DK0695751T3 - Middel indvirkende på det centrale nervesystem, fremgangsmåde til dets fremstilling og farmaceutiske præparater indeholdende det. - Google Patents

Middel indvirkende på det centrale nervesystem, fremgangsmåde til dets fremstilling og farmaceutiske præparater indeholdende det.

Info

Publication number
DK0695751T3
DK0695751T3 DK95907014.5T DK95907014T DK0695751T3 DK 0695751 T3 DK0695751 T3 DK 0695751T3 DK 95907014 T DK95907014 T DK 95907014T DK 0695751 T3 DK0695751 T3 DK 0695751T3
Authority
DK
Denmark
Prior art keywords
preparation
nervous system
central nervous
pharmaceutical preparations
preparations containing
Prior art date
Application number
DK95907014.5T
Other languages
English (en)
Inventor
Ges Jose Maria Caldero
Clotet Joan Huguet
Olondriz Francisco Marquillas
Barjoan Pere Dalmases
Rovira Anna Bosch
Acin Joan Roca
Nieto Juan Carlos Del Castillo
Original Assignee
Vita Invest Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vita Invest Sa filed Critical Vita Invest Sa
Application granted granted Critical
Publication of DK0695751T3 publication Critical patent/DK0695751T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK95907014.5T 1994-02-24 1995-02-02 Middel indvirkende på det centrale nervesystem, fremgangsmåde til dets fremstilling og farmaceutiske præparater indeholdende det. DK0695751T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ES09400362A ES2085234B1 (es) 1994-02-24 1994-02-24 Agente activo sobre el sistema nervioso central, procedimiento para su preparacion y composiciones farmaceuticas que lo contienen.

Publications (1)

Publication Number Publication Date
DK0695751T3 true DK0695751T3 (da) 1997-09-29

Family

ID=8285331

Family Applications (1)

Application Number Title Priority Date Filing Date
DK95907014.5T DK0695751T3 (da) 1994-02-24 1995-02-02 Middel indvirkende på det centrale nervesystem, fremgangsmåde til dets fremstilling og farmaceutiske præparater indeholdende det.

Country Status (12)

Country Link
US (1) US5658916A (da)
EP (1) EP0695751B1 (da)
JP (1) JP2848707B2 (da)
AT (1) ATE150752T1 (da)
AU (1) AU677146B2 (da)
CA (1) CA2160717A1 (da)
DE (1) DE69500198T2 (da)
DK (1) DK0695751T3 (da)
ES (2) ES2085234B1 (da)
GR (1) GR3023800T3 (da)
RU (1) RU2126005C1 (da)
WO (1) WO1995023144A1 (da)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2138908B1 (es) * 1997-08-14 2000-09-16 Vita Invest Sa Polimorfos de la 3-(2-(4-(6-fluorobenzo(d)isoxazol-3-il) 3,6. dihidro-2h-piridin-1-il)-etil)-2-metil-6,7,8,9-tetrahidropirido (1,2-a) pirimidin-4-ona y procedimientos para su obtencion.
ES2141671B1 (es) * 1997-12-26 2001-01-01 Vita Invest Sa Compuesto pirimidinico activo sobre el sistema nervioso central, procedimiento para su preparacion y composiciones farmaceuticas que lo contienen.
HU227118B1 (en) * 2001-11-13 2010-07-28 Egis Gyogyszergyar Nyilvanosan Process for the preparation of 3-{2-[4-(6-fluoro-1,2-benzizoxazol-3-yl)-1-piperidinyl]-ethyl}-6,7,8,9-tetrahydro-2-methyl-4h-pyrido[1,2-a]pyrimidin-4-one
RU2281085C2 (ru) * 2004-05-25 2006-08-10 Закрытое акционерное общество "Мастерлек" Антидепрессивные лекарственные средства для парентерального применения на основе сульфонатных солей пирлиндола
US8314110B2 (en) * 2007-04-19 2012-11-20 Youxin Li Compounds for treating mental disorders, and preparation and uses thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4342870A (en) * 1980-03-28 1982-08-03 Janssen Pharmaceutica N.V. Novel 3-(1-piperidinylalkyl)-4H-pyrido[1,2-a]pyrimidin-4-one derivatives
US4485107A (en) * 1982-11-01 1984-11-27 Janssen Pharmaceutica N.V. [[Bis(aryl)methylene]-1-piperidinyl]alkyl-pyrimidinones
KR910000165B1 (ko) * 1985-03-27 1991-01-21 쟈안센 파아마슈우티카 엔. 부이. 1,2-벤즈이소옥사졸-3-일과 1,2-벤즈이소티아졸-3-일 유도체의 제조방법
US4804663A (en) * 1985-03-27 1989-02-14 Janssen Pharmaceutica N.V. 3-piperidinyl-substituted 1,2-benzisoxazoles and 1,2-benzisothiazoles
US5158952A (en) * 1988-11-07 1992-10-27 Janssen Pharmaceutica N.V. 3-[2-[4-(6-fluoro-1,2-benzisoxozol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9 tetrahydro-9-hydroxy-2-methyl-4H-pyrido [1,2-a]pyrimidin-4-one, compositions and method of use
CA2000786C (en) * 1988-11-07 1999-01-26 Janssen Pharmaceutica, Naamloze Vennootschap 3-piperidinyl-1,2-benzisoxazoles
GB9008850D0 (en) * 1990-04-19 1990-06-13 Janssen Pharmaceutica Nv Novel 2,9-disubstituted-4h-pyridol(1,2-a)pyrimidin-4-ones

Also Published As

Publication number Publication date
RU2126005C1 (ru) 1999-02-10
DE69500198D1 (de) 1997-04-30
EP0695751A1 (en) 1996-02-07
CA2160717A1 (en) 1995-08-31
WO1995023144A1 (es) 1995-08-31
GR3023800T3 (en) 1997-09-30
JP2848707B2 (ja) 1999-01-20
EP0695751B1 (en) 1997-03-26
ES2100768T3 (es) 1997-06-16
ES2085234B1 (es) 1997-01-16
JPH08509505A (ja) 1996-10-08
AU677146B2 (en) 1997-04-10
AU1538195A (en) 1995-09-11
US5658916A (en) 1997-08-19
ES2085234A1 (es) 1996-05-16
DE69500198T2 (de) 1997-10-16
ATE150752T1 (de) 1997-04-15

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