	1993-11-22	Mitsubishi Kasei Corp	シンノリン−３−カルボン酸誘導体
JP2699794B2 (ja) *	1992-03-12	1998-01-19	三菱化学株式会社	チエノ〔３，２−ｂ〕ピリジン誘導体
DE4227747A1 (de) *	1992-08-21	1994-02-24	Basf Ag	Heteroaromatisch kondensierte Hydroxypyridoncarbonsäureamide, deren Herstellung und Verwendung
DE4444815A1 (de) *	1994-12-15	1996-06-20	Merck Patent Gmbh	Thienopyridone
EP1319409A4 (en) *	2000-09-22	2006-05-03	Takeda Pharmaceutical	SOLID PREPARATIONS
WO2003020728A1 (en) *	2001-08-30	2003-03-13	Pharmacia & Upjohn Company	4-THIOXO-4,7-DIHYDRO-THIENO[2,3-b]PYRIDINE-5-CARBOTHIOAMIDES AS ANTIVIRAL AGENTS
AR038118A1 (es)	2002-01-14	2004-12-29	Upjohn Co	Compuestos derivados de la bencinamida del acido 7-oxo-4,7-dihidrotien[2,3-b[piridin-6-carboxilico 3-sustituido que son utiles como antivirales
AR038117A1 (es) *	2002-01-14	2004-12-29	Upjohn Co	Agentes antivirales derivados de la 4- oxo-4,7 -dihidrofuro [2,3-b]piridin-5-carboxamida
AR038294A1 (es) *	2002-01-14	2005-01-12	Upjohn Co	Oxotieno(3,2-b)piridincarboxamidas como agentes antivirales
US7612078B2 (en)	2003-03-31	2009-11-03	Epix Delaware, Inc.	Piperidinylamino-thieno[2,3-D] pyrimidine compounds
US7488736B2 (en)	2004-05-17	2009-02-10	Epix Delaware, Inc.	Thienopyridinone compounds and methods of treatment
US7407966B2 (en) *	2004-10-07	2008-08-05	Epix Delaware, Inc.	Thienopyridinone compounds and methods of treatment
US7576211B2 (en)	2004-09-30	2009-08-18	Epix Delaware, Inc.	Synthesis of thienopyridinone compounds and related intermediates
US7598265B2 (en) *	2004-09-30	2009-10-06	Epix Delaware, Inc.	Compositions and methods for treating CNS disorders
CA2599925A1 (en) *	2005-03-14	2006-09-21	Merck & Co., Inc.	Cgrp receptor antagonists
ES2393326T3 (es)	2006-12-18	2012-12-20	Amgen, Inc	Compuestos basados en azaquinolona que presentan actividad inhibidora de prolil hidroxilasas, composiciones y usos de los mismos
ES2446418T3 (es)	2007-04-18	2014-03-07	Amgen, Inc	Derivados de indanona que inhiben la prolil hidroxilasa
EP2142509B1 (en)	2007-04-18	2013-12-04	Amgen, Inc	Quinolones and azaquinolones that inhibit prolyl hydroxylase
US8030346B2 (en)	2007-05-04	2011-10-04	Amgen Inc.	Heterocyclic quinolone derivatives that inhibit prolyl hydroxylase activity
WO2008137084A2 (en)	2007-05-04	2008-11-13	Amgen Inc.	Diazaquinolones that inhibit prolyl hydroxylase activity
EP2445877B1 (en)	2008-12-03	2014-07-23	Nanotherapeutics, Inc.	Bicyclic compounds and methods of making and using same
WO2016109706A1 (en) *	2014-12-31	2016-07-07	Ptc Therapeutics, Inc.	Fused polycyclic 2-pyridinone antibacterial compounds

