DK0617620T3 - Anvendelse af 5-HT4-modulatorer til fremstilling af et lægemiddel til behandling af blærelidelser - Google Patents

Anvendelse af 5-HT4-modulatorer til fremstilling af et lægemiddel til behandling af blærelidelser

Info

Publication number
DK0617620T3
DK0617620T3 DK93900327T DK93900327T DK0617620T3 DK 0617620 T3 DK0617620 T3 DK 0617620T3 DK 93900327 T DK93900327 T DK 93900327T DK 93900327 T DK93900327 T DK 93900327T DK 0617620 T3 DK0617620 T3 DK 0617620T3
Authority
DK
Denmark
Prior art keywords
treatment
modulators
medicament
manufacture
bladder
Prior art date
Application number
DK93900327T
Other languages
English (en)
Inventor
Gareth John Sanger
Kay Alison Wardle
Original Assignee
Smithkline Beecham Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB919127184A external-priority patent/GB9127184D0/en
Priority claimed from GB919127185A external-priority patent/GB9127185D0/en
Priority claimed from GB929219354A external-priority patent/GB9219354D0/en
Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc
Application granted granted Critical
Publication of DK0617620T3 publication Critical patent/DK0617620T3/da

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/235Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids having an aromatic ring attached to a carboxyl group
    • A61K31/24Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids having an aromatic ring attached to a carboxyl group having an amino or nitro group
    • A61K31/245Amino benzoic acid types, e.g. procaine, novocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Emergency Medicine (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Steroid Compounds (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Percussion Or Vibration Massage (AREA)
  • Infusion, Injection, And Reservoir Apparatuses (AREA)
DK93900327T 1991-12-21 1992-12-21 Anvendelse af 5-HT4-modulatorer til fremstilling af et lægemiddel til behandling af blærelidelser DK0617620T3 (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB919127184A GB9127184D0 (en) 1991-12-21 1991-12-21 Pharmaceuticals
GB919127185A GB9127185D0 (en) 1991-12-21 1991-12-21 Pharmaceuticals
GB929219354A GB9219354D0 (en) 1992-09-12 1992-09-12 Pharmaceuticals
PCT/GB1992/002376 WO1993012785A1 (en) 1991-12-21 1992-12-21 Use of 5-ht4 modulators for the manufacture of a medicament for the treatment of the bladder diseases

Publications (1)

Publication Number Publication Date
DK0617620T3 true DK0617620T3 (da) 1999-06-07

Family

ID=27265978

Family Applications (1)

Application Number Title Priority Date Filing Date
DK93900327T DK0617620T3 (da) 1991-12-21 1992-12-21 Anvendelse af 5-HT4-modulatorer til fremstilling af et lægemiddel til behandling af blærelidelser

Country Status (9)

Country Link
EP (1) EP0617620B1 (da)
JP (1) JPH07502528A (da)
AT (1) ATE170747T1 (da)
AU (1) AU671430B2 (da)
CA (1) CA2126354C (da)
DE (1) DE69226961T2 (da)
DK (1) DK0617620T3 (da)
ES (1) ES2121984T3 (da)
WO (1) WO1993012785A1 (da)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5998409A (en) * 1992-03-12 1999-12-07 Smithkline Beecham Plc Condensed indole derivatives as 5HT4 -receptor antagonists
US5852014A (en) * 1992-03-12 1998-12-22 Smithkline Beecham P.L.C. Condensed indole derivatives as 5HT4 -receptor antagonists
EP0664794A1 (en) * 1992-10-16 1995-08-02 Smithkline Beecham Plc N-alkylpiperidinyl-4-methyl carboxylic esters/amides of condensed ring systems as 5-ht4 receptor antagonists
TW344661B (en) * 1993-11-24 1998-11-11 Lilly Co Eli Pharmaceutical composition for treatment of incontinence
KR19990022096A (ko) * 1995-05-31 1999-03-25 쇼다 오사무 모노시클릭 아미노기를 갖는 인다졸 유도체
IL140118A0 (en) 1998-06-15 2002-02-10 Sepracor Inc Use of optically pure (+) norcisapride for treating apnea, bulimia and other disorders
HK1040059A1 (zh) * 1998-06-15 2002-05-24 塞普拉科有限公司 光学纯度(-)-降西沙必利对治疗呼吸暂停、贪食症和其它疾病的用途
US6353005B1 (en) 1999-03-02 2002-03-05 Sepracor, Inc. Method and compositions using (+) norcisapride in combination with proton pump inhibitors or H2 receptor antagonist
US6362202B1 (en) 1999-03-02 2002-03-26 Sepracor Inc. Methods and compositions using (−) norcisapride in combination with proton pump inhibitors or H2 receptor antagonists
TWI263496B (en) * 1999-12-10 2006-10-11 Novartis Ag Pharmaceutical combinations and their use in treating gastrointestinal disorders
EP1551394A1 (en) * 2002-08-14 2005-07-13 Janssen Pharmaceutica N.V. Treatment of lower urinary tract symptoms associated with overactive bladder in men and women

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2044854A1 (en) * 1990-07-19 1992-01-20 Hong-I Chen Method for preventing or treating urinary incontinence
GB9103862D0 (en) * 1991-02-25 1991-04-10 Glaxo Group Ltd Chemical compounds

Also Published As

Publication number Publication date
DE69226961D1 (de) 1998-10-15
AU671430B2 (en) 1996-08-29
CA2126354C (en) 2006-07-11
JPH07502528A (ja) 1995-03-16
EP0617620B1 (en) 1998-09-09
ATE170747T1 (de) 1998-09-15
WO1993012785A1 (en) 1993-07-08
EP0617620A1 (en) 1994-10-05
ES2121984T3 (es) 1998-12-16
AU3168393A (en) 1993-07-28
DE69226961T2 (de) 1999-04-29
CA2126354A1 (en) 1993-07-08

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