DK0610317T3 - Inhibitorer af dipeptidyl-aminopeptidase type IV - Google Patents

Inhibitorer af dipeptidyl-aminopeptidase type IV

Info

Publication number
DK0610317T3
DK0610317T3 DK92922300T DK92922300T DK0610317T3 DK 0610317 T3 DK0610317 T3 DK 0610317T3 DK 92922300 T DK92922300 T DK 92922300T DK 92922300 T DK92922300 T DK 92922300T DK 0610317 T3 DK0610317 T3 DK 0610317T3
Authority
DK
Denmark
Prior art keywords
inhibitors
dipeptidyl aminopeptidase
aminopeptidase type
type
inhibiting
Prior art date
Application number
DK92922300T
Other languages
Danish (da)
English (en)
Inventor
William W Bachovchin
Andrew G Plaut
George R Flentke
Original Assignee
New England Medical Center Inc
Univ Tufts
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by New England Medical Center Inc, Univ Tufts filed Critical New England Medical Center Inc
Application granted granted Critical
Publication of DK0610317T3 publication Critical patent/DK0610317T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Immunology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Peptides Or Proteins (AREA)
DK92922300T 1991-10-22 1992-10-21 Inhibitorer af dipeptidyl-aminopeptidase type IV DK0610317T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US78155291A 1991-10-22 1991-10-22
PCT/US1992/009026 WO1993008259A2 (en) 1991-10-22 1992-10-21 Inhibitors of dipeptidyl-aminopeptidase type iv

Publications (1)

Publication Number Publication Date
DK0610317T3 true DK0610317T3 (da) 2001-02-19

Family

ID=25123110

Family Applications (1)

Application Number Title Priority Date Filing Date
DK92922300T DK0610317T3 (da) 1991-10-22 1992-10-21 Inhibitorer af dipeptidyl-aminopeptidase type IV

Country Status (9)

Country Link
EP (2) EP1050540B1 (de)
JP (1) JPH07504158A (de)
AT (2) ATE349461T1 (de)
CA (1) CA2121369C (de)
DE (2) DE69233671T2 (de)
DK (1) DK0610317T3 (de)
ES (1) ES2153831T3 (de)
GR (1) GR3035730T3 (de)
WO (1) WO1993008259A2 (de)

Families Citing this family (87)

* Cited by examiner, † Cited by third party
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EP0764151A2 (de) * 1994-06-10 1997-03-26 Universitaire Instelling Antwerpen Reinigung von serine-protease und dessen synthetischen inhibitoren
FR2733995B1 (fr) * 1995-05-09 1997-07-25 Inst Nat Sante Rech Med Inhibiteurs de l'inactivation de neuropeptides endogenes notamment la cholecystokinine, leurs procedes de preparation leur utilisation comme medicaments et procede de criblage de medicaments
DE19616486C5 (de) 1996-04-25 2016-06-30 Royalty Pharma Collection Trust Verfahren zur Senkung des Blutglukosespiegels in Säugern
US5965532A (en) * 1996-06-28 1999-10-12 Trustees Of Tufts College Multivalent compounds for crosslinking receptors and uses thereof
US6011155A (en) * 1996-11-07 2000-01-04 Novartis Ag N-(substituted glycyl)-2-cyanopyrrolidines, pharmaceutical compositions containing them and their use in inhibiting dipeptidyl peptidase-IV
US6100234A (en) * 1997-05-07 2000-08-08 Tufts University Treatment of HIV
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DE19834591A1 (de) 1998-07-31 2000-02-03 Probiodrug Ges Fuer Arzneim Verfahren zur Steigerung des Blutglukosespiegels in Säugern
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EP1852108A1 (de) 2006-05-04 2007-11-07 Boehringer Ingelheim Pharma GmbH & Co.KG Zusammensetzungen von DPP-IV-Inhibitoren
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Also Published As

Publication number Publication date
DE69233671T2 (de) 2007-10-18
ES2153831T3 (es) 2001-03-16
EP1050540B1 (de) 2006-12-27
CA2121369A1 (en) 1993-04-29
GR3035730T3 (en) 2001-07-31
HK1015611A1 (en) 1999-10-15
ATE349461T1 (de) 2007-01-15
CA2121369C (en) 2003-04-29
EP1050540A2 (de) 2000-11-08
EP1050540A3 (de) 2002-01-02
EP0610317B1 (de) 2001-01-31
WO1993008259A3 (en) 1994-08-18
DE69231674T2 (de) 2001-08-09
DE69233671D1 (de) 2007-02-08
WO1993008259A2 (en) 1993-04-29
DE69231674D1 (de) 2001-03-08
JPH07504158A (ja) 1995-05-11
ATE199016T1 (de) 2001-02-15
EP0610317A4 (de) 1996-12-04
EP0610317A1 (de) 1994-08-17

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