DK0641791T3 - Nye benzothiophenderivater - Google Patents

Nye benzothiophenderivater

Info

Publication number
DK0641791T3
DK0641791T3 DK92923415T DK92923415T DK0641791T3 DK 0641791 T3 DK0641791 T3 DK 0641791T3 DK 92923415 T DK92923415 T DK 92923415T DK 92923415 T DK92923415 T DK 92923415T DK 0641791 T3 DK0641791 T3 DK 0641791T3
Authority
DK
Denmark
Prior art keywords
substituted
lower alkyl
benzothiophene derivatives
new benzothiophene
benzothiophene
Prior art date
Application number
DK92923415T
Other languages
English (en)
Inventor
Shigehiro Takegawa
Shigeki Iwashita
Tomoyuki Saito
Naoyuki Koizumi
Tomoko Kawachi
Teruaki Matsui
Mamoru Mieda
Hiroo Takahashi
Kenyu Shibata
Original Assignee
Teikoku Hormone Mfg Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teikoku Hormone Mfg Co Ltd filed Critical Teikoku Hormone Mfg Co Ltd
Application granted granted Critical
Publication of DK0641791T3 publication Critical patent/DK0641791T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/32—Antioestrogens
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/56—Radicals substituted by oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Saccharide Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK92923415T 1991-11-15 1992-11-11 Nye benzothiophenderivater DK0641791T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP32666691A JP3157882B2 (ja) 1991-11-15 1991-11-15 新規なベンゾチオフエン誘導体
PCT/JP1992/001465 WO1993010113A1 (fr) 1991-11-15 1992-11-11 Nouveau derive de benzothiophene

Publications (1)

Publication Number Publication Date
DK0641791T3 true DK0641791T3 (da) 1998-09-23

Family

ID=18190312

Family Applications (1)

Application Number Title Priority Date Filing Date
DK92923415T DK0641791T3 (da) 1991-11-15 1992-11-11 Nye benzothiophenderivater

Country Status (13)

Country Link
US (1) US5472962A (da)
EP (1) EP0641791B1 (da)
JP (1) JP3157882B2 (da)
KR (1) KR100220268B1 (da)
AT (1) ATE162788T1 (da)
AU (1) AU665588B2 (da)
CA (1) CA2123514C (da)
DE (1) DE69224308T2 (da)
DK (1) DK0641791T3 (da)
ES (1) ES2111652T3 (da)
GR (1) GR3026471T3 (da)
SG (1) SG47113A1 (da)
WO (1) WO1993010113A1 (da)

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EP0641791B1 (en) 1998-01-28
JP3157882B2 (ja) 2001-04-16
US5472962A (en) 1995-12-05
JPH05140148A (ja) 1993-06-08
DE69224308T2 (de) 1998-05-20
CA2123514C (en) 2003-07-29
SG47113A1 (en) 1998-03-20
GR3026471T3 (en) 1998-06-30
WO1993010113A1 (fr) 1993-05-27
AU2927692A (en) 1993-06-15
AU665588B2 (en) 1996-01-11
ATE162788T1 (de) 1998-02-15
EP0641791A1 (en) 1995-03-08
KR100220268B1 (ko) 1999-09-15
CA2123514A1 (en) 1993-05-27
EP0641791A4 (en) 1994-11-22
DE69224308D1 (de) 1998-03-05
ES2111652T3 (es) 1998-03-16

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