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3903095A (en) *	1972-02-18	1975-09-02	Merck & Co Inc	Certain substituted-thieno{8 3,2-c{9 -pyridines
NO140499C (no) *	1973-07-23	1979-09-12	Takeda Chemical Industries Ltd	Analogifremgangsmaate til fremstilling av thienopyridinkarboksylsyrederivcater med terapeutisk aktivitet
IL87674A (en) *	1987-09-08	1993-08-18	Lilly Co Eli	Azabicycloalkyl esters and amides of heterocyclic acids, their preparation and pharmaceutical compositions containing them

1992
- 1992-03-04 US US07/847,670 patent/US5155115A/en not_active Expired - Fee Related
- 1992-03-05 DE DE69200290T patent/DE69200290T2/de not_active Expired - Fee Related
- 1992-03-05 EP EP92301901A patent/EP0503844B1/en not_active Expired - Lifetime
- 1992-03-05 AT AT92301901T patent/ATE109484T1/de active
- 1992-03-05 ES ES92301901T patent/ES2057959T3/es not_active Expired - Lifetime
- 1992-03-05 DK DK92301901.2T patent/DK0503844T3/da active
- 1992-03-05 JP JP04048446A patent/JP3117777B2/ja not_active Expired - Fee Related

Also Published As

Publication number	Publication date
JP3117777B2 (ja)	2000-12-18
ATE109484T1 (de)	1994-08-15
DE69200290T2 (de)	1995-02-16
EP0503844A1 (en)	1992-09-16
US5155115A (en)	1992-10-13
ES2057959T3 (es)	1994-10-16
DE69200290D1 (de)	1994-09-08
EP0503844B1 (en)	1994-08-03
JPH0565289A (ja)	1993-03-19

Publication	Publication Date	Title
ATE109484T1 (de)	1994-08-15	Thienopyridin -derivative und diese enthaltende arzneimittel.
DK0641767T3 (da)	1999-08-23	Cytotoksiske stilbenderivater og farmaceutisk præparat indeholdende disse derivater
DK0458636T3 (da)	1995-08-21	Antiemetiske og migræneundertrykkende heterocycliske forbindelser og farmaceutiske præparater indeholdende disse
DK0731085T3 (da)	2000-04-17	Stilbenderivater og farmaceutiske sammensætinger indeholdende disse
IL110151A0 (en)	1994-10-07	Amide and urea derivatives and pharmaceutical compositions containing the same
DK0580502T3 (da)	1999-05-31	3-(hydroxybenzylidenyl)-indolin-2-oner og farmaceutiske sammensætninger indeholdende disse
DK0835888T3 (da)	2000-09-25	En ikke-tværbundet anionbytterharpiks og farmaceutisk sammensætning indeholdende denne
ES2103027T3 (es)	1997-08-16	Derivados de tienopiridina y composiciones farmaceuticas que los contienen.
DK599785A (da)	1986-06-22	Blokpolyestere og detergentkompositioner indeholdende disse
IL114785A0 (en)	1995-11-27	Pyrrolocarbazoles their preparation and pharmaceutical compositions containing them
DK0474243T3 (da)	1998-12-07	1-methylcarbapenemderivater og fremgangsmåde til fremstilling deraf
ATE122348T1 (de)	1995-05-15	Antipsychotische 3-piperazinylbenzazolderivate.
IL102652A0 (en)	1993-01-14	Indole derivatives,their preparation and pharmaceutical compositions containing them
HU9503090D0 (en)	1995-12-28	Novel bisoxadiazolidine derivative
TW363052B (en)	1999-07-01	Anti-arrhythmic fluorine-containing benzoylguanidines, and preparation process and pharmaceutical composition thereof
DE69118064D1 (de)	1996-04-25	Diamino-s-Triazinonderivate und diese enthaltende selbstlöschende polymere Zusammensetzungen
EP0601191A4 (en)	1994-08-17	Novel tetracyclic compound.
NO893523D0 (no)	1989-09-01	Antihypertensive 3-piperidinyl-indazolderivater.
DE3781986D1 (de)	1992-11-05	Substituierte chinoxaline.
GR3020323T3 (en)	1996-09-30	P-di(2-chloroethyl)amino)phenylalanine derivatives process for their preparation and pharmaceutical compositions containing them.